Fernando Albericio is Research Professor at the University of KwaZulu-Natal (UKZN) in Durban, South Africa & Honorary Full Professor of Organic Chemistry at the University of Barcelona.  

He was Inaugural Rector of Yachay Tech (Ecuador), which is called to be the first Latinoamerican university based into the Innovation, and Founder and General Director of the Barcelona Science Park (PCB).

He has published over 900 papers, filled more than 60 patents, and has co-authored four books. He is also Editor-in-Chief of several scientific journals and acted in the editorial board of several others.

His major research interests cover practically all aspects of peptide synthesis (new reactions, building blocks, coupling reagents, solid phase supports, protecting groups, and linkers) and combinatorial chemistry methodologies, as well as the synthesis of peptides and small molecules with therapeutic activities (cancer and infectious diseases).  Furthermore, his group is also involved in developing new systems for drug delivery and strategies for diagnostics as well.

Lastly, he was working in the development of multicomponent platforms for the preparation of bioconjugates, involving peptides, foldamers, oligonucleotides, and monoclonal antibodies, among others.  Special attention has been paid to the linkers responsible for binding the molecules.  Those are based in “click” chemistry, thiol chemistry, Diels-Alder, and Pd chemistry.   Finally, his group is working in the introduction of the green concept in solid-phase synthesis.

He is deeply involved in the creation of the Entrepreneurial University in Spain, in Latinoamerica, and, presently, in South Africa. During his tenure at the PCB, he catalyzed the creation of almost 100 start-up companies.

He was the founder of the “Emprendia” Network-Santander Bank, which was the first Latinoamerican University Network for the Incubation of Companies with the purpose of creating a Latinoamerican business network upon the R&D results from the universities.  

Presently, he is working in the development of BioDurban at UKZN.

• Peptides and Amino Acids

• Ernest Giralt, M. Dolors Ludevid, Fernando Albericio, and Mariona Bassedas. Acid-base properties of 4-nitro-L-histidine and related compounds. Bioorg. Chem.8, 59-67 (1979).
• Ernest Giralt, Fernando Albericio, David Andreu, Ramon Eritja, Pablo Martin, and Enrique Pedroso. Synthesis of Nbb-resin, a new polymer support for the solid-phase synthesis of protected peptides. An. Quím. 77, C,120-125 (1980).
• Ernest Giralt and Fernando Albericio. Free amino content of benzhydrylamine resins used as solid supports for peptide synthesis. An. Quím.77, C, 134-137 (1980).
• Ernest Giralt, David Andreu, Fernando Albericio, and Enrique Pedroso. Synthesis and properties of Pab- and Nbb-resins. Two new benzhydrylamine resin-derived solid supports for peptide synthesis. In Peptides 1980. Proceedings of the Sixteenth European Peptide Symposium (K. Brunfeldt, ed.), Scriptor, Copenhagen, Denmark, 1981, pp. 315-320.
• Enrique Pedroso, Fernando Albericio, Anna Grandas, Ernest Giralt, Jurphaas van Rietschoten, and Claude Granier. Two new methods for the solid-phase synthesis of protected peptides. Synthesis of apamin and LHRH protected fragments. In Peptides 1980. Proceedings of the Sixteenth European Peptide Symposium (K. Brunfeldt, ed.), Scriptor, Copenhagen, Denmark, 1981, pp. 334-338.
• Ernest Giralt, Fernando Albericio, Enrique Pedroso, Claude Granier, and Jurphaas van Rietschoten. Convergent solid-phase peptide synthesis. II. Synthesis of the 1-6 apamin protected segment on a Nbb-resin. Synthesis of apamin. Tetrahedron38, 1193-1201 (1982).
• Marie Tessier, Fernando Albericio, Enrique Pedroso, Anna Grandas, Ramon Eritja, Ernest Giralt, Claude Granier, and Jurphaas van Rietschoten. Amino acids condensations in the preparation of N-9-fluorenylmethyloxycarbonylamino acids with 9-fluorenylmethylchloro-formate. Int. J. Pept. Protein Res. 22, 125-128 (1983).
• Fernando Albericio, Claude Granier, Catherine Labbé-Jullié, Michael Seagar, Francois Couraud, and Jurphaas van Rietschoten. Solid-phase synthesis and HPLC purification of the protected 1-12 sequence of apamin for rapid synthesis of apamin analogues differing in the C-terminal region. Tetrahedron40, 4313-4326 (1984).
• Fernando Albericio and George Barany. Application of N,N-dimethylformamide dineopentyl acetal for efficient anchoring of Nα-9-fluorenylmethyloxycarbonyl amino acids as p-alkoxybenzyl esters in solid-phase peptide synthesis. Int. J. Pept. Protein Res. 23, 342-349 (1984).
• Fernando Albericio, Claude Granier, Catherine Labbé-Juillé, and Jurphaas van Rietschoten. Solid-phase segment synthesis and assembling. In Peptides: Structure and Function. Proceedings of the Eight American Peptide Symposium (V.J. Hruby and D.H. Rich, eds.), Pierce Chemical Company, Rockford, Illinois, 1984, pp. 107-110.
• Ernest Giralt, Ramon Eritja, Anna Grandas, Enrique Pedroso, Marie Tessier, Fernando Albericio, Claude Granier, and Jurphaas van Rietschoten. Solid-phase synthesis of two protected segments from the C-terminal region of Androctonus australis Hector toxin II. In Peptides 1984. Proceedings of the Eighteenth European Peptide Symposium (U. Ragnarsson, ed.), Alqvist and Wiksell, Stockolm, Sweden, 1984, pp. 173-176.
• Fernando Albericio, Urszula Slomczynska, Daniel G. Mullen, Shmuel Zalipsky, and George Barany. Orthogonal solid-phase peptide synthesis with Nα-dithiasuccinoyl (Dts) amino acids and N-(isopropyldithio)carbonylproline. In Peptides 1984. Proceedings of the Eighteenth European Peptide Symposium (U. Ragnarsson, ed.), Alqvist and Wiksell, Stockolm, Sweden, 1984, pp. 181-184.
• Fernando Albericio and George Barany. Improved approach for anchoring N-9-fluorenylmethyolxycarbonylamino acids as p-alkoxybenzyl esters in solid-phase peptide synthesis. Int. J. Peptide Protein Res. 26, 92-97 (1985).
• George Barany and Fernando Albericio. A three-dimensional orthogonal protection scheme for solid-phase peptide synthesis under mild conditions. J. Am. Chem. Soc. 107, 4936-4942 (1985).
• Shmuel Zalipsky, Fernando Albericio, and George Barany. Preparation and use of an aminoethyl polyethylene glycol-crosslinked polystyrene graft resin support for solid-phase peptide synthesis. In Peptides: Structure and Function. Proceedings of the Ninth American Peptide Symposium (C.M. Deber, V.J. Hruby, and K.D. Kopple, eds.), Pierce Chemical Co., Rockford, Illinois, 1985, pp. 257-260.
• Fernando Albericio, Rosa Ripoll, Enrique Pedroso, and Ernest Giralt. Properties of bromomethyl-Nbb-resin: Application to the synthesis of protected peptides and oligoamides, as demonstrated by synthesis of Boc-(β-Ala)4-OH. Afinidad42, 491-496 (1985).
• Fernando Albericio, Urszula Slomczynska, and George Barany. New handles for the synthesis of C-terminal peptide amides. In Forum Peptides: Proceedings of the 1st International Forum Peptides (B. Castro and J. Martínez, eds.), Les Impressions Dohr, Nancy, France, 1986, pp. 1-5.
• Jurphaas van Rietschoten, Fernando Albericio, Marie Tessier-Rochat, Claude Granier, Anna Grandas, Ramon Eritja, Enrique Pedroso, and Ernest Giralt. Solid phase synthesis of two segments: sequence 18-31 and 53-59 of the toxin II of Androctonus australis Hector. In Forum Peptides: Proceedings of the 1st International Forum Peptides (B. Castro and J. Martínez, eds.), Les Impressions Dohr, Nancy, France, 1986, pp. 357-360.
• Mariano Ruiz-Gayo, Fernando Albericio, Enrique Pedroso, and Ernest Giralt.(S)-9-Fluorenylmethyl-L-cysteine, a useful HF-stable derivative for peptide synthesis. J. Chem. Soc., Chem. Commun. pp. 1501-1502 (1986).
• Perry B. Hackett, Robert B. Petersen, Charles H. Hensel, Fernando Albericio, Fernando Albericio, Samuel I. Gunderson, Ann C. Palmenberg, and George Barany. Synthesis in vitro of a seven amino acid peptide encoded in the leader RNA of rous sarcoma virus. J. Mol. Biol. 190, 45-57 (1986).
• Jurphaas van Rietschoten, Jean M. Sabatier, Marie Tessier, Claude Granier, Enrique Pedroso, Anna Grandas, Fernando Albericio, Ramon Eritja, Ernesto Nicolás, Jaume Josa, and Ernest Giralt. Convergent solid-phase peptide synthesis: recent progresses. Protides of the Biol. Fluids34, 23-26 (1986).
• Fernando Albericio, Anna Porta, Enrique Pedroso, and Ernest Giralt. Solid phase coupling of protected peptide segments. Influence of the polymer support. In Peptides 1986. Proceedings to the Nineteenth European Peptide Symposium (D. Theodoropoulos, ed.) Walter der Gruyter, Berlin, 1987, pp. 167-170.
• Fernando Albericio and George Barany. Mild, orthogonal solid-phase peptide synthesis: use of N-dithiasuccinoyl (Dts) amino acids and N-(isopropyldithio)carbonylproline, together with p-alkoxybenzyl ester anchoring linkages. Int. J. Peptide Protein Res. 30, 177-205 (1987).
• Fernando Albericio and George Barany. An acid-labile anchoring linkage for solid-phase synthesis of C-terminal peptide amides under mild conditions. Int. J. Peptide Protein Res.30, 206-216 (1987).
• Shmuel Zalipsky, Fernando Albericio, Urszula Slomczynska, and George Barany. A convenient general method for synthesis of Nα- or Nω-dithiasuccinoyl (Dts) amino acids and dipeptides: application of polyethylene glycol as a carrier for functional purification. Int. J. Peptide Protein Res. 30, 740-783 (1987).
• Ramon Eritja, J. Paige Ziehler-Martin, Peter A. Walker, Terry D. Lee, Kassu Legesse, Fernando Albericio, and Bruce E. Kaplan. On the use of the S-t-butyl-sulphenyl group for protection of cysteine in solid-phase peptide synthesis using Fmoc-amino acids.Tetrahedron 43, 2675-2680 (1987).
• Fernando Albericio, Ernesto Nicolás, Jaume Josa, Anna Grandas, Enrique Pedroso, Ernest Giralt, Claude Granier, and Jurphaas van Rietschoten. Convergent solid phase peptide synthesis V. Synthesis of the 1-4, 32-34, and 53-59 protected segments of the toxin II of Androctonus australis Hector. Tetrahedron 43, 5961-5971 (1987).
• Jean M. Sabatier, Marie Tessier-Rochat, Claude Granier, Jurphaas van Rietschoten, Enrique Pedroso, Anna Grandas, Fernando Albericio, and Ernest Giralt. Convergent solid phase synthesis VI. Synthesis by the Fmoc procedure with a modified protocol of two protected segments, sequence 5-17 and 18-31 of the neurotoxin II of the scorpion Androctonus australis Hector. Tetrahedron43, 5973-5980 (1987).
• Fernando Albericio, Anna Grandas, Anna Porta, Enrique Pedroso, and Ernest Giralt. One-pot synthesis of S-acetamidomethyl-N-fluorenylmethoxycarbonyl-L-cysteine (Fmoc-Cys(Acm)-OH). Synthesis 271-272 (1987).
• Josep Rizo, Fernando Albericio, Guillermo Romero, Carlos García-Echeverría, Josep Claret, Carlos Muller, Ernest Giralt, and Enrique Pedroso. Use of polar picolyl protecting groups in peptide synthesis. J. Org. Chem. 53, 5836-5839 (1988).
• Fernando Albericio, Nancy Kneib-Cordonier, Lajos Gera, Robert P.Hammer, Derek Hudson, and George Barany. Solid-phase synthesis of C-terminal pepide amides under mild conditions. In Peptides - Chemistry and Biology: Proceedings of the Tenth American Peptide Symposium (G.R. Marshall, ed.), Escom Science Publishers, Leiden, The Netherlands, 1988, pp. 159-161.
• Virginia Stiefel, Lluis Perez-Grau, Fernando Albericio, Ernest Giralt, Luis Ruiz-Avila, M. Dolors Ludevid, and Pere Puigdomènech. Molecular cloning of cDNAs encoding a putative cell wall protein from Zea mays and immunological identification of related polypeptides. Plant Molecular Biology 11, 483-493 (1988).
• Jurphaas van Rietschoten, Jean M. Sabatier, Pierre Paroutaud, Fernando Albericio, Anna Grandas, Enrique Pedroso, and Ernest Giralt. Solid phase segment coupling: quality control by automated Edman degradation of peptidyl-resin. In Second Forum on Peptides (A. Aubry, M. Marraud, and B. Vitoux, eds.), Colloque INSERM/John Libbey Eurotext Ltd., Paris, 1989, vol 174, pp. 215-219.
• Mariano Ruiz-Gayo, Fernando Albericio, Miquel Pons, Enrique Pedroso, and Ernest Giralt. Synthesis of antiparallel and parallel dimers of bis-cysteine peptides. In Second Forum on Peptides (A. Aubry, M. Marraud, and B. Vitoux, eds.), Colloque INSERM/John Libbey Eurotext Ltd., Paris, 1989, vol 174, pp. 233-237.
• Anna Grandas, Fernando Albericio, Enrique Pedroso, Ernest Giralt, Jean M. Sabatier, and Jurphaas van Rietschoten. Coupling of peptide segments in convergent solid-phase peptide synthesis. In Peptide 1988: Proceedings of the Twenty European Peptide Symposium (G. Jung and E. Bayer, eds.), Walter der Gruyter, Berli, 1989, pp. 160-162.
• Fernando Albericio, Miquel Pons, Enrique Pedroso, and Ernest Giralt. Comparative study of supports for solid-phase coupling of protected-peptide segments. J. Org. Chem. 54, 360-366 (1989).
• Fernando Albericio, David Andreu, Ernest Giralt, Carles Navalpotro, Enrique Pedroso, Berta Ponsati, and Mariano Ruiz-Gayo. Use of the Npys thiol protection in solid phase peptide synthesis. Application to direct peptide-protein conjugation through cysteine residues. Int. J. Peptide Protein Res. 34, 124-128 (1989).
• MarionaBassedas, Fernando Albericio, and Francisco López-Calahorra. Quantitative monitoring of carboxyl groups in polymers. Anal. Chim. Acta219, 161-163 (1989).
• Fernando Albericio, Mariano Ruiz-Gayo, Enrique Pedroso, and Ernest Giralt. Use of polystyrene-1%-divinylbenzene and Kel-F-g-styrene for the simultaneous synthesis of peptides. Reactive Polym. 10, 259-268 (1989).
• Carlos García-Echeverría, Fernando Albericio, Miquel Pons, George Barany, and Ernest Giralt. Convenient synthesis of a cyclic peptide disulfide: a type II β-turn structural model. Tetrahedron Lett. 30, 2441-2444 (1989).
• Anna Grandas, Fernando Albericio, Jaume Josa, Ernest Giralt, Enrique Pedroso, Jean M. Sabatier, and Jurphaas van Rietschoten. Convergent solid phase peptide synthesis VII. Good yields in the coupling of protected segments on a solid support. Tetrahedron45, 4637-4648 (1989).
• Mariano Ruiz-Gayo, Fernando Albericio, Miriam Royo, Carlos García Echeverría, Enrique Pedroso, Miquel Pons, and Ernest Giralt. A convenient procedure for synthesis of cystine peptides via iodine oxidation of S-acetamidomethyl-cysteine peptides. An. Quím. 85, C, 116-118 (1989).
• Fernando Albericio, Nancy Kneib-Cordonier, Sara Biancalana, Lajos Gera, R. Irene Masada, Derek Hudson, and George Barany. Preparation and application of the 5-(4-(9-fluorenylmethyloxycarbonyl)-aminomethyl-3,5-dimethoxyphenoxy)-valeric acid (PAL) handle for the solid-phase synthesis of C-terminal peptide amides under mild conditions. J.Org. Chem. 55, 3730-3743 (1990).
• Fernando Albericio, Ernesto Nicolás, Josep Rizo, Mariano Ruiz-Gayo, Enrique Pedroso, and Ernest Giralt. Convenient synthesis of fluorenylmethyl-based side chain derivatives of glutamic and aspartic acids, lysine, and cysteine. Synthesis pp. 119-122 (1990).
• Carlos García-Echevarría, M. Antònia Molins, Fernando Albericio, Miquel Pons, and Ernest Giralt. Application of acetamidomethyl and 9-fluorenylmethyl groups for efficient side protection of penicillamine in solid-phase peptide synthesis. Int. J. Peptide Protein Res.35, 434-440 (1990).
• Fernando Albericio, Robert van Abel, and George Barany. Solid-phase synthesis of peptides with C-terminal asparagine or glutamine. Int. J. Peptide Protein Res.35, 284-286 (1990) .
• Nancy Kneib-Cordonier, Fernando Albericio, and George Barany. Orthogonal solid phase-peptide synthesis of human gastrin-I under mild conditions. Int. J. Peptide Protein Res. 35, 527-538 (1990).
• Robert P. Hammer, Fernando Albericio, Lajos Gera, and George Barany. Practical approach to solid-phase synthesis of C-terminal peptide amides under mild conditions based on a photolysable anchoring linkage. Int. J. Peptide Protein Res.36, 31-45 (1990).
• Nancy Kneib-Cordonier, Fernando Albericio, and George Barany. Orthogonal solid-phase synthesis of human gastrin-I under mild conditions. In Peptides - Chemistry and Biology: Proceedings of the Eleventh American Peptide Synposium (J. Rivier and G.R. Marshall, eds.), Escom, Science Publishers, Leiden, The Netherlands, 1990, pp. 895-897.
• Fernando Albericio, Josep Rizo, Ernesto Nicolás, Mariano Ruiz-Gayo, Francisco Cárdenas, Cristina Carreño, David Andreu, Enrique Pedroso, and Ernest Giralt. Fluorenylmethyl-based side chain protecting groups: towards a new strategy of peptide synthesis. In Peptides - Chemistry and Biology: Proceedings of the Eleventh American Peptide Synposium (J. Rivier and G.R. Marshall, eds.), Escom, Science Publishers, Leiden, The Netherlands, 1990, pp. 923-924.
• Carlos García-Echeverría, M. Antònia Molins, Robert P. Hammer, Fernando Albericio, Miquel Pons, George Barany, and Ernest Giralt. Cyclization of disulfide-containing peptides in solid-phase synthesis. In Peptides - Chemistry and Biology: Proceedings of the Eleventh American Peptide Synposium (J. Rivier and G.R. Marshall, eds.), Escom, Science Publishers, Leiden, The Netherlands, 1990, pp. 996-998.
• Ernest Giralt, Fernando Albericio, Francesc Bardella, Ramón Eritja, Miguel Feliz, Enrique Pedroso, Miquel Pons, and Josep Rizo. Gel-phase NMR spectroscopy as a useful tool in solid-phase synthesis. In Innovation and Perspectives in Solid-Phase Peptide Synthesis (R. Epton, ed.), SPPC (UK) Ltd, Birmingham, 1990, pp. 111-120.
• Carlos García-Echeverría, M. Antònia Molins, Fernando Albericio, Miquel Pons, and Ernest Giralt. Use of S-acetamidomethyl and S-9-fluorenylmethyl-penicillamine in solid-phase peptide synthesis. In "Innovation and Perspectives in Solid-Phase Peptide Synthesis" (R. Epton, ed.), SPPC (UK) Ltd, Birmingham, 1990, pp. 481-486.
• Eduard Bardají, Josep L. Torres, Pere Clapés, Fernando Albericio, George Barany, and Gregorio Valencia. Solid-phase synthesis of glicopeptide amides under mild conditions: morphiceptin analogues. Angew. Chem, In. Ed. Engl.29, 291-292 (1990); Angew. Chem. 102, 311-313.
• Xavier Jorba, Fernando Albericio, Anna Grandas, William Bannwarth, and Ernest Giralt. Arenesulphonyltriazolides as condensing reagents in solid phase peptide synthesis. Tetrahedron Lett. 31, 1915-1918 (1990)
• Berta Ponsati, Mariano Ruiz-Gayo, Ernest Giralt, Fernando Albericio, and David Andreu. Solid-phase-mediated peptide heterodisulfide formation. J. Am. Chem. Soc. 112, 5345-5347 (1990).
• Beatriz G. de la Torre, Josep L. Torres, Eduard Bardají, Pere Clapés, Núria Xaus, Xavier Jorba, Silvia Calvet, Fernando Albericio, and Gregorio Valencia. Improved method for the synthesis of O-glycosylated Fmoc-amino acids to be used in solid-phase glycopeptide synthesis. J. Chem. Soc., Chem, Commun. pp. 965-967 (1990).
• Margarida Gairí, Paul Lloyd-Williams, Fernando Albericio, and Ernest Giralt. Use of BOP reagent for the suppression of diketopiperazine formation in Boc/Bzl solid-phase peptide synthesis. Tetrahedron Lett. 31, 7363-7366 (1990).
• Fernando Albericio, Jordi Robles, Dolors Fernández-Forner, Yolanda Palom, Carles Celma, Enrique Pedroso, Ernest Giralt, and Ramón Eritja. NPE-resin, a new approach to the solid-phase synthesis of protected and oligonucleotides. In Peptides 1990. Proceedings of the Twenty-First European Peptide Symposium (E. Giralt and D. Andreu, eds.), Escom, Science Publishers, Leiden, The Netherlands, 1991, pp. 134-136.
• George Barany and Fernando Albericio. Mild orthogonal solid-phase synthesis. In Peptides 1990: Proceedings of the Twenty-First European Peptide Symposium (E. Giralt and D. Andreu, eds.), Escom, Science Publishers, Leiden, The Netherlands, 1991, pp. 139-142.
• Paul Lloyd-Williams, Margarida Gairí, Francisco Cárdenas, Fernando Albericio, and Ernest Giralt. Recent results in convergent solid-phase peptide synthesis. In Peptides 1990: Proceedings of the Twenty-First European Peptide Symposium (E. Giralt and D. Andreu, eds.), Escom, Science Publishers, Leiden, The Netherlands, 1991, pp. 146-148.
• Beatriz G. de la Torre, Josep L. Torres, Eduard Bardají, Pere Clapés, Fernando Albericio, and Gregorio Valencia. Solid-phase synthesis of new glycosyl enkephalinamides. In Peptides 1990: Proceedings of the Twenty-First European Peptide Symposium (E. Giralt and D. Andreu, eds.), Escom, Science Publishers, Leiden, The Netherlands, 1991, pp. 416-417.
• Fernando Albericio, Carlos García-Echeverría, Ernest Giralt, Juan J. Pérez, Miquel Pons, Miriam Royo, and Mariano Ruiz-Gayo. Effect of disulfide bonds in the conformation of cyclic dimer peptides. In Peptides 1990: Proceedings of the Twenty-First European Peptide Symposium (E. Giralt and D. Andreu, eds.), Escom, Science Publishers, Leiden, The Netherlands, 1991, pp. 535-537.
• Paul Lloyd-Williams, Fernando Albericio, and Ernest Giralt. Convergent solid-phase peptide synthesis. VIII. Synthesis, using a photolabile resin, and purification of a methionine-containing protected peptide. Int. J. Peptide Protein Res. 37, 58-60 (1991).
• Fernando Albericio, Robert P. Hammer, Carlos García-Echevarría, M. Antònia Molins, Jane L. Chang, Mark C. Munson, Miquel Pons, Ernest Giralt, and George Barany. Cyclization of disulfide-containing peptides in solid-phase synthesis. Int. J. Peptide Protein Res. 37, 402-413 (1991).
• Fernando Albericio and George Barany. Hypersensitive acid-labile (HAL) tris(alkoxy)-benzyl ester anchoring for solid-phase synthesis of protected peptide segments. Tetrahedron Lett. 32, 1015-1018 (1991).
• Ramon Eritja, Jordi Robles, Dolors Fernández-Forner, Fernando Albericio, Ernest Giralt, and Enrique Pedroso. NPE-resin, a new approach to the solid-phase synthesis of protected peptides and oligonucleotides. I: Synthesis of the supports and their application to oligonucleotide synthesis. Tetrahedron Lett. 32, 1511-1514 (1991).
• Fernando Albericio, Ernest Giralt, and Ramon Eritja. NPE-resin, a new approach to the solid-phase synthesis of protected peptides and oligonucleotides. II. Synthesis of protected peptides. Tetrahedron Lett. 32, 1515-1518 (1991).
• Catherine Labbé-Juillé, Claude Granier, Fernando Albericio, M. Léria Defendini, Brigitte Ceard, Hervé Rochat, and Jurphaas van Rietschoten. Binding and toxicity of apamin. Characterization of the active site. Eur. J. Biochem. 196, 639-645 (1991).
• Ramon Eritja, Anna Pons, Mónica Escarceller, Ernest Giralt, and Fernando Albericio. Synthesis of defined peptide-oligonucleotide hybrids containing a nuclear transport signal sequence. Tetrahedron47, 4113-4120 (1991).
• Eduard Bardají, Josep L. Torres, Pere Clapés, Fernando Albericio, George Barany, Raquel E. Rodríguez, María P. Sacristán, and Gregorio Valencia. Synthesis and biological activity of O-glycosylated morphiceptin analogues. J. Chem. Soc., Perkin I pp. 1755-1759. (1991).
• George Barany and Fernando Albericio. Peptide synthesis for biotechnology in the 1990's. In Biotechnology International1990 (K. North, ed.), Century Press Ltd., London, England, invited review article, 1991, pp. 155-163.
• George Barany and Fernando Albericio. Peptide synthesis for biotechnology in the 1990's. In Biotechnology International1991 (K. North, ed.), Century Press Ltd., London, England, invited review article, 1991, pp. 309-315 (revised and updated version).
• Paul Lloyd-Williams, Gemma Jou, Fernando Albericio, and Ernest Giralt. Solid-phase synthesis of peptides using allylic anchoring groups. An investigation of their palladium-catalysed cleavage. Tetrahedron Lett. 32, 4207-4210 (1991).
• Teresa Royo, José Ayté, Fernando Albericio, Ernest Giralt, Diego Haro, and Fausto G. Hegardt. Diurnal rhythm of rat liver cytosolic 3-hydroxy-3-methylglutaryl-CoA synthase. Biochem. J.280, 61-64 (1991).
• Paul Lloyd-Williams, Margarida Gairí, Fernando Albericio, and Ernest Giralt. Convergent solid-phase peptide synthesis X. Synthesis and purification of protected peptide fragments using the photolabile Nbb-resin. Tetrahedron47, 9867-9880 (1991).
• Urszula Slomczynska, Fernando Albericio, Francisco Cárdenas, and Ernest Giralt. Studies on the enzimatic coupling of peptide segments on the solid support. Biochem. Biochim. Acta10/11, 67-73 (1991).
• Carles Celma, Fernando Albericio, Enrique Pedroso, and Ernest Giralt. Convergent solid-phase peptide synthesis IX. Application to the synthesis of peptides with repetitive sequences. Peptide Res.5, 62-71 (1992).
• Roger J. Botems, Peter Heyges, Susan L. Botems, Fernando Albericio, and George Barany. Synthesis and applications of XAL, a new acid-labile handle for solid-phase synthesis of peptide amides. In Peptides - Chemistry and Biology: Proceedings of the Twelfth American Peptide Synposium (J. A. Smith and J. Rivier, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 601-602 (1992).
• George Barany, Fernando Albericio, Sara Biancalana, Susan L. Bontems, Jane L. Chang, Ramon Eritja, Marc Ferrer, Cynthia G. Fields, Gregg B. Fields, Mattew H. Lyttle, Nuria A. Solé, Zhenping Tian, Robert J. Van Abel, Peter B. Wright, Samuel Zalipsky, and Derek Hudson. Biopolymer syntheses on novel polyethylene glycol-polystyrene (PEG-PS) graft supports. In Peptides - Chemistry and Biology: Proceedings of the Twelfth American Peptide Synposium (J. A. Smith and J. Rivier, eds.), Escom, Science Publishers, Leiden, The Netherlands, 603-604 (1992).
• Mark C. Munson, Carlos García-Echeverría, Fernando Albericio, and George Barany. Novel cysteine protecting groups for the Nα-9-fluorenylmethyloxycarbonyl (Fmoc) strategy of peptide synthesis. In Peptides - Chemistry and Biology: Proceedings of the Twelfth American Peptide Synposium (J. A. Smith and J. Rivier, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 605-606 (1992).
• Fernando Albericio, Paul Lloyd-Williams, Margarida Gairí, Gemma Jou, Ramon Eritja, and Ernest Giralt. Convergent solid-phase peptide synthesis. In Peptides - Chemistry and Biology: Proceedings of the Twelfth American Peptide Synposium (J. A. Smith and J. Rivier, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 607-608 (1992).
• Carlos García-Echeverría, Fernando Albericio, Miquel Pons, and Ernest Giralt. Study of a parallel bis-cysteine peptide as a potential ionophore. In Peptides - Chemistry and Biology: Proceedings of the Twelfth American Peptide Synposium (J. A. Smith and J. Rivier, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 917-918 (1992).
• George Barany, Nuria A. Solé, Robert J. van Abel, Fernando Albericio, and Michael Selsted. Recent advances in solid-phase peptide synthesis. In Innovation and Perspectives in Solid-Phase Peptide Synthesis and Related Technologies: Peptides, Polypeptides and Oligonucleotides 1992 (R. Epton, ed.), Intercept, Andover (UK), pp. 29-38 (1992).
• Fernando Albericio, Paul Lloyd-Williams, Margarida Gairí, Gemma Jou, Carles Celma, Nancy Kneib-Cordonier, Anna Grandas, Ramon Eritja, Enrique Pedroso, Jurphaas van Rietschoten, George Barany, and Ernest Giralt. Convergent solid-phase peptide synthesis. In Innovation and Perspectives in Solid-Phase Peptide Synthesis and Related Technologies: Peptides, Polypeptides and Oligonucleotides 1992 (R. Epton, ed.), Intercept, Andover (UK), pp. 39-47 (1992).
• Miriam Royo, Carlos García-Echeverría, Mark C. Munson, Urszula Slomcynska, Ramon Eritja, Ernest Giralt, George Barany, and Fernando Albericio. Cysteine protection in solid-phase peptide synthesis. In Innovation and Perspectives in Solid-Phase Peptide Synthesis and Related Technologies: Peptides, Polypeptides and Oligonucleotides 1992 (R. Epton, ed.), Intercept, Andover (UK), pp. 461-465 (1992).
• Núria Xaus, Fernando Albericio, Xavier Jorba, Silvia Calvet, Pere Clapés, Josep L. Torres, and Gregorio Valencia. Racemization free coupling of peptide segments. Total synthesis of an insect neuropeptide. Int. J. Peptide Protein Res.39, 528-532 (1992).
• Núria Xaus, Xavier Jorba, Silvia Calvet, Fernando Albericio, Pere Clapés, Josep L. Torres, and Gregorio Valencia. Enzymatic peptide fragment condensation. Choice of reaction media for the synthesis of an insect neuropeptide derivative. Biotechnol. Tech.6, 69-72 (1992).
• Rei Matsueda, Susumu Higashida, Fernando Albericio, and David Andreu. Stability of S-Npys protecting group against HOBt. In "Peptide Chemistry 1991: Proceedings of the 29th Symposium on Peptide Chemistry" (A. Suzuki, ed.), Protein Research Foundation, pp. 111-114 (1992).
• Carlos García-Echeverría, Miquel Pons, Ernest Giralt, and Fernando Albericio. Synthesis and ion-binding properties of an immobilized bis-cysteine peptide. Bioorganic & Medicinal Chem. Lett.2, 281-284 (1992).
• Josep Rizo, Fernando Albericio, Ernest Giralt, and Enrique Pedroso. Reversible protection of lysine to facilitate the purification of protected peptide segments. Tetrahedron Lett. 33, 397-400 (1992).
• Francesc Rabanal, Ernest Giralt, and Fernando Albericio. A new fluorene-derived anchor for solid-phase synthesis of protected peptides. Tetrahedron Lett., 33, 1775-1778 (1992).
• Ernesto Nicolás, Javier Clemente, Margarita Perelló, Fernando Albericio, Enrique Pedroso, and Ernest Giralt. A new approach to the solid-phase peptide synthesis of peptide alkyl-amides and esters. Tetrahedron Lett. 33, 2183-2186 (1992).
• Miriam Royo, Carlos García-Echeverría, Ernest Giralt, Ramon Eritja, and Fernando Albericio. S-2-(2,4-Dinitrophenyl)ethyl-L-cysteine: a new derivative for solid-phase peptide synthesis. Tetrahedron Lett. 33, 2391-2394 (1992).
• Mark C. Munson, Carlos García-Echeverría, Fernando Albericio, and George Barany. S-2,4,6-Trimethoxybenzyl (Tmob): a novel cysteine protecting group for the Nα-9-fluorenylmethyloxycarbonyl (Fmoc) strategy of peptide synthesis. J. Org. Chem.57, 3013-3018 (1992).
• Montse Acedo, Fernando Albericio, and Ramon Eritja. 2-(2,4-Dinitrophenyl)-ethyloxycarbonylamino acids, new base labile protected derivatives suitable for solid-phase peptide synthesis. Tetrahedron Lett. 33, 4989-4952 (1992).
• Ramon Eritja, Jordi Robles, Fernando Albericio, and Enrique Pedroso. A synthetic procedure for the preparation of oligonucleotides without using ammonia and its application for the synthesis of oligonucleotides containing O-4-alkyl-thymidines. Tetrahedron 40, 4171-4182 (1992).
• Rei Matsueda, Susumu Higashida, Fernando Albericio, and David Andreu. Compatibility of the S-(3-nitro-2-pyridinesulfenyl) protecting group with DCC/HOBt coupling chemistry. Peptide Res.5, 262-264 (1992).
• M. Dolors Ludevid, Miguel A. Freire, Jordi Gómez, Christopher G. Burd, Fernando Albericio, Ernest Giralt, Gideon Dreyfuss, and Montserrat Pagès. RNA binding characteristics of a 16 kDa glycine-rich protein from maize. The Plant Journal2, 999-1003 (1992).
• Fernando Albericio and George Barany. Acidolytic cleavage of tris(alkoxy)benzyl-amide (PAL) "internal reference" amino acyl (IRAA) anchoring linkages: validation of accepted procedures in solid-phase peptide synthesis (SPPS). Int. J. Peptide Protein Res.41, 307-312 (1993).
• Fernando Albericio, George Barany, Gregg B. Fields, Derek Hudson, Steven A. Kates, Mattew H. Lyttle, and Nuria A. Solé. Allyl-based orthogonal solid-phase peptide synthesis. In Peptides 1992: Proceedings of the Twenty-Second European Peptide Symposium (C.H. Schneider and A.N. Eberle, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 191-193 (1993).
• George Barany, Fernando Albericio, Nuria A. Solé, G. Wiliam Griffin, Steven A. Kates, and Derek Hudson. Novel polyethylene glycol-polystyrene (PEG-PS) graft supports for solid-phase peptide synthesis. In Peptides 1992: Proceedings of the Twenty-Second European Peptide Symposium (C.H. Schneider and A.N. Eberle, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 267-268 (1993).
• Francesc Rabanal, Fernando Albericio, Ronald Cotton, and Ernest Giralt. 2-Amino-fluorene as a useful compound in convergent solid-phase peptide synthesis. In Peptides 1992: Proceedings of the Twenty-Second European Peptide Symposium (C.H. Schneider and A.N. Eberle, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 288-289 (1993).
• Marc Canas, Gemma Jodas, Fernando Albericio, David Andreu, Jose M. García-Antón, Antonio Parente, and Berta Ponsati. Optimization of iodine oxidation methods for S-Acm, S-Trt dicysteinyl-peptides on the resin. In Peptides 1992: Proceedings of the Twenty-Second European Peptide Symposium (C.H. Schneider and A.N. Eberle, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 401-402 (1993).
• Pere Clapés, Yolanda M. Sanchéz, Fernando Albericio, Josep L. Torres, and Gregorio Valencia. Solid-phase synthesis of carboxamidomethyl (CAM) peptide esters. Application to the enzymatic fragment condensation. In Peptides 1992: Proceedings of the Twenty-Second European Peptide Symposium (C.H. Schneider and A.N. Eberle, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 423-424 (1993).
• Miriam Royo, Fernando Albericio, Ernest Giralt, and Miquel Pons. Use of cyclic dimers of palindromic peptides for the study of coiled-coils. In Peptides 1992: Proceedings of the Twenty-Second European Peptide Symposium (C.H. Schneider and A.N. Eberle, eds.), Escom, Science Publishers, Leiden, The Netherlands, pp. 487-488 (1993).
• Steven A. Kates, Nuria A. Solé, Charles R. Johnson, Derek Hudson, George Barany, and Fernando Albericio. A novel, convenient, three-dimensional orthogonal strategy for solid-phase synthesis of cyclic peptides. Tetrahedron Lett., 34, 1549-1552 (1993).
• Fernando Albericio, Miriam Royo, Mark C. Munson, Nuria A. Solé, Robert J. Van Abel, Jordi Alsina, Carlos García-Echeverría, Urszula Slomczynska, Ramon Eritja, Miquel Pons, Ernest Giralt, and George Barany. Strategy and tactics for the solid-phase synthesis of cystine-containing peptides. In Proceedings of the 2nd Japan Symposium on Peptide Chemistry (N. Yanaihara, ed.), Escom, Science Publishers, Leiden, The Netherlands, pp. 19-23 (1993).
• Mariano Ruiz-Gayo, Miriam Royo, Imma Fernández, Fernando Albericio, Ernest Giralt, and Miquel Pons. Unequivocal synthesis and characterization of a parallel and an antiparallel bis-cysteine peptide. J. Org. Chem., 58, 6319-6328 (1993).
• Carlos García-Echeverría, Fernando Albericio, Ernest Giralt, and Miquel Pons. Design, synthesis, and complexing properties of (1Cys-1’Cys, 4Cys–4’Cys)-dithiobis(Ac-L-1Cys-L-Pro-D-Val-L-4Cys-NH2). The first example of a new family of ion-binding peptides. J. Am. Chem. Soc., 115, 11663-11670 (1993).
• Beatriz G. de la Torre, Anna M. Aviño, Mónica Escarceller, Miriam Royo, Fernando Albericio, and Ramon Eritja. Use of a base-labile protected derivative of 6-mercaptohexanol for the preparation of oligonucleotides containing a thiol group at the 5'end. Nucleosides & Nucleotides, 12, 993-1005 (1993).
• Steven A. Kates, Scott B. Daniels, and Fernando Albericio. Automated allyl cleavage for continuous-flow synthesis of cyclic and branch peptides. Anal. Biochem., 212, 303-310 (1993).
• Ernest Giralt, Fernando Albericio, David Andreu, Carlos García-Echeverrría, Miquel Pons, Xavier Roig, and Miriam Royo. Peptides in molecular recognition. An. Quím. 89, C, 79-84 (1993).
• Djamel Ait-Amara, Carlos Chavez-Olortegui, Régine Romi, Jean Mery, Jean Brugidou, Fernando Albericio, Christiane Devaux, and Claude Granier. Antibodies cross-reactive with the scorpion-toxin II from Androctonus australis Hector elicited in mice by a synthetic peptide. Natural Toxins, 1, 255-262 (1993).
• Louis A. Carpino, Hitesh Shroff, Salvatore A. Triolo, El-Sayed M.E. Mansour, Holger Wenschuh, and Fernando Albericio. The 2,2,4,6,7-pentamethyl-dihydrobenzofuran-5-sulfonyl group (Pbf) as arginine side chain protectant. Tetrahedron Lett., 34, 7829-7832 (1993).
• Paul Lloyd-Willimans, Margarida Gairí, Fernando Albericio, and Ernest Giralt. Convergent solid-phase peptide synthesis. XI. Synthesis and purification of protected peptide segments sapnning the entire sequence of the uteroglobin monemer using the photolabile Nbb-resin. Tetrahedron, 49, 10069-10078 (1993).
• Paul Lloyd-Williams, Fernando Albericio, and Ernest Giralt. Convergent solid-phase peptide synthesis. Tetrahedron, 49, 11065-11133 (1993).
• Louis A. Carpino, Ayman El-Faham, Charles A. Minor, and Fernando Albericio. Advantageous applications of azabenzotriazole-based coupling reagents to solid-phase peptide synthesis. J. Chem. Soc., Chem. Commun., 201-203 (1994).
• Margarida Gairí, Paul Lloyd-Williams, Fernando Albericio, and Ernest Giralt. Severe side-reaction in the acidolytic cleavage of a C-terminal Met-containing peptide from the solid-support. Formation of a homoserine lactone tripeptide. Tetrahedron Lett., 35, 175-178 (1994).
• Steven A. Kates, Beatriz G. de la Torre, Ramon Eritja, and Fernando Albericio. Solid-phase N-glycopeptide synthesis using allyl side-chain protected Fmoc amino acids. Tetrahedron Lett., 35, 1033-1034 (1994).
• Yongxin Han, Mark C. Munson, Fernando Albericio, and George Barany. Preparation and applications of Xanthenyalmide (XAL) handles for mild Fmoc solid-phase synthesis of C-terminal amides. In Proceedings of the First Chinese Peptide Symposium (D. Yu-cang, J.P. Tam, Y. Zhang, eds.), ESCOM, Science Publishers, Leiden, The Netherlands, 1993, pp. 301-304.
• Gloria del Solar, Fernando Albericio, Ramon Eritja, and Manuel Espinosa. Complete chemical synthesis of a fully active transcriptional repressor. Proc. Natl. Acad.Sci.. USA., 91, 5178-5182 (1994).
• Fernando Albericio, Louis A. Carpino, Scott B. Daniels, Ayman El-Faham, Hiroyuki Fukuda, G. William Griffin, Steven A. Kates, Charles A. Minor, Hitesh N. Shroff, Salvatore A. Triolo, G. Tony. Truran, and Kaoru Yamabe. New approaches in solid-phase peptide synthesis. In "Peptide Chemistry 1993: Proceedings of the 31th Symposium on Peptide Chemistry" (Y. Okada, ed.), Protein Research Foundation, Osaka (Japan) pp. 121-124 (1994).
• Ernest Giralt, Fernando Albericio, Ionara Dalcol, Margarida Gairí, Paul Lloyd-Williams, and Francesc Rabanal. Convergent solid-phase peptide synthesis. In Innovation and Perspectives in Solid-Phase Peptide Synthesis: Biological & Biomedical Applications (R. Epton, ed.), Mayflower WorlwideLimited, Birmingham, England, pp. 51-60 (1994).
• Louis A. Carpino, Ayman El-Faham, George A. Truran, Charles A. Minor, Steven A. Kates, G. William Griffin, Hitesh Shroff, Salvatore A. Triolo, and Fernando Albericio. New approaches for extending the scope of solid-phase peptide synthesis. In Innovation and Perspectives in Solid-Phase Peptide Synthesis: Biological & Biomedical Applications (R. Epton, ed.), Mayflower WorlwideLimited, Birmingham, England, pp. 95-104 (1994).
• Nuria A. Solé, Steve A. Kates, Fernando Albericio, and George Barany. Orthogonal solid-phase synthesis of bicyclic peptides. In Innovation and Perspectives in Solid-Phase Peptide Synthesis: Biological & Biomedical Applications (R. Epton, ed.), Mayflower WorlwideLimited, Birmingham, England, pp.105-110 (1994).
• David Andreu, Fernando Albericio, Nuria A. Solé, Mark C. Munson, Marc Ferrer, and George Barany. Formation of disulfide bonds in synthetic peptides and proteins. In “Methods in Molecular Biology, Vol. 35: Peptide Synthesis Protocols” (M.W. Pennington and B.M. Dunn, eds.), Humana Press, Totowa , N.J., pp. 91-169 (1994).
• Nuria A. Solé, Steven A. Kates, Fernando Albericio, and George Barany. Orthogonal solid-phase synthesis of bicyclic analogues of α-conotoxin SI. In Peptides - Chemistry and Biology: Proceedings of the Thirteenth American Peptide Synposium (R. S. Hodges and J. A. Smith, eds.), ESCOM, Science Publishers, Leiden, The Netherlands, 1994, pp. 93-94.
• Steven A. Kates, Scott B. Daniels, Nuria A. Solé, George Barany, and Fernando Albericio. Automated allyl chemistry for solid-phase peptide synthesis: Applications to cyclic and branched peptides. In Peptides - Chemistry and Biology: Proceedings of the Thirteenth American Peptide Synposium (R. S. Hodges and J. A. Smith, eds.), ESCOM, Science Publishers, Leiden, The Netherlands, 1994, pp. 113-115.
• Miriam Royo, Jordi Alsina, Ernest Giralt, Urszula Slomczynska, and Fernando Albericio. S-Phenylacetamidomethyl (Phacm). A versatile cysteine protecting group fopr Boc and fmoc solid-phase synthesis strategies. In Peptides - Chemistry and Biology: Proceedings of the Thirteenth American Peptide Synposium (R. S. Hodges and J. A. Smith, eds.), ESCOM, Science Publishers, Leiden, The Netherlands, 1994, pp. 116-118.
• Hitesh N. Shroff, Louis A. Carpino, Holger Wenschuh, El-Sayed M.E. Mansour, Salvatore A. Triolo, G. William Grifin, and Fernando Albericio. The 2,2,4,6,7-pentamethyldihydrobenzofuran-5-sulfonyl group (Pbf): A new acid-labile sulfonamide type side-chain protecting group for arginine. In Peptides - Chemistry and Biology: Proceedings of the Thirteenth American Peptide Synposium (R. S. Hodges and J. A. Smith, eds.), ESCOM, Science Publishers, Leiden, The Netherlands, 1994, pp. 121-123.
• Louis A. Carpino, Ayman El-Faham, George A. Truran, Salvatore A. Triolo, Hitesh Shroff, G. William Griffin, Charles A. Minor, Steven A. Kates, and Fernando Albericio. Azabenzotriazole-based coupling reagents in solid-phase peptide synthesis. In Peptides - Chemistry and Biology: Proceedings of the Thirteenth American Peptide Synposium (R. S. Hodges and J. A. Smith, eds.), ESCOM, Science Publishers, Leiden, The Netherlands, 1994, pp. 124-126.
• George Barany and Fernando Albericio. Recent progress on handles and supports for solid-phase peptide synthesis. In Peptides - Chemistry and Biology: Proceedings of the Thirteenth American Peptide Synposium (R. S. Hodges and J. A. Smith, eds.), ESCOM, Science Publishers, Leiden, The Netherlands, 1994, pp. 1078-1080.
• Steven A. Kates, Núria A. Solé, Fernando Albericio, and George Barany. Solid-phase synthesis of cyclic peptides. In Peptides: design, synthesis, and biological activity (C. Basava and G.M. Anantharamaiah, eds.), Birkhauser, Boston (Massachusetts), pp.39-58 (1994).
• Louis A. Carpino, Ayman El-Faham, and Fernando Albericio. Racemization studies during solid-phase peptide synthesis using azabenzotriazole-based coupling reagents. Tetrahedron Lett., 35, 2279-2283 (1994).
• Beatriz G. de la Torre, Anna Aviño, Gemma Tarrason, Jaume Piulats, Fernando Albericio, and Ramon Eritja. Stepwise solid-phase synthesis of oligonucleotide-peptide hybride. Tetrahedron Lett., 35, 2733-2736 (1994).
• Samuel Zalipsky, Jane L. Chang, Fernando Albericio, and George Barany. Preparation and applications of polyethylene glycol-polystyrene graft resin supports for solid-phase peptide synthesis. Reactive Polym., 22, 243-258 (1994).
• Paul Lloyd-Williams, Ahmed Merzouk, François Guibé, Fernando Albericio, and Ernest Giralt. Solid-phase synthesis of peptides using allylic anchoring groups 2. Palladium-catalysed cleavage of Fmoc-protected peptides. Tetrahedron Lett., 35, 4437-4440 (1994).
• Jordi Alsina, Francesc Rabanal, Ernest Giralt, and Fernando Albericio. Solid-phase synthesis of head-to-tail cyclic peptides via lysine side-chain anchoring. Tetrahedron Lett., 35, 9633-9636 (1994).
• Ernest Giralt, Fernando Albericio, Carlos García-Echeverría, Miquel Pons, Miriam Royo, Mariano Ruiz-Gayo. Peptides in molecular recognition: synthetic and conformational aspects. Biochem. Soc. Trans., pp. 1045-1048 (1994).
• Iman Abdelmoty, Fernando Albericio, Louis A. Carpino, Bruce F. Foxman, and Steven A. Kates. Structural studies of reagents for peptide bond formation: crystal and molecular structures of HBTU and HATU. Lett. Peptide Sci. 1, 57-67 (1994); https://doi.org/10.1007/BF00126274
• Fernando Albericio, Iman Abdelmoty, Josep M. Bofill, Louis A. Carpino, Ayman El-Faham, Bruce M. Foxman, Margarida Gairí, G. William Griffin, Steven A. Kates, Paul Lloyd-Williams, Louis M. Scarmoutzos, Hitesh Shroff, Salvatore A. Triolo, and Holger Wenschuh. Azabenzotriazole (HOAt) derivatives as superior coupling reagents for peptide synthesis. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, pp. 23-25.
• Ionara Dalcol, Francesc Rabanal, Fernando Albericio, Miquel Pons, M. Geli, M. Torrent, M.Dolors Ludevid, and Ernest Giralt. A proline-rich region from maize  zein adopts a left-handed amphipathic structure that may act as a signal for its retention in the endoplasmic reticulum. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, pp. 60-61.
• Miriam Royo, Fernando Albericio, Ernest Giralt, Miquel Pons. Helicity and superhelicity in cyclic coiled-coil peptides. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, 83-84.
• Louis A. Carpino, Hitesh N. Shroff, Hann-Guang Chao, El-Sayed M.E. Mansour, Fernando Albericio. New acid-labile, side-chain protecting groups for asparagine and glutamine. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, 155-156.
• Steven A. Kates, Charles A. Minor, Hitesh Shroff, Ronald C. Haaseth, Salvatore A. Triolo, Ayman El-Faham, Louis A. Carpino, and F. Albericio. Practical protocols for efficient solid-phase peptide synthesis. Minimization of side-reactions. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, 248-249.
• Steven A. Kates, Charles A. Minor, Fernando Albericio, Yongxin Han, and George Barany. Use of XAL handles for solid-phase synthesis of peptide amides. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, pp. 262-264.
• Fernando Albericio, Jordi Bacardi, George Barany, James M. Coull, Michael Egholm, Ernest Giralt, G. William Griffin, Steven A. Kates, Ernesto Nicolás, and Nuria A. Solé. Polyethylene glycol-polystyrene (PEG-PS) supports for Boc solid-phase peptide and PNA synthesis strategies. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, 271-272.
• Holger Wenschuh, Louis A. Carpino, Fernando Albericio, Eberhard Krause, Michael Beyermann, Michael Bienert. Stepwise solid phase synthesis of peptaibols using Fmoc amino acid fluorides. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, 287-288.
• Beatriz G. de la Torre, Anna Aviño, Fernando Albericio, Ramon Eritja. Stepwise solid-phase synthesis of oligonucleotide-peptide hybrids. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, 303-304.
• Knud J. Jensen, Eduard Bardají, Fernando Albericio, James M. Coull, and George Barany. Synthesis of peptide nucleic acid (PNA) oligomers from N-dithiasuccinoyl (Dts) protected monomers. In Peptides 1994: Proceedings of the Twenty-Third European Peptide Symposium (H.L.S. Maia, ed.), ESCOM, Science Publishers, Leiden, The Netherlands, 1995, 757-758.
• Fernando Albericio and Steven A. Kates. Azidotris(dimethylamino)phosphonium hexafluorophosphate. In Encyclopedia of reagents for organic synthesis (L.A. Paquette, ed.), Vol. 1, John Wiley & Sons Ltd, Chichester, U.K., 224-225.
• Steven A. Kates and Fernando Albericio. 1,1'-Azo-bis-1-cyclohexanenitrile. In Encyclopedia of reagents for organic synthesis (L.A. Paquette, ed.), Vol. 1, John Wiley & Sons Ltd, Chichester, U.K., 228-229.
• Fernando Albericio and Steven A. Kates. 1-Benzotriazolyl diethyl phosphate. In Encyclopedia of reagents for organic synthesis (L.A. Paquette, ed.), Vol. 1, John Wiley & Sons Ltd, Chichester, U.K., 300-301.
• Fernando Albericio, Steven A. Kates, and Ramon Eritja. 4,4'-Bis(2-amino-6-methylpyrimidyl) disulfide. In Encyclopedia of reagents for organic synthesis (L.A. Paquette, ed.), Vol. 1, John Wiley & Sons Ltd, Chichester, U.K., 421.
• Fernando Albericio and Steven A. Kates. O-Benzotriazol-1-yl-N,N,N',N'-tetramethyluronium hexafluorophosphate. In Encyclopedia of reagents for organic synthesis (L.A. Paquette, ed.), Vol. 1, John Wiley & Sons Ltd, Chichester, U.K., 304-306.
• Fernando Albericio, Louis A. Carpino, and Steven A. Kates. N-[(Dimethylamino)-1H-1,2,3-triazolo[4,5-b]pyridin-1-ylmethylene]-N-methylmethanaminium hexa-fluorophosphate N-oxide (HATU). In Encyclopedia of reagents for organic synthesis (L.A. Paquette, ed.), Vol. 3, John Wiley & Sons Ltd, Chichester, U.K., 2026-2028.
• Steven A. Kates, Louis A. Carpino, and Fernando Albericio. 7-Aza-1-hydroxybenzotriazole or 3-Hydroxy-3H-1,2,3-triazolo[4,5-b]pyridine (HOAt). In Encyclopedia of reagents for organic synthesis (L.A. Paquette, ed.), Vol. 4, John Wiley & Sons Ltd, Chichester, U.K., 2784-2784.
• Ramon Eritja, Steven A. Kates, and Fernando Albericio. Benzenesulfonyltetrazole. In Encyclopedia of reagents for organic synthesis (L.A. Paquette, ed.), Vol. 6, John Wiley & Sons Ltd, Chichester, U.K., 4058-4059.
• Francesc Rabanal, Ernest Giralt, and Fernando Albericio. Synthesis and applications of a new base-labile fluorene derived linker for solid-phase peptide synthesis. Tetrahedron , 51, 1449-1458 (1995).
• Holger Wenschuh, Michael Beyermann, Hanka Haber, Joachim K. Seydel, Eberhard Krause, Michael Bienert, Louis A. Carpino, Ayman El-Faham, Fernando Albericio. Stepwise automated solid phase synthesis of naturally occurring peptaibols using Fmoc amino acid fluorides. J. Org. Chem., 60, 405-410 (1995).
• Steven A. Kates and Fernando Albericio. Rearragement of Glu(OtBu) and Asp(OtBu)-containing peptides upon fluoride treatment in solid-phase synthesis. Lett. Peptide Sci., 1, 213-220 (1995).
• Miriam Royo, Jordi Alsina, Ernest Giralt, Urszula Slomcynska, and Fernando Albericio. S-Phenylacetamidomethyl (Phacm): an orthogonal cysteine protecting group for Boc and Fmoc solid-phase peptide synthesis strategies. J. Chem Soc. Perkin I, pp. 1095-1102 (1995).
• Margarida Gairí, Paul Lloyd-Williams, Fernando Albericio, Ernest Giralt. Convergent Solid-Phase Peptide Synthesis. 12. Chromatographic techniques for the purication of protected peptide segments. Int. J. Peptide Protein Res., 46, 119-133 (1995).
• Louis A. [1], Ayman El-Faham, and Fernando Albericio. Racemization control in peptide coupling. 1-Hydroxy-7-azabenzotriazole (HOAt) vs. 3,4-dihydro-3-hydroxy-4-oxo-1,2,3-benzotriazine (HODhbt). J. Org. Chem., 60, 3561-3564 (1995).
• Ionara Dalcol, Francesc Rabanal, M.Dolors Ludevid, Fernando Albericio, and Ernest Giralt. Convergent solid-phase peptide synthesis: an efficient approach to the synthesis of highly repetitive protein domains. J. Org. Chem.,60, 7575-7581 (1995).
• Louis A. Carpino, Hann Guang Gao, Shahnaz Ghassemi, E.E.E. Mansour, Cristoph Riemer, Ralf Warrass, Dean Sadat-Aalaee, George A. Truran, Hideko Imazumi, Ayman El-Faham, Mohamed Ismail, Thadeus L. Kowaleski, Chung Hwa Han, Holger Wenschuch, Michael Beyermann, Michael Bienert, Hitesh Shroff, Fernando Albericio, Salvatore A. Triolo, and Steven A. Kates. Novel carboxylic acid and carboxamide protective group based on the exceptional stabilization of the cyclopropylmethyl cation. J. Org. Cherm., 60, 7718-7719 (1995).
• Josep M. Bofill and Fernando Albericio. Theoretical and experimental structural studies of reagents for peptide bond formation: molecular structure and mechanism of HATU. J. Chem. Res., 302-303 (1996).
• Yongxin Han, Susan L. Botems, Peter Hegyes, Mark C. Munson, Charles A. Minor, Steven A. Kates, Fernando Albericio,and George Barany. Preparation and Applications of Xanthenylamide (XAL) Handles for Solid-Phase Synthesis of C-terminal Peptide Amides under Particularly Mild Conditions. J. Org. Cherm. 61, 6326-6339 (1996).
• Isabel González, Gemma Jou, Josep María Caba, Fernando Albericio, Paul Lloyd-Williams, and Ernest Giralt. Synthesis of derivatives of (2S, 4S)-4-hydroxy-2,5-dimethyl-3-oxo-hexanoic acid, a constituent of the Didemnins. J. Chem. Soc. Perkin I., 1427-1433 (1996).
• Anna Aviño, Ramon Güimil García, Fernando Albericio, Matthias Mann, Matthias Wilm, Gitte Neubauer, and Ramon Eritja. New Carbamate Supports for the Preparation of 3'Amino-modified Oligonucleotides. Bioorg. Med. Chem., 4, 1649-1658 (1996).
• Jordi Alsina, Ernest Giralt, and Fernando Albericio. Use of N-Tritylamino Acids and PyAOP for the Suppression of Diketopiperazine Formation in Fmoc/tBu Solid-Phase Peptide Synthesis Using Alkoxybenzyl Ester Anchoring Linkages. Tetrahedron Lett., 37, 4195-4198 (1996).
• Steven A. Kates,Nuria A. Solé, Michael Beyermann, George Barany,and Fernando Albericio. Optimized Preparation of Deca(L-Alanyl)-L-Valinamide by 9 Fluorenylmethyl-oxycarbonyl (Fmoc) Solid-Phase Synthesis on Polyethylene Glycol-Polystyrene (PEG-PS) Graft Supports, with 1,8-Diazobicyclo[5.4.0]-undec-7-ene (DBU) Deprotection. Peptide Res., 9, 106-113 (1996).
• Anna Aviño, Ramon Güimil García, Antonio Díaz, Fernando Albericio, and Ramon Eritja. A Comparative Study of Supports for the Synthesis of Oligonucleotides without using Ammonia for the final deprotection. Nucleotides & Nucleosides, 15, 1871-1889 (1996).
• Jan Lukszo, Dale Patterson, Fernando Albericio, Steven A. Kates. 3-(1-Piperidinyl)alanine formation during the preparation ofC-terminal cysteine peptides with the Fmoc/t-Bu strategy. Lett. Peptide Sci.,3, 157-166 (1996).
• Knud J. Jensen, Michael F. Songster, Jordi Alsina, Josef Vágner, Fernando Albericio, and George Barany. A novel handle approach for solid-phase peptide synthesis: backbone amide (BAL) anchoring. In Peptides - Chemistry and Biology: Proceedings of the Fourteenth American Peptide Synposium(P.T.P. Kaumaya and R. S. Hodges eds.), Mayflower Worlwide Limited, Birmingham, England, 1996, pp. 30-32.
• Steven A. Kates, Salvatore A. Triolo, Elke Diekmann, Louis A. Carpino, Ayman El-Faham, Dumitru Ionescu, and Fernando Albericio. Recent developments in azabenzotriazole-based coupling reagents for use in solid-phase peptide synthesis. In Peptides - Chemistry and Biology: Proceedings of the Fourteenth American Peptide Synposium (P.T.P. Kaumaya and R. S. Hodges eds.), Mayflower Worlwide Limited, Birmingham, England, 1996, 115-116.
• Brian F. McGuinness, Steven A. Kates, G. William Griffin, Lee W. Herman, Nuria A. Solé, Josef Vágner, Fernando Albericio, and George Barany. "High Load" polyethylene glycol-polystyrene graft-supports for solid-phase peptide synthesis. In Peptides - Chemistry and Biology: Proceedings of the Fourteenth American Peptide Synposium (P.T.P. Kaumaya and R. S. Hodges eds.), Mayflower Worlwide Limited, Birmingham, England, 1996, 125-126.
• Steven A.Kates, Louis A. Carpino, and Fernando Albericio. New coupling techniques for solid-phase peptide synthesis. In Peptides - Chemistry and Biology: Proceedings of the Fourteenth American Peptide Synposium (P.T.P. Kaumaya and R. S. Hodges eds.), Mayflower Worlwide Limited, Birmingham, England, 1996, 893-895.
• Steven A.Kates, Elke Diekmann, Ayman El-Faham, Dumitru Ionescu, Brian F. McGuinness, Salvatore A. Triolo, Fernando Albericio, and Louis A. Carpino. On the use of novel coupling reagents for solid-phase peptide synthesis. In Tecniques in Protein Chemistry VII (D.R. Marsshak, ed.) Academic Press, New York, 1996, 515-523.
• Steven A.Kates, Salvatore A. Triolo, G. Wiliam Griffin, Lee W. Herman, George Tarr, Nuria A. Solé, Elke Diekmann, Ayman El-Faham, Dumitru Ionescu, Fernando Albericio, and Louis A. Carpino. Advances in the use of onium-based oupling reagents: application for solid-phase peptide synthesis and combinatorial libraries. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Chemical Libraries. (R. Epton, ed.), Mayflower Scientific Ltd., Kingswinford, England, 1997, pp. 41-50.
• Knud J. Jensen, Michael F. Songster, Jordi Alsina, Josef Vágner, Fernando Albericio, and George Barany. Backbone amide (BAL) anchoring in solid-phase peptide synthesis. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Chemical Libraries: Biomedical & Biological Applications (R. Epton, ed.), Mayflower Scientific Ltd., Kingswinford, England, 1997, pp. 187-190.
• Paul Lloyd-Williams, Fernando Albericio, Margarida Gairí, and Ernest Giralt. The purification of protected peptide segments. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Chemical Libraries. 1996. (R. Epton, ed.), Mayflower Scientific Ltd., Kingswinford, England, 1997, pp. 195-200.
• Fernando Albericio, Paul Lloyd-Williams, and Ernest Giralt. Métodos de Síntesis Peptídica. In Péptidos: Química, Biología y Medicina. Colección Nuevas Tendencias (D. Andreu and L. Rivas, eds.) CSIC, Madrid, 1997, pp. 39-86.
• Fernando Albericio and David Andreu. Formación de Puentes Disulfuro en Péptidos Sintéticos. In Péptidos: Química, Biología y Medicina. Colección Nuevas Tendencias (D. Andreu and L. Rivas, eds.) CSIC, Madrid, 1997, pp. 87-115.
• Ernest Giralt, Fernando Albericio, and Paul Lloyd-Willimas. Síntesis de Péptidos de Gran Tamaño. In Péptidos: Química, Biología y Medicina. Colección Nuevas Tendencias (D. Andreu and L. Rivas, eds.) CSIC, Madrid, 1997, pp. 117-130.
• Yongxin Han, Fernando Albericio,and George Barany. Occurrence and Minimization of Cysteine Racemization During Stepwise Solid-Phase Peptide Synthesis. J. Org. Chem., 62, 4307-4312 (1997).
• Gemma Jou, Isabel González, Fernando Albericio, Paul Lloyd-Williams, and Ernest Giralt. New Syntheses of the Didemnins: Total Synthesis of Dehydrodidemnin B Based upon Two Novel Routes to Didemnin A. Use of Uronium and Phosphonium Salt Coupling Reagent in Peptide Synthesis in Solution. J. Org. Chem., 62, 354-366 (1997).
• Fernando Albericio and Louis A. Carpino. Coupling Reagents and Activation. In Methods in Enzymology, Solid-Phase Peptide Synthesis (G.B. Fields, ed.), Academic Press, Orlando, 289, 104-126 (1997).
• Fernando Albericio, Paul Lloyd-Williams, and Ernest Giralt. Convergent Solid-Phase Peptide Synthesis. In Methods in Enzymology, Solid-Phase Peptide Synthesis (G.B. Fields, ed.), Academic Press, Orlando, 289, 313-336 (1997).
• Eliandre Oliveira, Antonio Miranda, Fernando Albericio, David Andreu, Antonio C.M. Paiva, Clovis R. Nakaie, and Mineko Tominaga. Comparative Evaluation of the Synthesis and Purification of Transmembrane Peptide Fragments. Rat bradykinin receptor 64-97 as a model. J. Peptide Res., 49, 300-307 (1997).
• Ernesto Nicolás, Javier Clemente, Tina Ferrer, Fernando Albericio, and Ernest Giralt. The Use of the Nbb-Resin for Solid-Phase Synthesis of Peptide Alkylesters and Alkylamides. Synthesis of Leuprolide. Tetrahedron, 53, 3179-3194 (1997).
• Jordi Alsina, Cristina Chiva, Francesc Rabanal, Ernest Giralt, and Fernando Albericio. Active carbonate Resins for Solid-Phase Synthesis Through the Anchoring of an Hydroxyl Function. Tetrahedron Lett., 38, 883-886 (1997).
• Ernesto Nicolás, Montse Pujades, Jordi Bacardit, Ernest Giralt, and Fernando Albericio. A New Approach to the Hmb-backbone Protection into Peptides: Synthesis and Reactivity of N-Fmoc-N-(Hmb)amino Acids. Tetrahedron Lett., 38, 2317-2320 (1997).
• Sharlene Adams, Fernando Albericio, Emil R. Smith, and Robert E. Humphreys. Structure-Activity Relationships in Homologs of an Ii Peptide which Regulates Antigenic Peptide Binding to Cell Surface MHC Class II Molecules. Arznelmittel-Forschung, 47(II), 1069-1077 (1997).
• George Barany, Fernando Albericio, Steven A. Kates, and Maria Kempe. Polyethylene Glycol-Containing Supports for Solid-Phase Synthesis of Peptides and Combinatorial Organic Libraries. In Poly(ethylene glycol): Chemistry and Biological Applications (Harris, J.M. and Zalipsky, S., eds.), ACS Symposium Series 680, Washington, DC., pp. 239-264 (1997).
• Fernando Albericio, Marta Cases, Jordi Alsina,Salvatore A. Triolo, Louis A. Carpino,and Steven A. Kates. On the Use of PyAOP, a Phosphonium Salt Derived from HOAt, in Solid-Phase Peptide Synthesis. Tetrahedron Lett.,38, 4853-4856 (1997).
• David Andreu, Sergi Ruiz, Cristina Carreño, Jordi Alsina, Fernando Albericio, María Angeles Jiménez, Natalia de la Figuera, Rosario Herranz, María Teresa García-López, and Rosario González-Muñiz. IBTM-Containing Gramicidin S Analogues: Evidence for IBTM as a Suitable Type II' -Turn Mimetic. J. Am. Chem. Soc., 119, 10579-10586 (1997).
• Nathalie Thieriet,Jordi Alsina,Ernest Giralt,François Guibé, and Fernando Albericio. Use of Alloc-amino Acids in Solid-Phase Peptide Synthesis. Tandem Deprotection-Coupling Reactions Using Neutral Conditions. Tetrahedron Lett.,38, 7275-7278 (1997).
• Christopher Blackburn, Fernando Albericio, and Steven A. Kates. Functionalized Resins and Linkers for Solid-Phase Synthesis of Small Molecules.Drugs Future, 22, 1007-1025 (1997).
• George Barany, Fernando Albericio, Steven A. Kates, and Maria Kempe. Polyethylene Glycol-Containing Supports for Solid-Phase Synthesis of Peptides and Combinatorial Organic Libraries. Polymer Preprints Am. Chem. Soc. Div. Polym. Chem., 38, 587-588 (1997).
• Christopher Blackburn, Fernando Albericio, and Steven A. Kates. Resins and Linkers for Solid-Phase Synthesis of Small Molecules. In Recent Research Developments in Organic Chemistry (S.G. Pandalai, ed.), Vol. 1, Transworld Research Network, Trivandrum, India, 1997, pp.477-497.
• David Andreu, Sergi Ruiz, Cristina Carreño, Jordi Alsina, Fernando Albericio, M. Angeles Jiménez, Natalia de la Figuera, Rosario Herranz, M. Teresa García-López, and Rosario González-Muñiz. Efficient Synthesis of Gramicidin S and -Turn Dipeptide Mimetic-Containing Analogs by Solid-Phase-Mediated Cyclization via Lys side chain anchoring. In Peptides 1996 Proceedings of the Twenty-Fourth European Peptide Symposium (R. Ramage and R. Epton, eds.), Mayflower Scientific Ltd., Kingswinford, England, 1998, pp. 205-206.
• Beatriz G. de la Torre, Miguel A. Marcos, Jordi Alsina, Ramon Eritja, and Fernando Albericio. N-Tritylamino Acids. Synthesis and Application in Solid-Phase Peptide Synthesis. In Peptides 1996 Proceedings of the Twenty-Fourth European Peptide Symposium (R. Ramage and R. Epton, eds.), Mayflower Scientific Ltd., Kingswinford, England, 1998, pp. 327-328.
• Paul Lloyd-Williams, Gemma Jou, Isabel Gónzalez, Fernando Albericio, and Ernest Giralt. Total Synthesis of Dehydrodidemnin B Based upon Two Novel Routes to Didemnin A. Use of Uronium and Phosphonium Salt Coupling Reagent in Peptide Synthesis in Solution. In Peptides 1996 Proceedings of the Twenty-Fourth European Peptide Symposium (R. Ramage and R. Epton, eds.), Mayflower Scientific Ltd., Kingswinford, England, 1998, pp. 589-590.
• Marta Planas, Susumu Funakoshi, Eduard Bardají, and Fernando Albericio. Synthesis and Applications of a Bis-sulfonyl Handle for Solid-Phase Synthesis of Peptides. In Peptides - Chemistry and Biology: Proceedings of the Fifteen American Peptide Synposium (J.P. Tam and P.T.P. Kaumaya, eds.), Kluwer-ESCOM, Academic Publishers, Dordrecht, The Netherlands, 1998, pp. 307-308.
• Fernando Albericio, Montse del Fresno, Ariadna Frieden, Miriam Royo, Jordi Alsina, Knud J. Jensen, Steven A. Kates, and George Barany. Backbone Amide Linker (BAL) for Solid-Phase Synthesis of 2,5 Piperazinediones (DKP), Useful Scaffolds for Combinatorial Chemistry. In Peptides - Chemistry and Biology: Proceedings of the Fifteen American Peptide Synposium (J.P. Tam and P.T.P. Kaumaya, eds.), Kluwer-ESCOM, Academic Publishers, Dordrecht, The Netherlands, 1998, pp. 37-39.
• Steven A. Kates, Wade Hines, Michael A. Kelley, Paul Lynch, Fernando Albericio, and George Barany. Encoding Schemes for Application with Polyethylene Glycol-Polystyrene Graft (PEG-PS) Supports in Solid-Phase Peptide and Small Molecule Synthesis. In Peptides - Chemistry and Biology: Proceedings of the Fifteen American Peptide Synposium (J.P. Tam and P.T.P. Kaumaya, eds.), Kluwer-ESCOM, Academic Publishers, Dordrecht, The Netherlands, 1998, pp. 67-68.
• Yvonne M. Angell, Yongxin Han, Fernando Albericio, and George Barany. Minimization of Cysteine Racemization During Stepwise Solid-Phase Peptide Synthesis. In Peptides - Chemistry and Biology: Proceedings of the Fifteen American Peptide Synposium (J.P. Tam and P.T.P. Kaumaya, eds.), Kluwer-ESCOM, Academic Publishers, Dordrecht, The Netherlands, 1998, pp. 339-340.
• Seog Soo A. An, Daniel Marti, Cristina Carreño, Fernando Albericio, Johan Schaller, and Miguel Llinás. Functional/structural Analysis of the Glu1-HSer57N-terminal Fragment of Human Plasminogen: Solution Conformation and Interaction with Kringle Domains. Protein Science, 7, 1947-1959 (1998).
• Seog Soo A. An, Cristina Carreño, Daniel Marti, Johan Schaller, Fernando Albericio, and Miguel Llinás. Lysine-50 is a Most Likely Site for Anchoring the Plasminogen N-terminal Domain to Lysine-binding Kringles. Protein Science, 7, 1960-1969 (1998).
• Sharlene Adams, Robert Jackson, Christine Barbon, Hongkui Deng, George Koldzic, Jordi Alsina, Fernando Albericio, Alexander E. Kelly, Dale F. Mierke, Emil R. Smith, Robert E. Humphreys, and Minzhen Xu. Immunosuppression and Antigen Supercharging by Ii-Key peptide-related Compounds. A New Class of Drugs Controlling the First Step in Antigen Recognition. Current ResearchinRheumatoid Arthritis, 2, 1-6 (1998).
• Knud J. Jensen, Jordi Alsina, Michael F. Songster, Josef Vágner, Fernando Albericio,and George Barany. Backbone Amide Linker (BAL) Strategy for Solid-Phase Synthesis of C Terminal Modified and Cyclic Peptides. J. Am. Chem. Soc., 120, 5441-5452 (1998).
• Miriam Royo, Miquel A. Contreras, Ernest Giralt, Fernando Albericio, and Miquel Pons. An Easy Entry to a New High Symmetry, Large Molecular Framework for Molecular Recognition Studies and de novo Protein Design. Solvent Modulation of the Spontaneous Formation of a Cyclic Monomer, Dimer or Trimer from a Bis-Cysteine Peptide. J. Am. Chem. Soc., 120, 6639-6650 (1998).
• Marco Crisma, Giovanni Valle, Vittorio Moretto, Fernando Formaggio, Claudio Toniolo, and Fernando Albericio. Reactive Intermediates in Peptide Synthesis. Molecular and Crystal Structures of HOAt and HOOBt, and Some Ester and Amide Derivatives of HOBt, HOAt, and HOOBt. Lett. Pept. Sci.,5, 247-258 (1998).
• Montserrat del Fresno, Jordi Alsina, Miriam Royo, George Barany, and Fernando Albericio. Solid-Phase Synthesis of Diketopiperazines, Useful Scaffolds for Combinatorial Chemistry. Tetrahedron Lett., 39, 2639-2642 (1998).
• Jordi Alsina, Francesc Rabanal, Cristina Chiva, Ernest Giralt, and Fernando Albericio. Active Carbonate Resins: Application to the Solid-Phase Synthesis of Alcohol, Carbamate, and Cyclic Peptides. Tetrahedron, 54, 10125-10152 (1998).
• Fernando Albericio, Josep M. Bofill, Ayman El-Faham, and Steven A. Kates. On the Use of Onium Salt-Based Coupling Reagents in Peptide Synthesis. J. Org. Chem., 63, 9678-9683 (1998).
• Steven A. Kates, Brian F. McGuinness, Christopher Blackburn, G. William Griffin, Nuria A. Solé, George Barany, and Fernando Albericio. “High Load” Polyethylene Glycol-Polystyrene (PEG-PS) Graft Supports for Solid-Phase Synthesis. Biopolymers (Peptide Science), 47, 365-380 (1998).
• Fernando Albericio, Ariadna Frieden, Montse del Fresno, Miriam Royo, Jordi Alsina, Knud J. Jensen, Steven A. Kates, and George Barany. Strategies for Solid-Phase Synthesis of C-Terminal Modified and Cyclic Peptides. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Chemical Libraries. (R. Epton, ed.), Mayflower Scientific Ltd., Kingswinford, England, pp. 7-10, 1999.
• Christopher Blackburn, George Barany, Fernando Albericio, and Steven A. Kates. Handles for Solid-Phase Chemistry: Progress from Peptide to Small Molecule Synthesis. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Chemical Libraries. (R. Epton, ed.), Mayflower Scientific Ltd., Kingswinford, England, pp. 31-38, 1999.
• Nathalie Thieriet, Jordi Alsina, Michèle Dessolin, M.-G. Guillerez, Ernest Giralt, Fernando Albericio, Albert Loffet, and François Guibé. PhSiH3/Palladium Catalyst/CarboxyactivatedAminoacids: A Ternary System for Tandem Deprotection Coupling of N()-Allocaminoacids and Suppression of DKP Formation in SPPS. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Chemical Libraries. (R. Epton, ed.), Mayflower Scientific Ltd., Kingswinford, England, pp. 127-128, 1999.
• Yvonne M. Angell, Yongxin Han, Fernando Albericio, and George Barany. Minimization of Cysteine Racemization During Stepwise Solid-Phase Peptide Synthesis. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Chemical Libraries. (R. Epton, ed.), Mayflower Scientific Ltd., Kingswinford, England, pp. 247-248, 1999.
• Steven A. Kates, Linda E. Cammish, and Fernando Albericio. Continuous-Flow Solid-Phase Synthesis Using Polystyrene Resins. J. Pept. Res. 53, 682-683 (1999).
• Cristina Chiva, Marta Vilaseca,Ernest Giralt, and Fernando Albericio. An HPLC-ESMS Study on the Solid-Phase Assembly of C-Terminal Proline Peptides. J. Pept. Sci., 5, 131-140 (1999).
• Josep M. Bofill and Fernando Albericio. Understanding the Structure/Reactivity of Aminium/Uronium Salts as Coupling Reagents in Peptide Synthesis. Tetrahedron Lett., 40, 2641-2644 (1999).
• Miriam Royo, Montserrat del Fresno, Ariadna Frieden, Wim Van den Nest, Marina Sanseverino, Jordi Alsina, Steve A. Kates, George Barany, and Fernando Albericio. Useful Scaffolds and Handles for Creating Diversity in the Preparation of Chemical Libraries, Reactive and Functional Polymers, 41, 103-110 (1999).
• Jordi Alsina, George Barany, Fernando Albericio, and Steven A. Kates. Pyrrolidide Formation as a Side Reaction During Activation of Carboxylic Acids by Phosphonium Salt Coupling Reagent. Lett. Peptide Sci., 6, 243-245 (1999).
• Jordi Alsina, Knud J. Jensen, Fernando Albericio, and George Barany. Solid-Phase Synthesis with Backbone Amide Linker (BAL). Chem. Eur. J., 5, 2787-2795 (1999).
• Jordi Alsina, Scott S. Yokum, Fernando Albericio, and George Barany. Backbone Amide Linker (BAL) Strategy for Fluorenylmethoxycarbonyl (Fmoc) Solid Phase Synthesis of Peptides of Unprotected Peptide p-Nitroanilides and Thioesters. J. Org. Chem., 64, 8761-8769 (1999).
• Beatriz G. de la Torre, Fernando Albericio, Ester Saison-Behmoaras, Angela Bachi, Ramon Eritja. C Synthesis and binding properties of oligonucleotides carrying nuclear localization sequences. Bioconjugate Chem., 10, 1005-1012, 1999.
• Paloma Gómez-Martínez, Michèle. Dessolin, François Guibé, and Fernando Albericio. N-Alloc temporary protection in solid-phase peptide synthesis. The use of amine-borane complexes as allyl group scavengers. J. Chem. Soc., Perkin Trans. 1. 22871-2874 (1999).
• Miquel Pons, Fernando Albericio, Miriam Royo, and Ernest Giralt. Disulfide Bonded Cyclic Peptides Dimers and Trimers for Molecular Recognition Studies. Synlett, pp. 172-181 (2000).
• Cristina Carreño,M. Elena Méndez,Hack-Joo Kim, Steven A. Kates, David Andreu,and Fernando Albericio. Nsc and Fmoc N-Amino Protection for Solid-Phase Peptide Synthesis: A Parallel Study. J. Peptide Res., 56, 63-69 (2000)
• Fernando Albericio, Ioana Annis, Miriam Royo, and George Barany. Preparation and Handling of Peptides Containing Methionine and Cysteine. In Fmoc Solid Phase Peptide Synthesis: A Practical Approach (W.C. Chan and P.D. White, eds.) Oxford University Press, Oxford, UK, 2000, pp. 77-114.
• Fernando Albericio and Steven A. Kates. Coupling Methods: Solid-Phase Formation of Amide and Ester Bonds. In Solid-Phase Synthesis. A Practical Guide (S.A. Kates, F. Albericio; eds). Marcel Dekker, New York, NY, 2000, pp. 273-328.
• Nathalie Thieriet, Jordi Alsina, François Guibé, and Fernando Albericio, F. Solid-Phase Peptide Synthesis in the NC direction. In Peptides for the Next Millennium: Proceeding of the 16 th American Peptide Symposium (G.B, Fields, J.P. Tam, G. Barany,; eds.), ESCOM-Kluwer Academic Publishers, Dordrecht, The Netherlands, 2000, pp.78-79.
• Jordi Alsina, Scott S. Yokum, Fernando Albericio, and George Barany. Backbone Amide Linker (BAL) Methodology to Accommodate C-Terminal Hindered, Unreactive, and/or Sensitive Modifications. In Peptides for the Next Millennium: Proceeding of the 16 th the American Peptide Symposium (G.B, Fields, J.P. Tam, G. Barany; eds.), ESCOM-Kluwer Academic Publishers, Dordrecht, The Netherlands, 2000, 102-103.
• John F. McNamara, Holly Lombardo, Sasi K. Pillai, Ivar Jensen, Fernando Albericio, and Steven A. Kates. An Efficient Solid-Phase Strategy for the Construction of Chemokines. J. Pept. Science6, 512-518 (2000).
• Fernando Albericio, Javier García, Enrique L. Michelotti, Ernesto Nicolás, Colin M. Tice. Solid Phase Synthesis of Sulfahydantoins. Tetrahedron Lett. 41, 3161-3163, 2000.
• Nathalie Thieriet, François Guibé, and Fernando Albericio. Solid-Phase Peptide Synthesis in the Reverse Direction. Organic Lett.2, 1815-1817, 2000.
• Francesc Rabanal, Jose J. Pastor, Ernesto Nicolás, Fernando Albericio, and Ernest Giralt. Synthesis of aspartimide-free protected peptides on base-labile functionalized resins. Tetrahedron Lett., 41, 8093-8096 (2000).
• Jordi Alsina, Scott S. Yokum, Fernando Albericio, and George Barany. A Modified Backbone Amide Linker (BAL) Solid-Phase Peptide Synthesis Strategy Accommodating Prolyl, N-Alkylamino Acyl, or Histidyl Derivatives at the C-Terminus. Tetrahedron Lett., 41, 7277-7280 (2000).
• Àngel López-Macià, Jose C. Jiménez, Miriam Royo, Ernest Giralt, and Fernando Albericio. Kahalalide B. Synthesis of a Natural Cyclodepsipeptide. Tetrahedron Lett., 41, 9765-9769 (2000).
• Montserrat del Fresno, Ayman El-Faham, Louis A. Carpino, Miriam Royo, and Fernando Albericio. Substituted Guanidines: Introducing Diversity in Combinatorial Chemistry. Organic Lett., 2, 3539-3542 (2000).
• Fernando Albericio. Editorial: Current Perspectives in Peptide Chemistry. I. Synthesis & Supports. Biopolymers (Peptide Science), 55, 99-100 (2000).
• Fernando Albericio. Orthogonal Protecting Groups for NAmino and C-Terminal Carboxyl Functions in Solid-Phase Peptide Synthesis. Biopolymers (Peptide Science), 55, 123-139 (2000).
• Fernando Albericio. Editorial: Current Perspectives in Peptide Chemistry. II. Synthesis & Supports. Biopolymers (Peptide Science), 55, 187 (2000).
• Paloma Gomez-Martinez, François Guibé, and Fernando Albericio. Allylic Protection of Thiols and Cysteine: III. Use of Fmoc-Cys(Fsam)-OH for Solid-Phase Peptide Synthesis. Lett. Peptide Science,7, 187-194 (2000).
• Miriam Royo, Jose C. Jiménez, Àngel López-Macià, Ernest Giralt, and Fernando Albericio. Solid-Phase Synthesis of Peptides Containing Didehydroamino Acids. European J. Organic Chem., 45-48 (2001).
• Fernando Albericio, Montse Cruz, Laurent Debéthune, Ramon Eritja, Ernest Giralt, Anna Grandas, Vicente Marchán, Jose J. Pastor, Enrique Pedroso, Francesc Rabanal, and Miriam Royo. An Improved Synthesis of N-[(9-Hydroxymethyl)-2-Fluorenyl]Succinamic Acid (HMFS), a Versatile Handle for the Solid-Phase Synthesis of Biomolecules. Synthetic Comm., Synthetic Comm.,31, 225-232 (2001).
• Àngel López-Macià, Jose C. Jiménez, Miriam Royo, Ernest Giralt, and Fernando Albericio. Synthesis and Structural Determination of Kahalalide F. J. Am. Chem. Soc., 123, 11398-11401 (2001).
• Fernando Albericio, Rafael Chinchilla, David Dodsworth, and Carmen Nájera. New Trends in Peptide Coupling Reagents. Org. Prep. & Proc. Int. 33, 203-303 (2001).
• Wim Van den Nest, Shov Yuval, and Fernando Albericio. Cu(OBt)2 and Cu(OAt)2, Copper(II)-Based Racemic Suppressers Ready for Use in Fully Automated Solid-Phase Peptide Synthesis. J. Peptide Science, 7, 115-120 (2001).
• Jordi Alsina, Knud J. Jensen, Michael F. Songster, Josef Vágner, Fernando Albericio, and George Barany (Checked by John Flygare and Monica Fernandez). Backbone Amide Linker (BAL) Strategy for Solid-Phase Synthesis. In Solid-Phase Organic Reactions (SPOS). Vol I. (A. W. Czarnik, ed.), John Wiley & Sons, Inc. New York, 2001, pp. 121-138.
• Jordi Alsina, Scott S. Yokum, Fernando Albericio, and George Barany. Fmoc Solid-Phase Synthesis of Unprotecetd Peptide p-Nitroanilides and Thioesters Using a Backbone Amide Linker (BAL) Strategy. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Chemical Libraries. (R. Epton, ed.), Mayflower Scientific Ltd., Kingswinford, England, 2001, pp 223-226.
• Oscar García, Ernesto Nicolás, and Fernando Albericio. New Dihydrobenzopirane and Dihydrobenzofurane Based Cysteine Protecting Groups for Fmoc Chemistry. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Chemical Libraries. (R. Epton, ed.), Mayflower Scientific Ltd., Kingswinford, England, 2001, pp. 289-290.
• Josep M. Caba, Ignacio Rodriguez, Ignacio Manzanares, Ernest Giralt, and Fernando Albericio. Solid-phase total synthesis of Trunkamide A. J. Org. Chem. 66, 7568-7574, 2001.
• Fernando Albericio, Lois M. Bryman, Javier García, Enrique L. Michelotti, Ernesto Nicolás, and Colin M. Tice. Synthesis of a sulfahydantoin library. J. Comb. Chem.3, 290-300 (2001).
• Cristina Chiva, Fernando Albericio, Ernest Giralt, Frank Molina, Claude Granier, Tatsuya Inui, Hideki Nishio, Yuji Nishiuchi, Terutoshi Kimura, and Shumpei Sakakibara. Total synthesis by combined solid phase and solution approach of the P41 fragment. In Proccedings of the 26th European Peptide Symposium (J. Martinez, J.A. Fehrentz, eds.) Editions Médicales et Scientifiques, Paris (France), 2001, 157-158..
• Àngel López-Macià, Jose C. Jiménez, Miriam Royo, Ernest Giralt, and Fernando Albericio. Kahalalide F: synthesis and structural determination. In Proccedings of the 26th European Peptide Symposium (J. Martinez, J.A. Fehrentz, eds.) Editions Médicales et Scientifiques, Paris (France), 2001, 245-246.
• Àngel López-Macià, Miriam Royo, Jose C. Jiménez, Ernest Giralt, and Fernando Albericio. Solid-phase synthesis of peptides containing -didehydroamino acids. In Proccedings of the 26th European Peptide Symposium (J. Martinez, J.A. Fehrentz, eds.) Editions Médicales et Scientifiques, Paris (France), 2001, 247-248.
• Francesc Rabanal, Jose J. Pastor, Ernesto Nicolás, Fernando Albericio, and Ernest Giralt. Synthesis of protected peptides on N-[9-hydroxymethyl)-2-fluorenyl]succinamic acid (HMFS) derivatised resins: aspartimide side reaction suppression. In Proccedings of the 26th European Peptide Symposium (J. Martinez, J.A. Fehrentz, eds.) Editions Médicales et Scientifiques, Paris (France), 2001, 265-266.
• Wim Van Den Nest, Ruben Ventura, Nathalie Thieriet, Miriam Royo, Youval Shvo, and Fernando Albericio. Coupling reagents: on the use of Cu(OBt)2, Cu(OAt)2 and HOBt-Cl in solid-phase peptide synthesis. In Proccedings of the 26th European Peptide Symposium (J. Martinez, J.A. Fehrentz, eds.) Editions Médicales et Scientifiques, Paris (France), 2001, 287-288.
• Fernando Albericio, Ernest Giralt, Miquel Pons, and Miriam Royo. Solid-phase synthesis and structural studies of functionalized - and -peptides. In Proccedings of the 26th European Peptide Symposium (J. Martinez, J.A. Fehrentz, eds.) Editions Médicales et Scientifiques, Paris (France), 2001, 787-788.
• Laia Crespo, Glòria Sanclimens, Miriam Royo, Miquel Pons, Fernando Albericio, Ernest Giralt. Solid-phase polyproline dendrimer synthesis. In Proccedings of the 26th European Peptide Symposium (J. Martinez, J.A. Fehrentz, eds.) Editions Médicales et Scientifiques, Paris (France), 2001, 801-802.
• Montserrat del Fresno, Miriam Royo, Ayman El-Faham, Louis A. Carpino, and Fernando Albericio. Substituted and non-substituted guanidines introducing diversity for combintorial chemistry. In Proccedings of the 26th European Peptide Symposium (J. Martinez, J.A. Fehrentz, eds.) Editions Médicales et Scientifiques, Paris (France), 2001, 959-960.
• Dolors Fernández-Forner, Gaspar Casals, Elosia Navarro, Hamish Ryder, and Fernando Albericio. Solid-phase synthesis of 4-aminopiperidine analogues using Alloc protecting groups: an investigation of the Alloc removal from secondary amines. Tetrahedron Lett., 42, 4471-4474 (2001).
• Fernando Albericio, Miguel A. Bailén, Rafael Chinchilla, David J. Dodsworth, and Carmen Nájera. 2-Mercaptopyridone-1-oxide-based peptide coupling reagents. Tetrahedron, 57, 9607-9613 (2001).
• Jesús Vázquez and Fernando Albericio. A useful and sensitive color test to monitor aldehydes on solid-phase. Tetrahedron Lett., 42, 6691-6693 (2001).
• Miriam Royo, Wim Van Den Nest, Montserrat del Fresno, Ariadna Frieden, Dror Yahalom, Michael Rosenblatt, Mihael Chorev,and Fernando Albericio. Solid-Phase Syntheses of Constrained RGD Scaffolds and their Binding to the Integrin Receptor. Tetrahedron Lett.,42, 7387-7391 (2001).
• Fernando Albericio, Josep M. Caba, Àngel López-Macià, Jose C. Jiménez,Marta Carrascal, Laia Solé, Ignacio Rodriguez, Ignacio Manzanares, Miriam Royo,and Ernest Giralt. Solid-phase total syntheses of Trunkamide A and Kahalalide F, cyclic peptides from marine origin. In Peptides: The Wave of the Future (M. Lebl, R.A. Houghten; eds.), American Peptide Society, 2001, pp. 217-219.
• Ernest Giralt, Miriam Royo, Marcelo Kogan, Laia Crespo, Glòria Sanclimens, Josep Farrera, Miquel Pons, and Fernando Albericio. Proline: a key building block in “de novo” designed peptide molecules. In Peptides: The Wave of the Future (M. Lebl, R.A. Houghten; eds.), American Peptide Society, 2001, pp. 432-434.
• Miriam Royo, Miquel A. Contreras, Juan Cebrián, Ernest Giralt, Fernando Albericio, and Miquel Pons. Disulfide bond based self-assembly of peptides leading to spheroidal cyclic trimers. In Self-assembling Peptide Systems in Biology, Medicine and Engineering (A. Aggeli, N. Boden, S. Zhang, eds.) Kluwer Academic Publishers, Dordrecht (The Netherlands), 2001, pp. 243-256.
• Bouchaib Bahbouhi, Mourad Bendjennat, Cristina Chiva, Marcelo Kogan, Fernando Albericio, Ernest Giralt, Nabil Georges Seidah and Elmostafa Bahraoui Inhibition of HIV-2ROD replication in a lymphoblastoid cell line by the 1-antitrypsin Portland variant (alpha1-PDX) and the decRVKRcmk peptide: comparison with HIV-1LAI. Microbes and Infection, 3, 1073-1084 (2001).
• Pilar Forns and Fernando Albericio. Merrifield Resin. In e-EROS Encyclopedia of Reagents for Organic Synthesis. (L.A. Paquette, ed.), John Wiley & Sons Ltd, Chichester, U.K., http://www3.interscience.wiley.com/cgi-bin/mrwhome/104554785/HOME (2001).
• Beatriz G. de la Torre, Ramon Eritja, and Fernando Albericio. N-[9-(Hydroxymethyl)-2-fluorenyl]succinamic acid. In e-EROS Encyclopedia of Reagents for Organic Synthesis. (L.A. Paquette, ed.), John Wiley & Sons Ltd, Chichester, U.K., http://www3.interscience.wiley.com/cgi-bin/mrwhome/104554785/HOME (2001).
• Beatriz G. de la Torre, Ramon Eritja, and Fernando Albericio. 4-Hydroxymethyl-3-nitrobenzoic acid. In Electronic Encyclopedia of Reagents for Organic Synthesis. (L.A. Paquette, ed.), John Wiley & Sons Ltd, Chichester, U.K., http://www3.interscience.wiley.com/cgi-bin/mrwhome/104554785/HOME (2001).
• Ernest Giralt and Fernando Albericio. Synthesis of peptides on solid supports. In Houben-Weyl. Methods of Organic Chemistry. Vol. E 22. Synthesis of Peptides and Peptidomimetics (M. Goodman, A. Felix, L. Moroder, C. Toniolo, eds.) Georg Thieme Verlag, Stuttgart, 2001, 665–671.
• Fernando Albericio and Ernest Giralt. Handles and supports. In Houben-Weyl. Methods of Organic Chemistry. Vol. E 22. Synthesis of Peptides and Peptidomimetics (M. Goodman, A. Felix, L. Moroder, C. Toniolo, eds Georg Thieme Verlag, Stuttgart, 2001, 685–709.
• Fernando Albericio and Ernest Giralt. Loading methods. In Houben-Weyl. Methods of Organic Chemistry. Vol. E 22. Synthesis of Peptides and Peptidomimetics (M. Goodman, A. Felix, L. Moroder, C. Toniolo, eds.) Georg Thieme Verlag, Stuttgart, 2001, 710–725.
• Wim Van den Nest and Fernando Albericio. The choice of the solid support. In Optimization of Solid-Phase Combinatorial Synthesis (B. Yan and A. W. Czarnik, eds.). Marcel Dekker, New York (NY, USA), 2001, 91–107.
• Beatriz G. de la Torre, Miguel A. Marcos, Ramon Eritja, and Fernando Albericio. Solid-phase peptide synthesis using N-tritylamino acids. Lett. Pepide Sci.8, 331-338 (2001).
• Dolors Fernández-Forner, Josep M. Huertas, M. Ferrer, Gaspar Casals, Hammish Ryder, Ernest Giralt, and Fernando Albericio. Solid-phase syntheses of N-substituted carbamates reaction monitoring by gel-phase 13C-NMR using 13C enriched BAL-linker. Tetrahedron Lett., 43, 3543-3546 (2002).
• Laia Crespo, Glòria Sanclimens, Miriam Royo, Fernando Albericio, and Ernest Giralt. Branched poly-proline peptides: an efficient new approach to the synthesis of repetitive sequences. Eur. J. Org. Chem., 1756-1762 (2002).
• Francesc Rabanal, Josep M. Tusell, Lluis Sastre, M. Rosa Quintero, Montse Cruz, Dolors Grillo, Miquel Pons, Fernando Albericio, Joan Serratosa, and Ernest Giralt. Structural, kinetic and cytotoxic aspects of 12-28 -amyloid protein fragment: a reappraisal. J. Peptide Sci., 8, 578-588 (2002).
• Yvonne M. Angell, Jordi Alsina, Fernando Albericio, and George Barany. Practical Protocols for Stepwise Solid-Phase Synthesis of Cysteine-Containing Peptides. J. Peptide Res., 60, 292-299 (2002).
• Miriam Royo, Josep Farrera, Laia Solé, and Fernando Albericio. Four-Dimensional Orthogonal Solid-Phase Synthesis of New Scaffolds Based in Cyclic Tetra-ß-Peptides. Tetrahedron Lett., 43, 2029-2032 (2002).
• Josep Farrera, Miriam Royo, and Fernando Albericio. Undesired removal of the Fmoc group by the free -amino function of a lysine residue. Tetrahedron Lett., 43, 7813-7815 (2002).
• Eliandre Oliveira, Eduardo M. Cilli, Antonio Miranda,Guita N. Jubilut, Fernando Albericio, David Andreu,Antonio C. M. Paiva, Shirley Schreier, Mineko Tominaga, and Clovis R. Nakaie. Monitoring the chemical assembly of a transmembrane bradykinin receptor fragment: correlation between resin solvation, peptide chain mobility and rate of coupling. Eur. J. Org. Chem. 3686-3694 (2002).
• Laia Crespo, Glòria Sanclimens, Beatriz Montaner,Pérez-Tomás, Miriam Royo, Miquel Pons, Fernando Albericio, and Ernest Giralt. Peptide dendrimers based on poly-proline helices. J. Am. Chem. Soc., 124, 8876-8883 (2002).
• Colin M. Tice, Enrique L. Michelotti, Ernesto Mata, Ernesto Nicolàs, Javier Garcia, and Fernando Albericio. Solid phase synthesis of -acylamino--disubstitutedketones. Tetrahedron Lett., 43, 7491-7494 (2002).
• Javier Garcia, Ernesto Nicolàs, Fernando Albericio, Enrique L. Michelotti, and Colin M. Tice. Combined solid and solution phase synthesis of a library of -disubstituted--acylaminoketones. Tetrahedron Lett., 43, 7495-7498 (2002).
• Jesús Vázquez and Fernando Albericio. Synthesis of Fmoc-protected aminoketones bearing tert-butyl based side-chain protecting groups. Tetrahedron Lett., 43, 7499-7502 (2002).
• Oleg Marder, Youval Shvo, and Fernando Albericio. HCTU and TCTU. New Coupling Reagents: Development and Industrial Aspects. Chemistry Today 20 (7/8), 37-41 (2002).
• Bouchaib Bahbouhi, Nathalie Chazal, Nabil Georges Seidah, Cristina Chiva, Marcelo Kogan, Fernando Albericio, Ernest Giralt, and Elmostafa Bahraoui. Effect of L- and D-REKR amino acid-containing peptides on HIV and SIV envelope glycoprotein precursor maturation and viral replication. Biochem. J. 366, 863-872 (2002).
• Rosario González-Muñiz, Guillermo Gerona-Navarro, Mª Angeles Bonache, Carlos García-Aparicio, Mercedes Martín-Martínez, Mª Teresa García-López, Miriam Royo, and Fernando Albericio. Exploring Different Approaches for the Stereoselective Synthesis of Amino Acid-derived 4-Alkyl-4-carboxy-2-azetidinones. In Peptides 2002 (E. Benedetti and C. Pedone, eds.), Edizioni Ziino, Napoli, Italy, 2002, pp. 112-113.
• Jose C. Jiménez, Bibiana Chavarría, Ángel López-Macià, Miriam Royo, Ernest Giralt, and Fernando Albericio. Tentoxin as Scaffold for Drug Discovery. Total Solid-Phase Synthesis of Tentoxin. Solid-Phase Synthesis of Tentoxin. Synthesis of a Library of Analogues. In Peptides 2002 (E. Benedetti and C. Pedone, eds.), Edizioni Ziino, Napoli, Italy, 2002, pp. 150-151.
• Glòria Sanclimens, Laia Crespo, Miquel Pons, Ernest Giralt, Fernando Albericio,and Miriam Royo. Do beads suffer stress? In Peptides 2002 (E. Benedetti and C. Pedone, eds.), Edizioni Ziino, Napoli, Italy, 2002, pp. 402-403.
• Meritxell Teixido, Ignacio Belda, Sonia González, Miriam Fabre, Senen Vilaró, Josep M. Garrell, Xavier Roselló, Fernando Albericio, and Ernest Giralt. Evolutionary combinatorial chemistry: a novel tool for SAR studies on peptide transport across the blood-brain barrier. In Peptides 2002 (E. Benedetti and C. Pedone, eds.), Edizioni Ziino, Napoli, Italy, 2002, pp. 414-415.
• Miriam Royo, Glòria Sanclimens, Laia Crespo, Miquel Pons, Fernando Albericio, and Ernest Giralt. Design and Synthesis of Dendrimers Based on Poly(Pro) Sequences. Exploration of their Use as Drug-Delivery Agents. In Peptides 2002 (E. Benedetti and C. Pedone, eds.), Edizioni Ziino, Napoli, Italy, 2002, pp. 594-595.
• Miriam Royo, Glòria Sanclimens, Laia Crespo, Miquel Pons, Fernando Albericio, and Ernest Giralt. Design and Synthesis of Dendrimers Based on Poly(Pro) Sequences. Exploration of their Use as Drug-Delivery Agents. In Peptides 2002 (E. Benedetti and C. Pedone, eds.), Edizioni Ziino, Napoli, Italy, 2002, pp. 594-595.
• Ernest Giralt, Margarida Gairí, Xavier Salvatella, Ricard Alex Rodríguez-Mias, Jose Carlos Jiménez, Angel López-Macià, Josep Maria Caba, Francisco Cárdenas, Miguel Feliz, Paul lloyd-Williams, and Fernando Albericio. Conformational Analysis of Natural Marine Cyclopeptides with Anti-Tumor Properties. In Peptides 2002 (E. Benedetti and C. Pedone, eds.), Edizioni Ziino, Napoli, Italy, 2002, pp. 758-759.
• Miriam Royo, Josep Farrera-Sinfreu, Fabio Sgarzi, Fernando Albericio, Lucca Gentilucci, and Giuliana Cardillo. Are the Stable Secondary Structures of -Isomeric Peptides Similar to those of -Peptides. In Peptides 2002 (E. Benedetti and C. Pedone, eds.), Edizioni Ziino, Napoli, Italy, 2002, pp. 870-871.
• Laura Zaccaro, Maria T. García-López, Rosario Gonzalez-Muñiz, Carlonia García-Martínez, Antonio Ferrer-Montiel, Fernando Albericio, and Miriam Royo. Solid-Phase Tryptophan Modification: Use of a Rational Combinatorial Chemistry Approach to Develop New Analgesic Drugs. In Peptides 2002 (E. Benedetti and C. Pedone, eds.), Edizioni Ziino, Napoli, Italy, 2002, pp. 1024-1025.
• Àngel López-Macia, Josep M. Caba, Jose C. Jiménez, Xavier Salvatella, Sonia Varon, Miriam Royo, Ignacio Rodriguez, Ignacio Manzanares, Ernest Giralt, Fernando Albericio. Solid-phase synthesis of marine cyclic peptides with antitumoral activity. In Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries: Peptides, Proteins and Nucleic Acids--Small Molecule Organic Chemistry Diversity, Collected Papers, International Symposium, 7th(R. Epton, ed.) Mayflower Worldwide Ltd., Kingswinford, UK, 2002, pp. 13-16.
• Jose C. Jiménez, Nuria Bayó, Bibiana Chavarría, Àngel López-Macià, Miriam Royo, Ernesto Nicolás, Ernest Giralt, and Fernando Albericio. Synthesis of Peptides Containing -Didehydroamino Acids. Scope and Limitations. Lett. Pep. Sci., 9, 135-145 (2002).
• Nuria Bayó, Jose C. Jiménez, Luis Rivas, Ernesto Nicolás, and Fernando Albericio. Solid-phase síntesis of the cyclic lipononadepsipeptide [N-Mst(Ser1), D-Ser4, L-Thr6, L-Asp8, L-Thr9]Syringotoxin. Chem. Eur. J., 9, 1096-1103 (2003).
• Xavier Salvatella, Josep Maria Caba, Fernando Albericio, and Ernest Giralt. Solution structure of the antitumour candidate Trunkamide A by 2D-NMR and restrained simulated annealing methods. J. Org. Chem., 68, 211-215 (2003).
• Colin M. Tice, Robert E. Hormann,Christine S. Thompson,Jennifer L. Friz, Caitlin K. Cavanaugh, Enrique L. Michelotti, Javier Garcia, Ernesto Nicolas, and Fernando Albericio. Synthesis and SAR of -Acylaminoketone Ligands for Control of Gene Expression.Bioorganic Medicinal Chemistry Letters, 13, 474-478 (2003).
• Cristina Chiva, Philippe Barthe, Anna Codina, Margarida Gairí, Franck Molina, Claude Granier, Martine Pugnière, Tatsuya Inui, Hideki Nishi, Yuji Nishiuchi, Terutoshi Kimura, Shumpei Sakakibara, Fernando Albericio, and Ernest Giralt. Synthesis and NMR Structure of P41icf, a Potent Inhibitor of Human Cathepsin L. J. Am. Chem. Soc., 125, 1508-1517 (2003).
• Meritxell Teixido, Ignasi Belda, Xavier Roselló, Sonia González, Miriam Fabre, Xavier Llorà, Jaume Bacardit, Josep M. Garrell, Senen Vilaró, Fernando Albericio, and Ernest Giralt. Development of a genetic algorithm to design and identify peptides that can cross the blood-brain barrier: 1. Design and validation in silico. QSAR & Combinatorial Science, 22, 745-753 (2003).
• Jesús Vázquez, Gregory Qushair, and Fernando Albericio. Qualitative Colorimetric Tests for Solid Phase Synthesis. In Methods in Enzymology, Vol. 369 (G. Morales, ed.) Academic Press, San Diego, 2003, pp. 21-35.
• Meritxell Teixido, Maria Altamura, Laura Quartara, Alessandro Giolitti, Carlo Alberto Maggi, Ernest Giralt, and Fernando Albericio. Bicyclic Homodetic Peptide Libraries: Comparison of Synthetic Strategies for their Solid-Phase Synthesis. J. Comb. Chem., 5, 760-768 (2003).
• Pablo G. Cironi, Fernando Albericio, and Mercedes Àlvarez. Total Solid-Phase Synthesis of the Pentacyclic System Lamellarins U and L. Organic Lett., 5, 2959-2962 (2003).
• Glòria Sanclimens, Laia Crespo, Miquel Pons, Ernest Giralt, Fernando Albericio,and Miriam Royo. Saturated Resins or the Stress of the Resin. Tetrahedron Lett., 44, 1751-1754 (2003).
• Jose C. Jiménez, Bibiana Chavarría, Ángel López-Macià, Miriam Royo, Ernest Giralt, and Fernando Albericio. Tentoxin as Scaffold for Drug Discovery. Total Solid-Phase Synthesis of Tentoxin. Synthesis of a Library of Analogues. Organic Lett., 5, 2115-2118 (2003).
• Guillermo Gerona-Navarro, Miriam Royo, Mª Teresa García-López, Fernando Albericio, and Rosario González-Muñiz. Exploring Solid-Phase Approaches for the Preparation of New -Lactams from Amino Acids. Molecular Diversity, 6, 75-84 (2003).
• Oscar García, Ernesto Nicolás, and Fernando Albericio. Solid-Phase Synthesis:A Linker for Side-Chain Anchoring of Arginine. Tetrahedron Lett., 44, 5319-5321 (2003).
• Oscar García, Ernesto Nicolás, and Fernando Albericio. o-Formylation of Electron-rich Phenols with Dichloromethylmethyl Ether and TiCl4. Tetrahedron Lett., 44, 4961-4963 (2003).
• Jesper Brask, Fernando Albericio, and Knud J. Jensen. Fmoc Solid-Phase Synthesis of Peptide Thioesters by Masking as Trithioortho Ester.Org. Lett., 5, 2951-2953 (2003).
• Jordi Alsina and Fernando Albericio. Solid-Phase Synthesis of C-Terminal Modified Peptides. Biopolymers (Peptide Science), 71, 454-477 (2003).
• Oleg Marder and Fernando Albericio. Industrial Applications of Coupling Reagents in Peptides. Chemistry Today 21 (6), 35-40 (2003).
• Abderaouf Ahaidar, David Fernández, Olga Pérez, Gerardo Danelón, Carmen Cuevas, Ignacio Manzanares, Fernando Albericio, John A. Joule, and Mercedes Álvarez. Synthesis of Variolin B. Tetrahedron Lett., 44, 6191-6194 (2003).
• Rosa Planells-Cases, Carolina García-Martínez, Miriam Royo, Enrique Pérez-Payá, Cristina Carreño,Fernando Albericio, Angel Messeguer, and Antonio Ferrer-Montiel. Small Molecules Targeting the Vanilloid Receptor Complex as Drugs for Inflammatory Pain. Drugs Future, 28, 787-795 (2003).
• Pilar Forns, Sara Sevilla, Montserrat Erra, Alberto Ortega,Joan-Carles Fernàndez, Natalia de la Figuera, Dolors Fernández-Forner, and Fernando Albericio. BAL resin for the preparation of secondary amines. Tetrahedron Lett., 44, 6907-6910 (2003).
• Silvia A. Camperi, Nancy B. Iannucci, G.J. Albanesi, M. Oggero, Marina Etcheverrigaray, Fernando Albericio, and Osvaldo Cascone.Monoclonal antibody purification by affinity chromatography with ligands derived from the screening of peptide combinatory libraries. Biotechnology Lett., 25, 1545-1548 (2003).
• Pablo G. Cironi, Mercedes Álvarez, and Fernando Albericio. 1H-NMR with Internal and External Standards for Quantification of Libraries. Molecular Diversity, 6, 165-168 (2003).
• AbderaoufAhaidar,David Fernández, Gerardo Danelón, Carmen Cuevas, Ignacio Manzanares, Fernando Albericio,John A. Joule, and Mercedes Álvarez. Total Syntheses of Variolin B and Deoxyvariolin B. J. Org. Chem.,68, 10020-10029 (2003).
• Javier Garcia,Blanca Martínez-Teipel,Ernesto Nicolás, David H. Young, Enrique L. Michelotti,and Fernando Albericio. Adding Diversity to Acivicine, an Antitumoral Natural Product. Synthesis and Biological Activity of a Dipeptide Library Based on Acivicine. Lett. Peptide Sci., 10, 645-653 (2003).
• Ernest Giralt, Miriam Royo, Marcelo Kogan, Laia Crespo, Glòria Sanclimens, Josep Farrera-Sinfreu, Miquel Pons, and Fernando Albericio. Proline-Rich Peptides: From Plants to Dendrimers. In 3rd Hellenic Forum on Bioactive Peptides (P.A. Cordopatis, E. Manessi-Zoupa, and G. Pairas, eds.), Typorama, Patras (Greece), 2003, pp. 53-59.
• Luis J. Cruz, E. Iglesias, Julio C. Aguilar, Luis J. González, Osvaldo Reyes, Fernando Albericio, and David Andreu. A Comparative Study of Different Presentations of a HIV Peptide Immunogen. Biooconjugate Chem., 15, 112-120 (2004).
• Pablo Cironi, Mercedes Álvarez, and Fernando Albericio. A Combination of different Spectroscopy Techniques to monitor “in situ” solid-phase synthesis of organic molecules. QSAR & Combinatorial Science, 23, 61-68 (2004).
• Thomas Bruckdorfer, Oleg Marder, and Fernando Albericio. From Production of Peptides in Milligram Amounts for Research to Multitons Quantities for Drugs of the Future. Current Pharm. Biotech., 5, 29-43 (2004).
• Abderaouf Ahaidar,David Fernández,Olga Pérez, Carmen Cuevas, Fernando Albericio, John A. Joule,and Mercedes Álvarez, Derivatives of pyrido[3´,2´:4,5]pyrrolo[1,2-c]pyrimidones. ARKIVOC, (iv) pp. 74-85 (2004).
• Josep Farrera-Sinfreu,Laura Zaccaro,David Vidal, Xavier Salvatella, Ernest Giralt, Miquel Pons, Fernando Albericio and Miriam Royo. A New Class of Foldamers Based on cis--amino-L-proline. J. Am. Chem. Soc.,126, 6048-6057 (2004).
• Pablo Cironi,Carmen Cuevas,Fernando Albericio, andMercedes Álvarez. Gaining Diversity in Solid-Phase Synthesis by Modulation of Cleavage Conditions from Hydroxymethyl Based Supports. Application to Lamellarin Synthesis. Tetrahedron, 60, 8669-8675 (2004).
• David Fernández,Abderaouf Ahaidar, Gerardo Danelón, Pablo Cironi, Marta Marfil, Olga Pérez, Fernando Albericio, John A. Joule, and Mercedes Álvarez. Synthesis of Polyheterocyclic Nitrogen-Containing Marine Natural Products. Monatshefte fuer Chemie/ Chemical Monthly, 135, 615-627 (2004).
• Francesc Yraola, Ruben Ventura, Marc Vendrell, Aina Colombo, Joan-Carles Fernàndez, Natalia de la Figuera, Dolors Fernández-Forner,Miriam Royo, Pilar Forns, and Fernando Albericio. A revaluation on the use of Rink, BAL, and PAL resins and linkers QSAR & Combinatorial Science, 23,145-152 (2004).
• Marta Marfil, Fernando Albericio, and Mercedes Álvarez. Solid Phase Synthesis of Lamellarins Q and O. Tetrahedron, 60, 8659-8668 (2004).
• Ksenia Pumpor, Elisabeth Windeisen, Jan Spengler, Fernando Albericio, and Klaus Burger. Hexafluoroacetone as a Protecting and Activating Reagent. Regioselective Esterification of Aspartic, Malic and Thiomalic Acid. Monatshefte fuer Chemie/Chemical Monthly, 135, 1427-1443 (2004).
• Fernando Albericio. Developments in peptide and amide synthesis. Current Opinion Chem. Biol., 8, 211-221 (2004).
• Jose Carlos Jiménez, Ernest Giralt, and Fernando Albericio. Péptidos y la Industria Farmacéutica. Anal. Quim., 100(1), 10-16 (2004).
• Jesús Vázquez, Miriam Royo, and Fernando Albericio. Re-evaluation of a Solid-Phase Hydantoin Synthesis. Lett. Org. Chem., 1, 224-226 (2004).
• Pablo Cironi,Judit Tulla-Puche,George Barany,Fernando Albericio,and Mercedes Álvarez. Solid-Phase Syntheses of Furopyridine and Furoquinoline Systems. Organic Lett., 6, 1405-1408 (2004).
• Pablo Cironi, Fernando Albericio, and Mercedes Álvarez. Lamellarins: Isolation, Activity and Synthesis. In Progress in Heterocyclic Chemistry. Volume 16. (G.W. Gribble and J.A. Joule, eds.) Pergamon: Oxford (UK), 2004, pp. 1-26.
• Montse Cruz, Josep M. Tusell, Dolors Grillo-Bosch, Fernando Albericio, Joan Serratosa, Francesc Rabanal, and Ernest Giralt. Inhibition of -amyloid toxicity by short peptides containing N-methyl amino acids. J. Peptide Res., 63, 324-3f28 (2004).
• Glòria Sanclimens,Laia Crespo, Ernest Giralt, Miriam Royo, and Fernando Albericio. Solid-Phase Syntheses of a Second Generation of Polyproline Dendrimers. Biopolymers (Pept. Sci.), 76, 283-297 (2004).
• Luis J. Cruz,Natalia G. Beteta, Ariel Ewenson, and Fernando Albericio. ‘One-pot’ Preparation of N-Carbamate Protected Amino Acids via the Azide. Org. Proc. Res. Develop.,8, 920-924 (2004).
• Pablo Cironi, Fernando Albericio, and Mercedes Álvarez. Solid-Phase Synthesis of 4H-2-(3-Hydroxy-4-methoxyphenyl)naphtho[1,2-b]pyran-1-one. Tetrahedron Lett., 45, 7311-7314 (2004).
• Judit Tulla-Puche, Irina V. Getun, Jordi Alsina, Fernando Albericio, and George Barany. Synthetic Circularized Analogues of Bovine Pancreatic Trypsin Inhibitor. Eur. J. Org. Chem., 4541-4544 (2004).
• Ana Montero, Fernando Albericio, Miriam Royo, and Bernardo Herradón. Solid-Phase Combinatorial Synthesis of Peptide-Biphenyl Hybrids as Calpain Inhibitors. Org. Lett.,6, 4089-4092 (2004).
• Beatriz G. de la Torre and Fernando Albericio. 2,4-Dimethoxy-4’-hydroxybenzophenone. In Electronic Encyclopedia of Reagents for Organic Synthesis. (L.A. Paquette, ed.), John Wiley & Sons Ltd, Chichester, U.K., www.mrw.interscience.wiley.com/eros/.
• Beatriz G. de la Torre and Fernando Albericio. 4-Bromomethyl-3-nitrobenzoic acid. In Electronic Encyclopedia of Reagents for Organic Synthesis. (L.A. Paquette, ed.), John Wiley & Sons Ltd, Chichester, U.K., www.mrw.interscience.wiley.com/eros/.
• Jesper Brask, Fernando Albericio, and Knud J. Jensen. Synthesis of Peptide Thioesters by Masking as Trithioortho Esters in a Fmoc Backbone Amide Linker (BAL) Strategy. In Peptide Revolution: Genomics, Proteomics & Therapeutics (M. Chorev, T.K. Sawyer, eds.), American Peptide Society, 2004, pp. 125-126.
• Jesús Vázquez and Fernando Albericio. Solid-Phase Synthesis of Amidoketones: Towards Caspase Inhibitors. In Peptide Revolution: Genomics, Proteomics & Therapeutics (M. Chorev, T.K. Sawyer, eds.), American Peptide Society, 2004, pp. 319-320.
• Josep Farrera-Sinfreu, Ernest Giralt, Miquel Pons, Susanna Castel, Fernando Albericio, and Miriam Royo. Structure-Activity Studies of cis--Amino-L-Proline Oligomers: Probing the Relationship between Conformational Stability and Cellular Internalization Capacity. In Peptide Revolution: Genomics, Proteomics & Therapeutics (M. Chorev, T.K. Sawyer, eds.), American Peptide Society, 2004, pp. 437-438.
• Meritxell Teixido, Ignasi Belda, Sonia González, Miriam Fabre, Senén Vilaró, Josep M. Garrell, Xavier Roselló, Fernando Albericio, and Ernest Giralt. Evolutionary Combinatorial Chemistry: a Novel Tool for SAR Studies on PeptideTransport Across the Blood-Brain Barrier. 1. Design, In Silico Validation and First Peptide Generation. In Peptide Revolution: Genomics, Proteomics & Therapeutics (M. Chorev, T.K. Sawyer, eds.), American Peptide Society, 2004, pp. 800-801.
• Marc Vendrell, Rubén Ventura, Fernando Albericio, Rosario González-Muñiz, Laura García-Diego, Crsitina Carreño, Antonio Ferrer-Montiel, and Miriam Royo. Minimalism Applied to a Hit to Lead Program. In Peptide Revolution: Genomics, Proteomics & Therapeutics (M. Chorev, T.K. Sawyer, eds.), American Peptide Society, 2004, pp. 831-832.
• Rubén Ventura, Marc Vendrell, Fernando Albericio, Rosario González-Muñiz, Laura García-Diego, Crsitina Carreño, Antonio Ferrer-Montiel, and Miriam Royo. Is it Possible to Minimize the Toxicity of a Hit Compound Without Reducing its Activity?. In Peptide Revolution: Genomics, Proteomics & Therapeutics (M. Chorev, T.K. Sawyer, eds.), American Peptide Society, 2004, pp. 833-834.
• MariCruz Pozo-Carrero and Fernando Albericio. Revolución Combinatoria. In Combinatoria Molecular (Nelson Santiago Vispo, ed.) Elfos Scientiae, La Habana (Cuba), 2004, pp. 1-12.
• Jordi Alsina, Steven A. Kates, George Barany, and Fernando Albericio. Backbone Amide Linker (BAL) Strategies for the Solid-Phase Synthesis of C-Terminal Modified Peptides. In Methods in Molecular Biology, vol. 298: Peptide Synthesis and Applications (Ed. John Howl), Humana Press Inc., Totowa, NJ, 2005, pp.195-208.
• Laia Crespo, Glòria Sanclimens, Miquel Pons, Ernest Giralt Miriam Royo, and Fernando Albericio. Peptide Dendrimers. Chem. Rew., 105, 1663-1681 (2005).
• Montserrat del Fresno, Dolors Fernández-Forner,Montserrat Miralpeix, Victor Segarra, Hamish Ryder,Miriam Royo,and Fernando Albericio. Combinatorial Approaches Towards the Discovery of New Tryptase Inhibitors. Bioorg. Med. Chem. Lett., 15, 1659-1664 (2005).
• Fernando Albericio, Klaus Burger, Javier Ruíz-Rodríguez, and Jan Spengler. A New Strategy for Solid Phase Depsipeptide Synthesis Using Recoverable Building Blocks. Org. Lett.,7, 597-600 (2005).
• Josep Farreras-Sinfreu, Ernest Giralt, Susanna Castel, Fernando Albericio, and Miriam Royo. Cell Penetrating cis--Amino-L-Proline Derivated Peptide. J. Am. Chem. Soc.,127, 9459-9468 (2005).
• Estela Riego, Nuria Bayó, Carmen Cuevas, Fernando Albericio, and Mercedes Álvarez. A New Approach to 3-Hydroxyquinoline-2-carboxylic Acid. Tetrahedron, 61, 1407-1411 (2005).
• Glòria Sanclimens, Hong Shen, Ernest Giralt, Fernando Albericio, Mark W. Saltzman, Miriam Royo. Synthesis and Screening of a Small Library of Proline Based Biodendrimers for Use as Delivery Agents. Biopolymers (Peptide Sci.), 80, 800-814 (2005) with cover.
• Meritxell Teixidó, Fernando Albericio, and Ernest Giralt. Solid-Phase Synthesis and Characterization of N-Methyl Rich Peptides. J. Peptide Res.,65, 153-166 (2005).
• Jan Spengler,Jose-Carlos Jiménez, Ernest Giralt, and Fernando Albericio. Abbreviated nomenclature for Cyclic and Branched Homo- and Heterodetic Peptides. J. Peptide Res., 65, 550-555 (2005).
• Javier Garcia, Robert E. Hormann, Christine S. Thompson, Jennifer L. Friz, Caitlin K. Cavanaugh, Jessica A. Saggers, Ernesto G. Mata, Ernesto Nicolas, Fernando Albericio, Enrique L. Michelotti, and Colin M. Tice. Different approaches to the synthesis of a -disubstituted--acylaminoketones library and their evaluation as ligands for control of gene expression. J. Comb. Chem., 7, 843-863 (2005).
• Klaus Burger, Gabor Radies, Lothar Henning, Christoph Böttcher, Jan Spengler, and Fernando Albericio. Orthogonally Protected, Carboxy-Activated L-Homoserine, 2-Methyl-L-homoisoserine and Homoisocysteine Derivatives, New Building Blocks for Peptide and Depsipeptide Modification. Monatshefte fuer Chemie/Chemical Monthly, 136, 763-776 (2005).
• Aina Colombo, Joan-Carles Fernàndez,Natalia de la Figuera, Dolors Fernández-Forner, Pilar Forns, and Fernando Albericio. Solid Phase preparation of a Library based on a Phenylalanine Scaffold. QSAR & Combinatorial Science, 24, 913-922 (2005).
• Christian A. Olsen,Núria Parera, Fernando Albericio, and Mercedes Álvarez. 5,6-Dihydropyrrolo[1,2-b]-isoquinolines as Scaffolds for Synthesis of Lamellarin Analogs. Tetrahedron Lett., 46, 2041-2044 (2005).
• Glòria Sanclimens, Laia Crespo,Ernest Giralt, Fernando Albericio, and Miriam Royo. A Straightforward Preparation of De Novo Globular Proteins Based on Proline Dendrimers. J. Org. Chem., 70, 6274-6281 (2005).
• Silvia A. Camperi, Mariela M. Marani, Nancy B. Iannucci, Simon Côté, Fernando Albericio,and Osvaldo Cascone. An Efficient Strategy for the Preparation of One-Bead-One-Peptide Libraries on a New Biocompatible Solid Support. Tetrahedron Lett.,46, 1561-1564 (2005).
• Klaus Burger, Lothar Hennig, Annett Fuchs, Dieter Greif, Jan Spengler, and Fernando Albericio. Domino Reactions with Fluorinated Five-membered Heterocycles - Syntheses of Trifluoromethyl Substituted Butenolides and -Ketoacids. Monatshefte fuer Chemie/Chemical Monthly, 136, 1763-1779 (2005).
• Meritxell Teixido, Ignacio Belda, Ester Zurita, Xavier Llorá, Miriam Fabre, SenenVilaró, Fernando Albericio, and Ernest Giralt. Evolutionary Combinatorial Chemistry: a Novel Tool for SAR Studies on PeptideTransport Across the Blood-Brain Barrier. 2. Design, Synthesis and Evaluation of a First Generation of Peptides. J. Peptide Sci., 11, 789-804 (2005).
• Natalia de la Figuera, Pilar Forns, Joan-Carles Fernàndez, Dolors Fernández-Forner, and Fernando Albericio. Avoiding the Undesired Opening of the Pyrane Ring during C-Glycosidation Catalyzed by Palladium Acetate. Tetrahedron Lett.,46, 7271-7274 (2005).
• Fernando Albericio, Klaus Burger, Tommaso Cupido, Javier Ruiz, and Jan Spengler. Approaches to Synergistic Connection of the Hexafluoroacetone-Route with Solid Phase Peptide Synthesis. ARKIVOC, 191-199 (2005, vi).
• Estela Riego, Delia Hernández, Fernando Albericio, and Mercedes Álvarez. Directly Linked Polyazoles: Important Moieties in Natural Products. Synthesis, 1907-1922 (2005).
• Marc Vendrell,Rubén Ventura, Ariel Ewenson, Miriam Royo, and Fernando Albericio. N-[Chloro(dimethylamino)methylene]-N-methylmethanaminium chloride (TMUCl Cl), the Reagent of Choice for the Solid-Phase Synthesis of Anilides. Tetrahedron Lett., 46, 5383-5386 (2005).
• Daniel Pla, Antonio Marchal, Christian A. Olsen, Fernando Albericio, and Mercedes Álvarez. Modular Total Síntesis of Lamellarin D. J. Org. Chem., 70, 8231-8234 (2005).
• Tommaso Cupido, Jan Spengler, Klaus Burger, Fernando Albericio. NO as Temporary Guanidino-Protecting Group: An Efficient Access to Pbf-Protected Argininic Acid. Tetrahedron Lett., 46, 6733-6735 (2005).
• Albert Isidro-Llobet, JuditGuasch-Camell, Mercedes Álvarez, and
• Sandra M. Ocampo, Fernando Albericio, Irene Fernández, Marta Vilaseca, and Ramon Eritja. A Straightforward Synthesis of 5’-Peptide Oligonucleotide Conjugates Using N-Fmoc-protected amino acids. Organic Lett., 7, 4349-4352 (2005).
• Marta Marfil, Fernando Albericio, and Mercedes Álvarez. Chloromethoxymethyl polystyrene (CMM resin), an acid labile resin for anchoring/cleavage of N-heterocycles and oxygen aromatic compounds. Lett. Org. Chem., 2, 371-373 (2005).
• Pilar E. López,Albert Isidro-Llobet,Carolina Gracia,Andrés García-Granados, Andrés Parra, Mercedes Álvarez, and Fernando Albericio.Use of p-Nitrobenzyloxycarbonyl (pNZ) as a Permanent Protecting Group in the Synthesis of Kahalalide F Analogues. Tetrahedron Lett.,46, 7737-7741 (2005).
• Albert Isidro-Llobet,Mercedes Álvarez, and Fernando Albericio p-Nitrobenzyloxycarbonyl (pNZ) as a Semipermanent Protecting Group for the Side Chain of Orn and Lys. Application for the Synthesis of Cyclic Peptides and to Avoid Undesired α-Fmoc Removal. Tetrahedron Lett.,46, 7733-7736 (2005).
• Meritxell Teixidó, Ignasi Belda, Sonia González, Myriam Fabre, Senén Vilaró, Joseph M. Garrell, Xavier Roselló, Fernando Albericio, and Ernest Giralt. Evolutionary combinatorial chemistry: a novel tool for SAR studies on peptide transport across the blood-brain barrier. 2. Design, synthesis and evaluation of the first peptide generation. In Peptides 2004 (M. Flegel, M. Fridkin, C. Gilon, and J. Slaninova, eds.), Kenes International, Geneva, Switzerland, 2005, pp. 13-14.
• Fernando Albericio, Klaus Burger, Pierre Rousselot-Pailley, Javier Ruiz, and Jan Spengler. A novel strategy for solid-phase synthesis of depsipeptides using hexafluoroacetone. In Peptides 2004 (M. Flegel, M. Fridkin, C. Gilon, and J. Slaninova, eds.), Kenes International, Geneva, Switzerland, 2005, pp. 186-187.
• Josep Farrera-Sinfreu, Ernest Giralt, Susanna Castel, Fernando Albericio, and Miriam Royo. Cell uptake properties of cis--amino-L-proline oligomers. In Peptides 2004 (M. Flegel, M. Fridkin, C. Gilon, and J. Slaninova, eds.), Kenes International, Geneva, Switzerland, 2005, pp. 539-540.
• Jesús Vázquez, Jaime Rubio, Enrique Pérez-Payá, and Fernando Albericio. Solid-phase síntesis of hydantoins as caspase inhibitors. In Peptides 2004 (M. Flegel, M. Fridkin, C. Gilon, and J. Slaninova, eds.), Kenes International, Geneva, Switzerland, 2005, pp. 686-687.
• Pablo Cironi, Mercedes Álvarez, and Fernando Albericio. Total Solid-Phase Synthesis of Non-peptidic Natural Products. Mini-reviews Med. Chem., 6, 11-25 (2006).
• Luis J. Cruz,Marta Martínez Insua, Julia Pérez Baz,Martha Trujillo, Ricard A Rodriguez-Mias, Eliandre Oliveira, Ernest Giralt, Fernando Albericio, and Librada M. Cañedo. IB-01212, A New Cytotoxic Cyclodepsipeptide Isolated from the Marine Fungus Chlonostachys pitirodes. J. Org. Chem., 71, 3335-3338 (2006) with cover.
• Luis J. Cruz,Carmen Cuevas,Librada M. Cañedo, Ernest Giralt, and Fernando Albericio.Total Solid-Phase Synthesis of the Marine Cyclodepsipeptide IB-01212. J. Org. Chem., 71, 3339-3344 (2006) with cover.
• Joan-Carles Fernàndez, Laia Solé-Feu,Dolors Fernández-Forner,Natalia de la Figuera,Pilar Forns, and Fernando Albericio Solid-phase N-electrophilic amination of 2-aminopyridines: preparation of 2-substituted-[1,2,4]triazolo[1,5-a]pyridine derivatives. QSAR & Combinatorial Science, 25, 913-922 (2006).
• Ayman El-Faham,Sherine N. Khattab,M. Abdul-Ghani,and Fernando Albericio. Design and Synthesis of a New Immonium Type Coupling Reagents. Eur. J. Org. Chem., 6, 1563-1573 (2006).
• Fayna García-Martín, Martina Quintanar-Audelo, Yésica García-Ramos, Luis J. Cruz, Catherine Gravel, RobertFuric, Simon Côté, Judit Tulla-Puche, and Fernando Albericio. ChemMatrix®, a Polyethylene glycol (PEG)-based Support for the Solid-Phase Synthesis of Complex Peptides J. Comb. Chem., 8, 213-220 (2006).
• Jesús Vázquez and Fernando Albericio. A Semicarbazide Resin for the Solid-Phase Synthesis of Peptide Ketones and Aldehydes. Tetrahedron Lett.,47, 1657-1661 (2006).
• Puig Mora, Carlos Mas-Moruno,Silvia Tamborero,Luis J. Cruz, Enrique Pérez-Payá, and Fernando Albericio. Design of a Minimized Cyclic Tetrapeptide that Neutralizes Bacterial Endotoxins. J. Peptide Sci. ,11, 1335-1342 (2006).
• Judit Tulla-Puche, Irina V. Getun, Yvonne M. Angell, Jordi Alsina, Fernando Albericio, Clare Woodward, and George Barany. Synthetic Approaches for Disulfide-Free Circular Bovine Pancreatic Trypsin Inhibitor (c-BPTI) Analogues. Int. J. Peptides Res. Therapeutics, 12, 93-104 (2006).
• Jan Spengler, Javier Ruiz-Rodriguez, Klaus Burger, and Fernando Albericio. Homologation of α-hydroxy acids to α-unsubstituted β-hydroxy carboxamides via Arndt-Eistert reaction. Tetrahedron Lett.,47, 4557-4560 (2006).
• Nuria Roqué, Pablo Cironi, Xavier Solans, Fernando Albericio, and Mercedes Álvarez. 1-Hydroxy- 6,7-Dimethoxy-8-nitro-1,2,3,4-tetrahydroisoquinoline. Acta Cryst., E62, o2285-o2287 (2006).
• Francesc Yraola, Silvia García-Vicente, Juan Fernandez-Recio, Fernando Albericio, Antonio Zorzano, Luc Marti, and Miriam Royo. 4-Phenylbutylamine as a New Efficient Substrate for Semicarbazide-Sensitive Amine Oxidase/VAP-1 Enzyme: Analysis by SARs and Computational Docking. J. Med. Chem.,49, 6197-6208 (2006).
• Natalia de la Figuera, Sandra Fiol, Pilar Forns, Joan-Carles Fernàndez, Dolors Fernández-Forner, and Fernando Albericio. Role of the acid group in the Pictet Spengler Reaction of -amino acids. SYNLETT., 1903-1907 (2006).
• Klaus Burger, Lothar Henning, P. Tsouker, Jan Spengler, Fernando Albericio, and Beathe Koksch. Synthesis of -Trifluoromethyl -Amino Acids with Aromatic, Heteroaromatic and Ferrocenyl Subunits in the Side Chain. Amino Acids, 31, 55-62 (2006).
• Carolina Gracia,Albert Isidro-Llobet,Luis J. Cruz,Osvaldo Acosta, Mercedes Álvarez, Carmen Cuevas, Ernest Giralt, and Fernando Albericio. Convergent Approaches for the Synthesis of the Antitumoral Peptide, Kahalalide F. Investigation of Orthogonal Protecting Groups. J. Org. Chem.,71, 7196-7204 (2006).
• Hortensia Rodríguez, Osnieski Martín, Estael Ochoa, Margarita Suárez, Osvaldo Reyes,Hilda Garay, Fernando Albericio,Carlos Seoane, and Nazario Martín. Solid-phase Synthesis and Structural Study of Substituted 1,4,5,6-Tetrahydro-6-oxopyridine-3-carboxylicacids. QSAR & Combinatorial Science, 25, 921-927 (2006).
• Daniel Pla, Antonio Marchal, Christian A. Olsen, Andrés Francesch, Carmen Cuevas, Fernando Albericio, Mercedes Álvarez. Synthesis and Structure–Activity Relationship Study of Potent Cytotoxic Analogs of the Marine Alkaloid Lamellarin D. J. Med. Chem.,49, 3257-3268 (2006).
• Elisabet Prats-Alonso,Fayna Garcia,Nuria Bayo,Luis J. Cruz,Mateu Pla-Roca, Josep Samitier, Abdelhamid Errachid, Fernando Albericio. Facile Solid-Phase Synthesis of Biotinylated Alkyl Thiols. Tetrahedron, 62, 6876-6881 (2006).
• Sara Sevilla,Pilar Forns, Natalia de la Figuera, Joan-Carles Fernàndez,Paul Eastwood, and Fernando Albericio. Microwave-assisted synthesis of 1,3-dihydro-[1,2,5]thiadiazolo[3,4-b]pyrazine-2,2-dioxides. Tetrahedron Lett.,47, 8603-8606 (2006).
• Jan Spengler, Christoph Böttcher, Fernando Albericio, and Klaus Burger. Hexafluoroacetone as Protecting and Activating Reagent: New Routes to Amino, Hydroxy and Mercapto Acids and their Application for Peptide, Glyco- and Depsipeptide Modification. Chem Rev., 106, 4728-4746 (2006).
• Fayna García-Martín, Peter White, René Steinauer, Simon Côté, Judit Tulla-Puche, Fernando Albericio. The Synergy of ChemMatrix Resin and Pseudoproline Building Blocks Renders Rantes, A Complex Aggregated Chemokine. Biopolymers (Peptide Science) with cover, 84, 566-575 (2006).
• Klaus Burger, Lothar Hennig, Pavel Tsouker, Jan Spengler, Fernando Albericio, and Beate Kotsch.Domino reactions with Fluoranited Five-Membered Heterocycles -Trifluoromethyl -Amino acids with Unsaturated Side-Chains. Amino Acids, 31, 427-433 (2006).
• Núria Bayó, Ariadna Fernández, Estela Riego, Judit Tulla-Puche, Carmen Cuevas, Mercedes Álvarez, and Fernando Albericio. Solid-Phase Syntheses of Azathiocoralines. Chem. Eur. J, 12, 9001-9009 (2006).
• Klaus Burger, Lothar Hennig, Jan Spengler, Fernando Albericio. Synthesis of Partially Fluorinated Heterocycles from 4,4-bis(trifluoromethyl) Substituted Hetero-1,3-dienes via C-F Bond Activation and their Application as Trifluoromethyl Substituted Building Blocks. Heterocycles, 68, 569-592 (2006).
• Aina Colombo, Fernando Albericio, Pilar Forns. Sulfoxidations in Solid Phase. Tetrahedron Asymmetry, 17, 3327-3331 (2006).
• Jan Spengler, Javier Ruíz-Rodríguez, Tommaso Cupido, Klaus Burger, and Fernando Albericio. Enhancing Atom Economy of SPS: Recoverable and Reusable Building Blocks for Depsipeptide Synthesis. In Proccedings of the 19th American Peptide Symposium. Understanding Biology Using Peptides (S.E. Blondelle, ed.), American Peptide Symposium, La Costa (CA), 2006, pp. 108-109.
• Fernando Albericio, Nuria Bayo, Silvia A. Camperi, Osvaldo Cascone, Simon Côté, Luis J. Cruz, Abdelhamid Errachid, Robert Furic, Fayna García-Martín, Yesica García-Ramos, Nancy B. Iannucci, Mariela M. Marani, Mateu Pla-Roca, Martina Quintanar-Audelo, Josep Samitier and Judit Tulla-Puche. Solid-Phase Peptide Synthesis Using ChemMatrix®, a Polyethylenglycol (PEG)-based Solid. In Proccedings of the 19th American Peptide Symposium. Understanding Biology Using Peptides (S.E. Blondelle, ed.), American Peptide Symposium, La Costa (CA), 2006, pp. 114-115.
• Albert Isidro-Llobet, Pilar E. López, Judit Guasch-Camell, Mercedes Álvarez, and Fernando Albericio. p-Nitrobenzyloxycarbonyl (pNZ) as an Alternative to Fmoc for the Protection of Amines in Solid-Phase Peptide Synthesis. In Proccedings of the 19th American Peptide Symposium. Understanding Biology Using Peptides (S.E. Blondelle, ed.), American Peptide Symposium, La Costa (CA), 2006, pp. 116-117.
• Jan Spengler, José-Carlos Jiménez, Klaus Burger, Ernest Giralt and Fernando Albericio. New Nomenclature for Complex Cyclopeptides. In Proccedings of the 19th American Peptide Symposium. Understanding Biology Using Peptides (S.E. Blondelle, ed.), American Peptide Symposium, La Costa (CA), 2006, pp. 142-143.
• Luiz J. Cruz, Marta Martínez, Julia Pérez, Marta Trujillo, Librada M. Cañedo, Ricard Rodríguez, Ernest Giralt and Fernando Albericio. Total Solid Phase Synthesis of a Marine Cyclodepsipeptide IB-01212. In Proccedings of the 19th American Peptide Symposium. Understanding Biology Using Peptides (S.E. Blondelle, ed.), American Peptide Symposium, La Costa (CA), 2006, pp. 210-211.
• Fayna García-Martín, Nuria Bayo, Luis J. Cruz, James Bohling and Fernando Albericio. Chlorotrityl Chloride (CTC) Resin as a Convenient Reusable Protecting Group. In Proccedings of the 19th American Peptide Symposium. Understanding Biology Using Peptides (S.E. Blondelle, ed.), American Peptide Symposium, La Costa (CA), 2006, pp. 220-221.
• Josep Farrera-Sinfreu, Ernest Giralt, Miriam Royo, and Fernando Albericio. Cell Penetrating Proline Rich Peptidomimetics. In Methods in Molecular Biology, vol. 386: Peptide Characterization and Applications Protocols (Ed. Gregg Fields), Humana Press Inc., Totowa, NJ, 2007, pp. 241-267.
• Josep Farrera-Sinfreu,Ernest Giralt, Miriam Royo, and Fernando Albericio. Cell-penetrating cis-γ-amino-L-proline derived peptides. In Handbook of Cell Penetrating Peptides, 2nd edition (U. Langel, ed.), CRC press, Boca Raton (FL), 2007, pp. 61-75.
• Ana Montero, Fernando Albericio, Miriam Royo, and Bernardo Herradón. Synthesis of macrocyclic peptide-biphenyl hybrids. Eur. J. Org. Chem.,pp. 1301-1308 (2007).
• Silvia García-Vicente, Francesc Yraola, Luc Marti, Elena González-Muñoz, M. Jose García-Barrado, Carles Canto, Anna Abella, Sandy Bour, Rafael Artuch, Cristina Sierra, Nuria Brandi, Christian Carpéné, Julio Morations, Marta Camps, Manuel Palacín, Xavier Testar, Anna Guma, Fernando Albericio, Miriam Royo, Alec Mian, and Antonio Zorzano. Oral Insulin-mimetic compounds that act independently of insulin. Diabetes, 56, 486-493 (2007).
• Cecilia Portela, Ramón Eritja, Fernando Albericio, and José L. Mascareñas. Ds-Oligonucleotide-Peptide Conjugates Featuring Peptides from the Leucine Zipper Region of FOS as Switchable Receptors for the Oncoprotein Jun. Towards the Development of Selective Receptors for Transcription Factor Components. ChemBiochem., 8, 1110-1114 (2007).
• Delia Hernandez,Estela Riego, Gemma Vilar, Andrés Francesch, Carmen Cuevas,Fernando Albericio,Mercedes Álvarez. Synthesis of IB-01211. A Cyclic Peptide Containing 2,4-Concatenated Thia- and Oxazoles. Org. Lett., 9, 809-811 (2007).
• Klaus Burger, Brigitte Helmreich, Lothar Henning, Jan Spengler, Fernando Albericio, Annett Fuchs. Partially Fluorinated Heterocycles from 4,4-Bis(trifluoromethyl)-hetero-1,3-dienes via C-F Bond Activation. Monatshefte fuer Chemie/Chemical Monthly, 138, 227-236 (2007).
• Josep Farrera-Sinfreu, Fernando Albericio, and Miriam Royo. Solid-Phase Synthesis of Sulfamate Peptidomimetics. J. Comb. Chem., 9, 501-506 (2007).
• Daniel Pla, Fernando Albericio, and Mercedes Álvarez. Efficient regioselective Monobromination of Highly Activated Benzenes. Eur. J. Org. Chem., pp. 1921-1924 (2007).
• Carlos Mas-Moruno, Luis J. Cruz, Puig Mora,Angel Messeguer, Enrique Pérez-Payá, Fernando Albericio. The Smallest Peptoids with Anticancer Activity. J. Med. Chem., 50, 2443-2449 (2007).
• Albert Isidro-Llobet, Mercedes Alvarez, Klaus Burger, Jan Spengler, Fernando Albericio. p-Nitromandelic Acid (Pnm) as Highly Acid Stable Safety-Catch Linker for Solid Phase Synthesis of Peptide and Depsipeptide Acids. Org. Lett., 9, 1429-1432 (2007).
• Francesc Yraola, Fernando Albericio, and Miriam Royo. Inhibition of VAP1: Quickly Gaining Ground as an Anti-inflammatory Therapy. ChemMedChem., 2, 173-174 (2007).
• Judit Tulla-Puche, Núria Bayó-Puxan, Juan A. Moreno, Andrés M. Francesch, Carmen Cuevas, Mercedes Álvarez, and Fernando Albericio. Solid-Phase Synthesis of Oxathiocoraline by a Key Intermolecular Disulfide Dimer. J. Am. Chem. Soc., 129, 5322-5323 (2007).
• Mariela M. Marani,Marta Paradís, Judit Tulla-Puche, Simón Côte, Silvia Camperi, Osvaldo Cascone, and Fernando Albericio. From one-bead-one-compound concept to one-bead-one-reactor. J. Comb. Chem.,9, 395-398 (2007).
• Roger Soley,Fernando Albericio, Mercedes Álvarez. Novel Synthesis of Bisaryl Acetylenes. Synthesis¸ pp. 1559-1565 (2007).
• Marcelo J Kogan, Ivonne Olmedo, Leticia Hosta, Ariel R. Guerrero, Luis J. Cruz, Fernando Albericio. Peptides and Metallic Nanoparticles For Biomedical Applications. Nanomedecine, 2, 287-306 (2007).
• Núria Bayó-Puxan, Ariadna Fernández, Judit Tulla-Puche, Estela Riego, Mercedes Álvarez,and Fernando Albericio. BeyondAzathicoraline Síntesis. Synthesis of Analogues. Int. J. Peptide Res. Therapeutics, 13, 205-306 (2007).
• Carina M.L. Delpiccolo,Fernando Albericio,Robert A. Schiksnis, Enrique L. Michelotti. Formation of Dihydrouracils via Cyclization of N-Substituted 3-Thioureidopropanoic Acids and Facile Desulfurization. Tetrahedron,63¸8949-8953 (2007).
• Silvia Frutos, Judit Tulla-Puche, Fernando Albericio, and Ernest Giralt. Chemical Synthesis of 19F-labeled HIV-1 Protease Using Fmoc-Chemistry and ChemMatrix Resin. Int. J. Peptide Res. Therapeutics, 13, 221-227 (2007).
• Fayna García-Martín,Núria Bayó-Puxan, Luis J. Cruz, James C. Bohling,and Fernando Albericio. .Chlorotrityl Chloride (CTC) Resin as a Convenient Reusable Protecting Group. QSAR &Comb. Sci. 26, 1027-1035 (2007)s.
• Luis J. Cruz,Andres Francesch,Carmen Cuevas, and Fernando Albericio. Synthesis and Structure-Activity Relationship of Novo Cytotoxic Marine Cyclodepsipeptide IB-01212 Analogs. ChemMedChem., 2, 1076-1084 (2007).
• Meritxell Teixidó, Josep M. Caba, Roger Prades, Esther Zurita, Marc Martinell, Marta Vilaseca, Fernando Albericio, and Ernest Giralt. Does the solid-phase synthesis of a tetrapeptide represent a challenge at the onset of the XXI century? The case of cyclo(3R)-3-hydroxydecanoyl-L-seryl-(3R)-3-hydroxydecanoyl-L-seryl]. Int. J. Peptide Res. Therapeutics, 13, 313-327 (2007).
• Albert Isidro-Llobet, Xavier Just-Baringo, Ariel Ewenson, Mercedes Álvarez, and Fernando Albericio. Fmoc-2-Mercaptobenzothiazole, for the Introduction of the Fmoc Moiety Free of Side-Reactions. Biopolymers (Peptide Science), 88, 733-737 (2007).
• Lidia Feliu, Patricia Vera-Luque, Fernando Albericio, and Mercedes Álvarez. Advances in Solid-Phase Cycloadditions for Heterocyclic Synthesis. J. Comb. Chem.,9, 521-565 (2007).
• Aina Colombo,Natalia de la Figuera, Joan-Carles Fernàndez,Dolors Fernández-Forner,Fernando Albericio,and Pilar Forns.A Nonacid Degradable Linker for Solid-Phase Synthesis.Organic Lett., 9, 4319-4322 (2007).
• Francesc Yraola, Silvia García-Vicente, Luc Marti, Fernando Albericio, Antonio Zorzano, and Miriam Royo.Understanding the mechanism of action of the novel SSAO substrate (C7NH10)6(V10O28)• 2H2O, a prodrug of peroxovanadate insulin mimetics. Chem. Biol. Drug Design, 49, 423-428(2007).
• Jessica A. Scheike, Carsten Baldauf, Jan Spengler, Fernando Albericio, M. Teresa Pisabarro, Beate Koksch. Amide-to-ester substitution in coiled coils: the effect of removing hydrogen bonds on protein structure.Angew. Chem. Int. Ed. 46, 7766-7769 (2007).
• Marc Vendrell, Ester Angulo, Vicent Casado, Carme Lluis, Rafael Franco, Fernando Albericio, Miriam Royo. Novel Ergopeptides as Dual Ligands for Adenosine and Dopamine Receptors.J. Med. Chem., 50, 3062-3069 (2007).
• Ayman El-Faham, Fernando Albericio. Novel Proton Acceptor Immonium-Type Coupling Reagents: Application in Solution and Solid Phase Peptide Synthesis. Org. Lett.,9, 4475-4477 (2007).
• Delia Hernández, Estela Riego,Andrés Francesch, Carmen Cuevas, Fernando Albericio, Mercedes Álvarez. Preparation of penta-azole containing cyclopeptides: challenges in macrocyclization. Tetrahedron, 63, 9862-9870 (2007).
• Gilmer Vanegas, Wilfredo Quiñones, Cesar Carrasco-López, Juan Luis Concepción, Fernando Albericio, Luisana Avilán. Enolase as a plasminogen binding protein in Leishmania Mexicana. Parasitology Res., 101, 1511-1516 (2007).
• Mariela M. Marani, Eliandre Oliveira, Simón Côte, Silvia A. Camperi, Fernando Albericio, Osvaldo Cascone. Identification of protein-binding peptides by direct MALDI-TOF-MS analysis of peptide beads selected from the screening of one-bead-one peptide combinatorial libraries. Anal. Biochem., 370, 215-222 (2007).
• Tommaso Cupido, Judit Tulla-Puche, Jan Spengler, Fernando Albericio. The synthesis of naturally occurring peptides and their analogs. Curr. Opin. Drug Discover Develop., 10, 768-783 (2007).
• Cecilia Portela, José Luis Mascareñas, Fernando Albericio, Stefania Mazzini, Clara Caminal, Roger Ramos, Sandra M. Ocampo, Ramon Eritja. New developments on the synthesis of oligonucleotide-peptide conjugates. Nucleosides, Nucleotides & Nucleic Acids, 26, 963-967 (2007).
• Martina Quintanar-Audelo,Asia Fernández-Carvajal, Wim Van Den Nest, Cristina Carreño, Antonio Ferrer-Montiel, Fernando Albericio.Design and Synthesis of Indole-Based Peptoids as Potent Noncompetitive Antagonists of Transient Receptor Potential Vanilloid 1.J. Med. Chem., 50, 6133-6143 (2007).
• Jan Spengler,Beate Koksch,Fernando Albericio. A Simple Machine-Assisted Protocol for Solid-Phase Synthesis of Depsipeptides. Biopolymers (Peptide Sci.)., 88, 823-828 (2007).
• Angela G. Torres, Ernest Giralt, Fernando Albericio, and Miriam Royo. New Synthetic Approaches to Proline-Based Dendrimers. In Peptide 2006, Proceedings of the 29th Euroepan Peptide Symposium. (K. Rolka, P. Rekowski, J. Silberring, eds.), Kenes International, Geneva (Switzerland), 2007, pp. 272-273.
• Jan Spengler, Javier Ruiz-Rodriguez, Francesc Yraola, Miriam Royo, Manfred Winter, Klaus Burger, and Fernando Albericio. Hexafluoroacetone as a versatile Protecting/Activating Reagent for Beta-Hydroxy Acids, Serine, and Threonine. In Peptide 2006, Proceedings of the 29th Euroepan Peptide Symposium. (K. Rolka, P. Rekowski, J. Silberring, eds.), Kenes International, Geneva (Switzerland), 2007, pp. 320-321.
• Martina Quintanar-Audelo, Laura Garcia de Diego, Wim Van Den Nest, Cristina Carreño, Antonio Ferrer-Montiel, and Fernando Albericio. Solid phase synthesis of arginine based peptoids as inhibitors of TRPV1 Chanel. In Peptide 2006, Proceedings of the 29th Euroepan Peptide Symposium. (K. Rolka, P. Rekowski, J. Silberring, eds.), Kenes International, Geneva (Switzerland), 2007, pp. 510-511.
• Fayna Garcia-Martin, Peter White, René Steinauer, Simon Cote, Judit Tulla-Puche, and Fernando Albericio. The Challenging of Synthesizing Complex Peptides: the Synergy between ChemMatrix resin and Pseudo-Proline Building Blocks. In Peptide 2006, Proceedings of the 29th Euroepan Peptide Symposium. (K. Rolka, P. Rekowski, J. Silberring, eds.), Kenes International, Geneva (Switzerland), 2007, pp. 752-753.
• Luis J. Cruz, Enrique Iglesias, Julio C. Aguilar, Luis J. Gonzalez, Osvaldo Reyes, Fernando Albericio, and David Andreu. Comparison of the Antibody Response in Mice Immunized with Different Presentations of JY1 Peptide. In Peptide 2006, Proceedings of the 29th Euroepan Peptide Symposium. (K. Rolka, P. Rekowski, J. Silberring, eds.), Kenes International, Geneva (Switzerland), 2007, pp. 792-793.
• Stefania Mazzini, Fayna García-Martin, Margarita Alvira, Anna Aviñó, Brendan Manning, Fernando Albericio, Ramon Eritja. Synthesis of Oligonucleotide Derivatives Using ChemMatrix Supports. Chemisty and Biodiversity, 5, 209-218 (2008).
• Eleonora Marcucci, Núria Bayó-Puxan, Judit Tulla-Puche, Jan Spengler, and Fernando Albericio. Cysteine-S-trityl a key derivative to prepare N-methyl cysteines J. Comb. Chem., 10, 69-78 (2008).
• Francesc Yraola, Fernando Albericio, Montserrat Corbella, Miriam Royo. [{Cu(pzPh)(Opo)}2Cl)2]: A New Dinuclear Copper(II) Complex with Chloride Bridge and Mixed Blocking Ligands: Inorg. Chim. Acta, 361, 2455-2461 (2008).
• Aina Colombo,Joan-Carles Fernàndez,Dolors Fernández-Forner,Natalia de la Figuera, Fernando Albericio, and Pilar Forns. Stereomeric Studies in the Oxidation and Alkylation of 4-Thiazolidinones. Tetrahedron Lett., 49, 1569-1572 (2008).
• Josep Farrera-Sinfreu, Yaiza Español, Renaud Geslain, Tanit Guitart, Fernando Albericio, Lluís Ribas de Pouplana, and Miriam Royo. Solid-Phase Combinatorial Synthesis of a Lysyl-tRNA Synthetase (LysRS) Inhibitory Library. J. Comb. Chem.,10, 391-400 (2008).
• Francesc Yraola, Fernando Albericio, Miriam Royo, and Xavier Solans. Crystal Structure of Hexaquis(4-fluorophenethylamonium) decavanadate (V) tetrahydrate, (C8H11FN)6[V10O28] • 4H2OZ. Kristallogr. NCS, 223, 45-47(2008).
• Natalia de la Figuera,Sandra Fiol,Joan-Carles Fernández,Pilar Forns,Dolors Fernández-Forner,and Fernando Albericio.A 6H-Pyran-3-one Scaffold derived from a C-Glycoside. Lett. Org. Chem., 5, 374-378 (2008).
• Fernando Albericio, Per I Arvidson, Krishna Bisetty, Ernest Giralt, Thavendran Govender, Samuel Jali, Palangpon Kongsaeree, Hendrik G Kruger, and Samram Prabpai. Trishomocubane amino acid as a -turn scaffold. Chem. Biol. Drug Design, 71, 125-130 (2008).
• Jan Spengler, Javier Ruíz-Rodríguez, Francesc Yraola, Miriam Royo, Manfred Winter, Klaus Burger, Fernando Albericio. A Novel Protecting/Activating Strategy for β-Hydroxy Acids and its Use in Convergent Peptide Synthesis. J. Org. Chem., 73, 2311-2314 (2008).
• Ayman El-Faham and Fernando Albericio. Morpholine-Based Immonium and Halogenoamidinium Salts as Coupling Reagents in Peptide Synthesis.J. Org. Chem., 73, 2731-2737 (2008).
• Jan Spengler andFernando Albericio. Asymmetric Synthesis of α-Unsubstituted β-Hydroxy Acids. Curr. Org. Chem., 5, 151-161 (2008).
• Daniel Pla, Fernando Albericio, and Mercedes Álvarez. Recent Advances in Lamellarin Alkaloids: Isolation, Synthesis and Activity. Anti-Cancer Ag. Med. Chem., 8, 746-760 (2008).
• Laura Cascales, Carles Mas-Moruno Silvia Tamborero, José Luis Aceña, Juan F. Sanz, Santos Fustero, Luis J. Cruz , Puig Mora, Fernando Albericio, and Enrique Pérez-Payá.Tiratricol neutralizes bacterial endotoxins and reduces lipopolysaccharide-induced TNF-alpha production in the cell. Chem. Biol. Drug Design, 72, 320-328 (2008).
• Jesús Vázquez,Alicia Garcia-Jareño,Laura Mondragón, Jaime Rubio,Enrique Pérez-Payá,and Fernando Albericio. Conformationally Restricted Hydantoin-Based Peptidomimetics as Inhibitors of Caspase-3 with Basic Groups allowed at the S3 Enzyme Subsite. ChemMedChem., 3, 979-985 (2008).
• Carlos Mas-Moruno, Laura Cascales, Luis J. Cruz, Puig Mora, Enriqe Pérez-Payá, and Fernando Albericio. Nanostructure formation enhances the activity of LPS-neutralizing peptides. ChemMedChem, 3, 1748-1755 (2008); with cover.
• Fayna Garcia-Martin, Luis J. Cruz, Ricard A. Rodriguez-Mias, Ernest Giralt,and Fernando Albericio. Design and Synthesis of FAJANU: a de novo C2 symmetric cyclopeptide family. J. Med. Chem., 51, 3194-3202 (2008).
• Albert Isidro-Llobet,Mercedes Álvarez,and Fernando Albericio.Phenyl-EDOTn derivatives as super acid labile carboxylic acid protecting groups for peptide síntesis. Tetrahedron Lett., 49, 3304-3307 (2008).
• Ayman El-Faham, Mercedes Armand-Ugon, Jose A. Este, and Fernando Albericio. Use of N-Methylpiperazine for the Preparation of Piperazine-Based Unsymmetrical Bis-Ureas as Anti-HIV Agents. ChemMedChem., 3, 1034-1037 (2008).
• Judit Tulla-Puche, Eleonora Marcucci, Manuel Fermin, Núria Bayó-Puxan, and Fernando Albericio. Protection by Conformationally Restricted Mobility: First Solid-Phase Synthesis of Triostin A. Chem. Eur. J. 14, 4475-4478 (2008).
• José C. Jiménez,Angel López-Macià,Carol Gracia,Sonia Varón, Marta Carrascal, Josep M. Caba,Miriam Royo,Andrés M. Francesc, Carmen Cuevas, Ernest Giralt,and Fernando Albericio. Structure-Activity Relationship (SAR) of Kahalalide F synthetic analogues. J. Med. Chem, 51, 4920-4931 (2008).
• Anna Aviñó, Isabel Navarro, Josep Farrera-Sinfreu, Miriam Royo, Juan Aymamí, Antonio Delgado,Amadeu Llebaria, Fernando Albericio,and Ramon Eritja. Solid-Phase Synthesis of Oligomers Carrying Several Chromophore Units Linked by Phosphodiester Backbones. Bioorg. Med. Chem Lett., 18, 2306-2310 (2008).
• Josep Farrera-Sinfreu, Anna Aviñó, Isabel Navarro, Juan Aymamí, Natàlia G. Beteta, Sònia Varón, Ricardo Pérez-Tomás, Wilmar Castillo-Avila, Ramon Eritja, Fernando Albericio, and Miriam Royo. Design, Synthesis and Antiproliferative Properties of Oligomers with Chromophore Linked by Amide Backbones. Bioorg. Med. Chem Lett., 18, 2440-2444 (2008).
• Albert Isidro-Llobet, Ulrik Boas,Knud J. Jensen, Mercedes Álvarez, and Fernando Albericio. THAL, a Sterically Unhindered Linker for the Solid-Phase Synthesis of Acid Sensitive Protected Peptide Acids. J. Org. Chem., 73, 7342-7344 (2008).
• Delia Hernandez,Estela Riego, Fernando Albericio, and Mercedes Álvarez.Synthesis of Natural Product Derivatives Containing 2,4-Concatenated Oxazoles. Eur. J. Org. Chem., 3389-3396 (2008).
• Fernando Albericio and Judit Tulla-Puche. The (Classic Concept of) Solid Support. InThe Power of Functional Resins in Organic Chemistry (J. Tulla-Puche, F. Albericio, eds.) Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim (Germany), 2008, pp.3-14.
• Judit Tulla-Puche and Fernando Albericio. Peptides. InThe Power of Functional Resins in Organic Chemistry (J. Tulla-Puche, F. Albericio, eds.) Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim (Germany), 2008, pp. 495-527.
• Fernando Albericio, Matthieu Giraud, Myriam Gongora-Benitez, Marta Paradis-Bas, Oleg Werbitzky. Solid-Phase Synthesis of the Cys-Rich Peptide Linaclotide. In Peptides 2008. Chemistry of Peptides in Life Science Technology and Medicine. Proceedings of the Thirtieth European Peptide Symposium (H. Lankinen, J. Vallivirta, T. Strandin, and J. Hepojoki, eds.) Finsih Peptide Society and The European Peptide Society, 2008, pp. 88-89.
• Ramon Subirós-Funosas, Ayman El-Faham, Fernando Albericio. A Potent and Non-Explosive Substituent for the Classical Benzotriazole-based Additives: Oxyma Pure. In Peptides 2008. Chemistry of Peptides in Life Science Technology and Medicine. Proceedings of the Thirtieth European Peptide Symposium (H. Lankinen, J. Vallivirta, T. Strandin, and J. Hepojoki, eds.) Finsih Peptide Society and The European Peptide Society, 2008, pp. 120-121.
• Ayman El-Faham, Ramon Subirós-Funosas, Fernando Albericio. A Non-Explosive Replacement for Benzotriazole Based Coupling Reagents. In Peptides 2008. Chemistry of Peptides in Life Science Technology and Medicine. Proceedings of the Thirtieth European Peptide Symposium (H. Lankinen, J. Vallivirta, T. Strandin, and J. Hepojoki, eds.) Finsih Peptide Society and The European Peptide Society, 2008, pp. 128-129.
• Athanassios S. Galanis, Fernando Albericio, Morten Grøtli. Enhanced microwave assisted on-bead disulfide bond formation: Synthesis of α-Conotoxin MII. In Peptides 2008. Chemistry of Peptides in Life Science Technology and Medicine. Proceedings of the Thirtieth European Peptide Symposium (H. Lankinen, J. Vallivirta, T. Strandin, and J. Hepojoki, eds.) Finsih Peptide Society and The European Peptide Society, 2008, pp. 162-163.
• Athanassios S. Galanis, Fernando Albericio, Morten Grøtli. Solid-phase peptide synthesis in aqueous environment using microwave assistance heating. In Peptides 2008. Chemistry of Peptides in Life Science Technology and Medicine. Proceedings of the Thirtieth European Peptide Symposium (H. Lankinen, J. Vallivirta, T. Strandin, and J. Hepojoki, eds.) Finsih Peptide Society and The European Peptide Society, 2008, pp. 164-165.
• Carlos Mas-Moruno, Laura Cascales, Luis J. Cruz, Puig Mora, Enriqe Pérez-Payá, and Fernando Albericio. N-acylation of anti-LPS peptides renders micellar and tubular nanoestructures with enhaced LPS-neutralizing activity. In Peptides 2008. Chemistry of Peptides in Life Science Technology and Medicine. Proceedings of the Thirtieth European Peptide Symposium (H. Lankinen, J. Vallivirta, T. Strandin, and J. Hepojoki, eds.) Finsih Peptide Society and The European Peptide Society, 2008, pp. 218-219.
• Delia Hernández,Marta Altuna, Carmen Cuevas, Rosa Aligué, Fernando Albericio, and Mercedes Álvarez. Synthesis and Antitumor Activity of MechercharmycinA Analogues.J. Med. Chem., 51, 5722-5730 (2008).
• Judit Tulla-Puche, Ángela Torres, Pilar Calvo, Miriam Royo, and Fernando Albericio. N,N,N',N'-Tetramethylchloroformamidinium hexafluorophosphate (TCFH), a powerful coupling reagent for bioconjugation. Bioconjugate Chem., 19, 1968-1971 (2008).
• Ramon Subiros-Funosas, Juan A. Moreno, Núria Bayó-Puxan, Khalil Abu-rabeah, Ariel Ewenson, and Fernando Albericio. PyCloc, the phosphonium salt derived from Cl-HOBt. Chem. Today, 26/4, 10-12 (2008).
• Fayna García-Martin and Fernando Albericio. Solid Supports for the Synthesis of Peptides. From first used resin to the most sophisticated in the market. Chem. Today, 26/4, 29-34 (2008).
• Natalia de la Figuera,Sandra Fiol,Joan-Carles Fernández,Pilar Forns,Paul Eastwood,and Fernando Albericio. Solid-phase preparation of 1,3-disubstituted imidazole derivatives. QSAR & Comb. Sci., 27¸ 1267-1273 (2008).
• Albert Isidro-Llobet, Xavier Just-Baringo, Mercedes Alvarez, and Fernando Albericio. EDOTn and MIM, new peptide backbone protecting groups.Biopolymers (Peptide Sci.)90, 444-449 (2008).
• Leticia Hosta, Mateu Pla-Roca, Jordi Arbiol, Carmen López-Iglesias, Josep Samitier, Luis J. Cruz, Marcelo Kogan, Fernando Albericio. Conjugation of Kahalalide F with gold nanoparticles to enhance in vitro antitumoral activity. Bioconjuagte Chem., 20, 138-146 (2009).
• Mariela M. Marani, María C. Martínez Ceron, Silvana L. Giudicessi, Eliandre de Oliveira, Simon Côté, Rosa Erra-Balsells, Fernando Albericio, Osvaldo Cascone, and Silvia A. Camperi.Screening of one-bead-one-peptide combinatorial library using red fluorescent dyes. Presence of positive and false positive beads. J. Comb. Chem., 11, 146-150 (2009).
• Andres Parra, Francisco Rivas, Pilar E. Lopez, Andres Garcia-Granados, Antonio Martinez, Fernando Albericio, Nieves Marquez, Eduardo Muños. Solution- and solid-phase síntesis and anti-HIV activity of maslinic acid derivatives containing amino acids and peptides. Bioorg. Medic. Chem. 17, 1139-1145 (2009).
• Judit Tulla-Puche, Eleonora Marcucci, Elisabet Prats-Alfonso, Núria Bayó-Puxan, and Fernando Albericio. NMe Amide as Synthetic Surrogate for the Thioester Moiety in Thiocoraline. J. Med. Chem., 52, 834-839 (2009).
• Athanassios S. Galanis, Fernando Albericio, and Morten Grøtli. Enhanced Microwave Assisted On-Bead Disulfide Bond Formation Method. Synthesis of –Conotoxin MII. Biopolymers (Peptide Sci)., 92, 23-34 (2009).
• Carles Ayats, Roger Soley, Fernando Albericio, and Mercedes Álvarez. Synthesis of the Pyrrolo[2,3-c]carbazole Core of the Dictyodendrins. Org. Biomol. Chem, 7, 860-862 (2009).
• Francesc Yraola, Antonio Zorzano, Fernando Albericio, and Miriam Royo. Structure-Activity Relationship of SSAO/VAP-1 Arylalkylamine Based Substrates. ChemMedChem, 4, 495-503 (2009).
• Ayman El-Fahm and Fernando Albericio. Synthesis and Applications of N-Hydroxylamine Derivatives as Potential Replacement for HOBt. Eur.J. Org. Chem. 1499-1501 (2009).
• Albert Isidro-Llobet, Mercedes Álvarez, and Fernando Albericio. Amino Acids Protecting Groups. Chem. Rev., 109, 2455-2504 (2009).
• Luis J. Cruz, Juan R. Luque-Ortega, Luis Rivas, Fernando Albericio. Structure-activity relationship of Kahalalide F and its analogs as anti-leishmanial agents. Molec. Pharmac., 6, 813-824 (2009).
• Daniel Pla, Andy Sischka, Fernando Albericio, Mercedes Alvarez, Xavier Fernàndez-Busquets, and Dario Anselmetti. Optical Tweezers Study of Topoisomerase Inhibtion. Small, 51, 1269-1272 (2009).
• Vera Martos, Pilar Castreño, Miriam Royo, Fernando Albericio, Javier de Mendoza. Solid phase synthesis of chiral bicyclic guanidinium oligomers. J. Comb. Chem.,11, 410-421 (2009).
• Albert Isidro-Llobet,Daniel Latassa, Matthieu Giraud, Mercedes Álvarez,and Fernando Albericio.1,2-Dimethylindole-3-sulfonyl (MIS), the Most Acid-LabileSulfonyl-Protecting Group for the Side Chain of Arginine. Org. Biomol. Chem, 7, 2565-2569 (2009).
• Daniel Pla,Pilar Calvo, Andrés Francesch, Carmen Cuevas, Rosa Aligué, Fernando Albericio,and Mercedes Álvarez.Lamellarin D Bioconjuagtes I: Synthesis and Cellular Internalization of PEG Conjugates. Bioconjugate Chem.,20, 1100-1111 (2009).
• Daniel Pla,Marc Martí, Josep Farrera-Sinfreu,Daniel Pulido, Pilar Calvo, Andrés Francesch, Carmen Cuevas, Miriam Royo, Rosa Aligué, Fernando Albericio,Mercedes Álvarez.Lamellarin D Bioconjuagtes II: Synthesis and Cellular Internalization of Dendrimer- and NLS-Derivatives. Bioconjugate Chem.,20, 1112-1121 (2009).
• Núria Bayó-Puxan, Judit Tulla-Puche, and Fernando Albericio. Oxathiocoraline: Lessons to Be Learnt in the Synthesis of Complex N Methylated Depsipeptides. Eur. J. Org. Chem,pp. 2957-2974 (2009).
• Aikaterini A. Zompra, Athanassios S. Galanis, Oleg Werbitzky, Fernando Albericio. Preparation of Peptides as Active Pharmaceutical Ingredients (API). Future Med.Chem., 1, 361-377 (2009).
• Ramon Subirós-Funosas,Rafel Prohens,Rafael Barbas,Ayman El-Faham, Fernando Albericio. Oxyma: an efficient additive for peptide synthesis to replace benzotriazole-based HOBt and HOAt with a lower risk of explosion. Chem.Eur. J. 15, 9394-9403 (2009).
• Ayman El-Faham, Ramon Subirós-Funosas,Rafel Prohens,Fernando Albericio.COMU, A Safer and More Effective Replacement for Benzotriazole Based Uronium Coupling Reagents. Chem.Eur. J.15, 9404-9416 (2009).
• Gerardo A. Acosta, Montserrat del Fresno, Marta Paradis-Bas, Maria Rigau-deLlobet, Simon Côté, Miriam Royo, Fernando Albericio.Solid-Phase Peptide Synthesis using Acetonitrile as a Solvent in Combination with PEG-based Resins. J. Peptide Sci., 15, 629-633 (2009).
• Daniel Pla, Keith Mills, John A. Joule, Fernando Albericio, and Mercedes Álvarez. The synthesis of 1,2,3,6,6a,7-hexahydro-7-methyl-5-imino-1H-pyrrolo[1,2-c]imidazolo[5,4-b]indole. ARKIVOC, 260-269 (2009).
• Marc Vendrell,Aroa Soriano, Vicent Casadó, José Luis Díaz, Rodolfo Lavilla, Enric I. Canela, Carme Lluis, Rafael Franco, Fernando Albericio, Miriam Royo. Indoloquinolizidine-Peptide Hybrids as Novel Multiple Agonists for D 1 and D 2 Dopamine Receptors. Chem. Med. Chem, 4, 1514-1522 (2009).
• Aroa Soriano, Ruben Ventura, Anabel Molero, Rob Hoen, Vicent Casadó, Antoni Cortés, Francesca Fanelli, Fernando Albericio, Carmen Lluis, Miriam Royo, Rafael Franco. Dopamine D2R-agonist/adenosine A2AR-antagonist bivalentligands as chemical tools to study A2A/D2 receptor heteromers. J. Med. Chem., 52, 5590-5602 (2009).
• Luísa Custódio, Eliana Fernandes,Ana Luísa Escapa, Sandra López-Avilés, Alba Fajardo, Rosa Aligué,Fernando Alberício,and Anabela Romano. Antioxidant and in Vitro Inhibition of Tumor Cell groth by Leaf Extracts from the Carob Three (Ceratonia siliqua L). Pharm. Biol., 47, 721-728 (2009).
• Ramon Subiros-Funosas, Gerardo A. Acosta, Ayman El-Faham, Fernando Albericio.Microwave irradiation and COMU: a superior tool for SPPS. Tetrahedron Lett. 50, 6200-6202 (2009).
• Mireck Sisa, Daniel Pla, Marta Altuna, Andrés Francesch, Carmen Cuevas, Fernando Albericio, and Mercedes Álvarez. Total Synthesis of ()-Aplicyanins A, B, and E. J. Med. Chem., 52, 6217-6223 (2009).
• Javier Ruíz-Rodríguez, Jan Spengler, and Fernando Albericio. Siamese Depsipeptides: New Constrained Bicyclic Architectures. Angew. Chem., Int. Ed.48, 8564-8567 (2009).
• Athanassios S. Galanis, Fernando Albericio, and Morten Grøtli. Solid Phase Peptide Synthesis in Water using Microwave-Assisted Irradiation. Org. Lett.,11, 4488-4491 (2009).
• Carlos Mas-Moruno, Laura Cascales, Puig Mora, Luis J. Cruz, Enriqe Pérez-Payá, and Fernando Albericio. Design and facile solid-phase synthesis of LPS-inhibitors containing PEG-like functionalities. Biopolymers (Peptide Sci.),92, 508-517 (2009).
• Yésica García-Ramos, Matthieu Giraud, Judit Tulla-Puche, and Fernando Albericio. Optimized Fmoc Solid-Phase Synthesis of Thymosin 1 by Side-Chain Anchoring onto a PEG Resin. Biopolymers (Peptide Sci)., 92, 565-572 (2009).
• Pablo Cironi, Mercedes Alvarez, Fernando Albericio. Solid-phase synthesis of non-peptidic natural compounds. Rossiiskii Khimicheskii Zhurnal 53, 73-86 (2009).
• Judit Tulla-Puche, Eleonora Marcucci, Irene Izzo, Gerardo Acosta, Sara Auriemma, Chiara Falciani, and Fernando Albericio. N-Methylation as a Synthetic Resource for Increasing Stability in Depsipeptides. In Breaking Away: Proceedings of the 21st American Peptide Symposium. (M. Lebl, ed.), American Peptide Society, 2009, pp. 48-49.
• Silvia Cavalli, Fernando Albericio, and Alexander Kros. Amphiphilic Peptides and their cross-disciplinary role as building blocks for nanoscience. Chem. Soc. Rev., 39, 241-263 (2010).
• Sherine N. Khattab, Seham Y. Hassan, Ezzat A. Hamed, Fernando Albericio, Ayman. El-Faham
• Leticia Hosta-Rigau, Brigitte Städler, Yan Yan, Edouard Nice, Joan K. Heath, FernandoAlbericio andFrank Caruso. Capsosomes with Multilayered Subcompartments: Assembly and Loading with Hydrophobic Cargo.Adv. Funct. Mat., 20, 59-66 (2010).
• Ayman El-Faham and Fernando Albericio. COMU: A Third Generation of Uronium-Type Based Coupling Reagent. J. Peptide Sci. 16, 6-9 (2010).
• Javier Ruiz-Rodríguez, Fernando Albericio,and Rodolfo Lavilla. Postsynthetic Modification of Peptides. Chemoselective C-Arylation of Tryptophan residues. Chem., Eur. J., 16, 1124-1127 (2010).
• Frank Sicherl, Tommaso Cupido, and Fernando Albericio. A Novel Dipeptidomimetic Containing a Cyclic Threonine. Chem.Commun., 46, 1266-1268 (2010).
• Hortensia Rodríguez, Margarita Suarez, and Fernando Albericio. A Convenient Microwave-Enhanced Solid-Phase Synthesis of Short Chain Highly Hindered N-Methyl-Rich Peptides. J. Peptide Sci. 16, 136-140 (2010).
• Aroa Soriano, Marc Vendrell, Sergio Gonzalez, Josefa Mallol, Fernando Albericio, Miriam Royo Carmen Lluís, Enric I. Canela, Rafael Franco, Antoni Cortés, Vicent Casadó. A Hybrid Indoloquinolizidine/Peptide As Allosteric Modulator of Dopamine D1 Receptors. J. Pharmac. Exper. Therap.,33, 876-885 (2010).
• Fernando Albericio, Mercedes Álvarez,Carmen Cuevas, Andres Francesch, Daniel Pla, and Judit Tulla-Puche. The Sea as Source of New Drugs. In Molecular Imaging for Integrated Medical Therapy and Drug Development (N, Tamaki, Y. Kuge, eds) Springer-Japan, Tokyo (Japan), 237-249 (2010).
• Tommaso Cupido, Javier Ruiz-Rodriguez, Jaume Adan, Francesc Mitjans, Jaume Piluats, Jan Spengler, and Fernando Albericio.Ester Scan of Cyclopeptides as a Tool for Biological Activity Modulation: Synthesis, Conformational and Biological Analysis of RGD Depsipeptides. Angew. Chemie.,49, 2732-2737 (2010).
• María C. Martínez-Ceron, Silvana L. Giudicessi, Mariela M. Marani, Fernando Albericio, Osvaldo Cascone, Rosa Erra-Balsells, and Silvia A. Camperi. Sample preparation for sequencing hits from one-bead one-peptide combinatorial libraries by MALDI MS. Anal. Biochem.,400, 295-297 (2010).
• Rona Chandrawati, Leticia Hosta-Rigau,Dirk Vanderstraaten, Shalitha Lokuliyana, Brigitte Städler, Fernando Albericio, and Frank Caruso. Essentials on Capsosomes: Maximizing the Number of Subcompartments, Cargo Retention, and Temperature-Triggered Reaction. ACS Nano, 4, 1351-1361 (2010).
• Jan Spengler, Marta Pelay, Judit Tulla-Puche, Fernando Albericio. Synthesis of Orthogonally Protected L-threo-β-Ethoxyasparagine. Amino Acids, 39, 161-165 (2010).
• Luis J. Cruz, Paul J. Tacken, RemcoFokkink, Ben Joosten, Martien Cohen Stuart, Fernando Albericio, RuurdTorensma, Carl G. Figdor. Targeted PLGA nano- but not microparticles specifically deliver antigen to human dendritic cells in vitro. J. Control. Release.144, 118-126 (2010).
• Karen Muthusamy, Fernando Albericio, Per I. Arvidsson, Patrick Govender, Hendrik G. Kruger and Thavendran Govender Microwave assisted SPPS of amylin and its toxicity of the pure product to RIN-5F cells. Biopolymers (Peptide Sci.) 94, 323-330 (2010).
• Irene Izzo, Gerardo A. Acosta, Judit Tulla-Puche, Tommaso Cupido, Maria Jesus Martin-Lopez, Carmen Cuevas, and Fernando Albericio. Solid-phase synthesis of aza Kahalalide F analogues. (2R,3R)-2-amino-3-azidobutanoic acid as precursor of the aza-threonine. Eur. J. Org. Chem.2536–2543 (2010).
• Sherine N. Khattab, Ramon Subirós-Funosas, Ayman El-Faham, and Fernando Albericio. Oxime Carbonates, Novel Reagents for the Introduction of Fmoc and Alloc protecting groups, free of Side-Reactions. Eur. J. Org. Chem., 3275-3280 (2010).
• Leticia Hosta-Rigau, Ivonne Olmedo, Jordi Arbiol, Luis J. Cruz, MarceloJ. Kogan, and Fernando Albericio Multifunctionalized Gold Nanoparticles with Peptides Targeted to Gastrin-releasing Peptide Receptorof a Tumour Cell Line. Bioconjugate Chem,21, 1070-1078 (2010).
• Ayman El-Faham, Ramon Subirós-Funosas, and Fernando Albericio. A Novel Family of Onium Salts Based Upon Isonitroso Meldrum's Acid Proves Useful as Peptide Coupling Reagents. Eur. J. Org. Chem. 3641-3649 (2010).
• Simon Guerrero, Eyleen Araya, Jenny Fiedler, J. Ignacio Arias, Carolina Adura, Fernando Albericio, Ernest Giralt, Jose Luis Arias, M. Soledad Fernández,and Marcelo J. Kogan. Improving the Brain Delivery of Gold Nanoparticles by Conjugation with an Amphipathic Peptide. Nanomedicine, 5, 897-913 (2010).
• Oscar Garcia,Josep M. Bofill, Ernesto Nicolas, and Fernando Albericio. 2,2,4,6,7-Pentamethyl-2,3-dihydrobenzofuran-5-methyl (Pbfm) as Alternative to Trityl Group for the Side-chain Protection of Cysteine and Asparagine/Glutamine. Eur. J. Org. Chem., 3631-3640 (2010).
• M. Jesús Pérez de Vega, M. Teresa García-López, Laura Zaccaro, Miriam Royo, Fernando Albericio, Asia Fernández-Carvajal, Antonio Ferrer-Montiel,and Rosario González-MuñizSolid-Phase Synthesis of New Trp(Nps)-Containing Dipeptide Derivatives as TRPV1 Channel Blockers. Molecules, 15, 4924-4933 (2010).
• Jan Spengler,Ana I. Fernández-Llamazares, Javier Ruiz-Rodríguez,Klaus Burger,and Fernando Albericio. Total Regioselective Control of Tartaric Acid. J. Org. Chem.,75, 5746-5749 (2010).
• Ramon Subirós-Funosas,Ayman El-Faham,FernandoAlbericio. PyOxP and PyOxB: the Oxyma-based novel family of phosphonium salts. Org. Biomol. Chem, 8, 3665-3673 (2010).
• Rodrigo Gonzalez, Fernando Albericio, Osvaldo Cascone, Nancy B. Iannucci. Improved Antimicrobial Activity of h-Lysozyme (107-115) by Rational Ala Substitution. J. Peptide Sci.,16, 424-429 (2010).
• Yésica García-Ramos, Marta Paradís-Bas, Judit Tulla-Puche, and Fernando Albericio. ChemMatrix® for Complex Peptides and Combinatorial Chemistry. J. Peptide Sci.,16, 675-678 (2010).
• Adriana Lorente, Daniel Pla, Librada M. Cañedo, Fernando Albericio and Mercedes Álvarez. Isolation, Structural Assignment and Total Synthesis of Barmumcyn. J. Org. Chem., 75, 8508-8515 (2010).
• Juan R. Luque-Ortega, Luis J. Cruz, Fernando Albericio, and Luis Rivas. The antitumoral depsipeptide IB-01212 kills Leishmania through an apoptosis-like process involving intracellular targets. Molec. Pharm. 7, 1608-1617 (2010).
• Sandra Gonçalves, Celine Xavier, Patrícia Costa, Fernando Alberício, and Anabela Romano. Antioxidant, cytotoxic and apoptotic activity of Drosophyllum lusitanicum extracts. J. Med. Plants Res., 4, 1601-1608 (2010).
• Tarfah I. Al-Warhi, Hassan M.A. AL-Hazimi, Ayman El-Faham, Fernando Albericio. Synthesis of 2-(4,6-dimethyoxy-1,3,5-triazin-2-yloxyimino) Derivatives: Application in Solution Peptide Synthesis. Molecules,15, 9403-9417 (2010).
• Davide Bello, Javier Ruiz, Fernando Albericio, Rosario Ramón, Rodolfo Lavilla. Streamlined Access to Functionalized Chromenes and Quinolines via Domino Reactions of Salicylic Aldehydes and Methyl 4-Chloro-2-Butynoate. Eur. J. Org. Chem., 5373-5379 (2010).
• Silvia A. Camperi, Mariela M. Marani, María C. Martínez-Ceron, Fernando Albericio, and Osvaldo Cascone. Protein purification by affinity chromatography with peptide ligands selected from the screening of combinatorial libraries. Trends in Chromatography, 6, 11-22 (2010).
• Hilda Garay, Tamara Menéndez, Yoelys Cruz-Leal, Edelgis Coizeau, Jesus Noda, Vivian Morera, Gerardo Guillén, Fernando Albericio and Osvaldo Reyes. Study of various presentation forms for a peptide mimetic of Neisseria meningitidis serogroup capsular polysaccharide. Bioconj. Chem., 22, 33-41 (2011).
• Pau Ruiz-Sanchis, Svetlana Savina, Fernando Albericio, and Mercedes Álvarez. Structure, Synthesis, and Bioactivity of Natural Products with Hexahydropyrrolo[2,3-b]indole. Chem, Eur. J.,17, 1388-1408 (2011).
• Among the top 20 most cited Reviews in Chemistry—A European Journal of the past 20 years
• Luis J. Cruz, Felix Rueda, Begoña Cordobilla, Lorena Simon, Leticia Hosta, Fernando Albericio, Joan Carles Domingo. Targeting nanosystems to human DCs via Fc receptor as an effective strategy to deliver antigen for immunotherapy.Molec. Pharm., 8, 104-116 (2011).
• Myriam Gongora, Judit Tulla-Puche, Marta Paradis-Bas, Oleg Werbitzky, Matthieu Giraud, and Fernando Albericio. Optimized Fmoc Solid-Phase Synthesis of the Cysteine-Rich Peptide Linaclotide. Biopolymers (Peptide Sci).,96, 69-80 (2011).
• Marc Vendrell, Anabel Molero, Sergio Gonzalez, Kamil Pérez-Capote,Carme Lluis, Peter J. McCormick, Rafael Franco, Antoni Cortés, Vicent Casadó, Fernando Albericio, and Miriam Royo. Biotin Ergopeptide Probes for Dopamine Receptors. J. Med. Chem. 54, 1080-1090 (2011).
• Amaranta Gómez-Arreaza, Hector Acosta, Ximena Barros-Álvarez, Juan L. Concepcion, Fernando Albericio, Luisana Avilan. Leishmania mexicana: LACK (Leishmania homologue of receptors for activated C-kinase) is a plasminogen binding protein. Exp. Parasitology, 127, 752-761 (2011).
• Konrad G. Jastrząbek, Ramon Subiros-Funosas, Fernando Albericio, Beata Kolesinska, Zbigniew J. Kamiński.4-(4,6-[2,2,2-Trifluoroethoxy]-1,3,5-triazin-2-yl)-4-methylomorpholinium tetrafluoro-borate (DFET/ NMM/BF4). Triazine based coupling reagents designed for coupling sterically hindered substrates. J. Org. Chem., 76, 4506-4513 (2011).
• Selected as one of the best 25 papers dealing with peptides published by the ACS in the period 2011-2012.
• Luisa Custodio, Eliana Fernandes, Ana Luisa Escapa, Alba Fajardo, Rosa Aligué, Fernando Albericio, Nuno Neng, Jose Manuel Nogueira, Anabela Romano. Phytochemical profile, antioxidant and cytotoxic activities of carob tree (Ceratonia siliqua L.) germ flour extracts. Plant Foods for Human Nutrition, 66, 78-84 (2011).
• Hortensia Rodriguez,Julieta Coro, Osnieski Martin, Anabel Lam, Esperanza Salfrán, Javier Rodríguez-Salarichs, Margarita Suárez, Fernando Albericio,and Nazario Martín. Efficient preparation of alkyl 4-aryl substituted-2-methyl-6-thioxo-1,4,5,6-tetrahydropyridine-3-carboxylates under microwave irradiation conditions. ARKIVOC, 125-141 (2011).
• María C. Martínez-Ceron, Mariela M. Marani, Marta Taulés, Marina Etcheverrigaray, Fernando Albericio, Osvaldo Cascone, and Silvia A. Camperi. Affinity Chromatography-Based Combinatorial Strategy for rErythropoietin Purification. ACS Comb. Sci.13, 251-258 (2011).
• Claudio Jofré, Fanny Guzmán, Constanza Cárdenas, Fernando Albericio, and Sergio H. Marshall. A natural peptide and its variants from the processing of Infectious Pancreatic Necrosis Virus (IPNV) display enhanced antimicrobial activity: A novel alternative to control bacterial diseases. Peptides, 32, 852-858 (2011).
• Daniel Pla, Fernando Albericio, and Mercedes Álvarez. Progress on Lamellarins. MedChemComm., 2, 689-697 (2011), with cover.
• Sherine N. Khattab, Ezzat Awad Hamed, Fernando Albericio and Ayman El-Faham. Synthesis and Aminolysis of 2,4-Dinitro Phenyl and 5-Nitro Pyridine N-Hydroxy Oxime Derivatives, Bull. Chem. Soc. Jpn. 84, 633-639 (2011).
• Laura Zaccaro, M. Teresa Garcia-Lopez, Rosario Gonzalez-Muñiz, Carolina Garcia- Martinez, Antonio Ferrer-Montiel, Fernando Albericio, Miriam Royo. TRPV1 modulators: Structure-activity relationship using a rational combinatorial approach. Bioorg. Med. Chem., 21, 3541-3545 (2011).
• Rubén Ferreira, Roberto Artali, Josep Farrera-Sinfreu, Fernando Albericio, Miriam Royo, Ramon Eritja, Stefania Mazzini. Acridine and quindoline oligomers linked through a 4-aminoproline backbone prefer G-quadruplex structures. Biochim. Biophys. Acta. 1810, 769-776 (2011).
• Guillermo Gerona-Navarro, Rosario González-Muñiz, Asia Fernández-Carvajal, José M. González-Ros, Antonio Ferrer-Montiel,Cristina Carreño,Fernando Albericio,Miriam Royo. Solid-phase synthesis of a library of amphipatic hydantoins. Discovery of new hits for TRPV1 blockade. ACS Comb. Sci.13, 458-465 (2011).
• Luisa Custodio, Eliana Fernandes, Ana Luisa Escapa, Alba. Fajardo, Rosa Aligué, Fernando Albericio, Nuno Neng, Jose Manuel Nogueira, Anabela Romano. Antioxidant and Cytotoxic Activities of Carob TreeFruit Pulps are StronglyInfluenced by Gender and Cultivar. J. Agric. Food Chem.59, 7005-7012 (2011).
• Ayman El-Faham and Fernando Albericio. Peptide Coupling Reagents, More than a Letter Soup. Chem. Rev. 111, 6557-6602 (2011).
• Ángela Torres,Carlos Mas-Moruno, Enrique Pérez-Payá, Fernando Albericio, and Miriam Royo. Trivalent PEGylated Platform for the Conjugation of Bioactive Compounds. Bioconjugate Chem,22, 2172-2178 (2011).
• M.E.S. Martins-Santos, R.R. Resende, F.C.H. Pinto, A.M. Soares, S. Marangoni, Eliandre de Oliveira, Fernando Albericio, and Saulo L. Da Silva. Effect of a Pool of Peptides Isolated from Crotalus durissus terrificus (South American Rattlesnake) Venom on Glucose Levels of Mice Fed on a High-Fat Diet.Int. J. Peptide Res. Therap. 17, 225-230 (2011).
• Xavier Just-Baringo, Paolo Bruno, Fernando Albericio, Mercedes Álvarez. Highly Efficient, Multigram and Enantiopure Synthesis of 2-(2,4’-bithiazol-2-yl)pyrrolidine. Tetrahedron Lett.,52, 5435-5437 (2011).
• Paolo Bruno, Stella Peña,Xavier Just-Baringo, Fernando Albericio and Mercedes Álvarez. Total synthesis of Aeruginazole A. Organic Lett., 13, 4648-4651 (2011).
• Ramon Subirós-Funosas, Ayman El-Faham, Fernando Albericio. Aspartimide formation in peptide chemistry: occurrence, prevention strategies and the role of N-hydroxylamines. Tetrahedron, 67, 8595-8606 (2011).
• Elisabet Prats-Alfonso and Fernando Albericio. Functionalization of Gold Surfaces: Recent Developments and Applications. J. Mat. Sci. 46, 7643-7648 (2011).
• Venugopala K. Narayanaswamy, Fernando Albericio,Yacoob M. Coodavia, Hendrik G. Kruger,Glenn E. M. Maguire, Melendran Pillaym and Thavendran Govender. Total synthesis of a Depsidomycin analogue by convergent solid phase peptide synthesis and macrolactonization Strategy for antitubercular activity. J. Peptide Sci. 17, 683-689 (2011).
• Hortensia Rodríguez, Julieta Copro, Margarit Suárez, Roberto Martínez-Álvarez, Nazario Martín, Fernando Albericio. Eco-Friendly Methodology to Prepare N-Heterocycles Related to Dihydropyridines: Microwave-Assisted Synthesis of Alkyl 4-Arylsubstituted-6-chloro-5-formyl-2-methyl-1,4-dihydropyridine-3-carboxylate and 4-Arylsubstituted-4,7-dihydrofuro[3,4-b]pyridine-2,5(1H,3H)-dione. Molecules, 16, 9620-9635 (2011).
• Luisa Custodio, Eliana Fernandes, Ana Luisa Escapa, Rosa Aligué, Fernando Albericio, Anabela Romano. In vitro cytotoxic effects and apoptosis induction by a methanol leaf extract of carob tree (Ceratonia siliqua). J. Med. Plants Res.5, 1987-1996 (2011).
• Fernando Alberico, Judit Tulla-Puche, and Steven A. Kates. The Fmoc Methodology: Cleavage from the Resin and Final Deprotection. In Amino Acids, Peptides and Proteins in Organic Chemistry. Vol.3 – Building Blocks, Catalysis and Coupling Chemistry (A.B. Hughes, ed.) Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim (Germany), pp. 349-369 (2011).
• Ayman El-Faham and Fernando Albericio. Coupling Reagents. In Amino Acids, Peptides and Proteins in Organic ChemistryVol.3 – Building Blocks, Catalysis and Coupling Chemistry (A.B. Hughes, ed.) Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim (Germany), pp. 407-444 (2011).
• Ramon Subiros-Funosas, Fernando Albericio, Ayman El-Faham. N-Hydroxylamines for Peptide Synthesis. In The Chemistry of Hydroxylamines, Oximes and Hydroxamic Acids, Vol. 2 (Z. Rappoport and J. F. Liebman, eds.) John Wiley & Sons Ltd (Chichester, United Kingdom), pp. 623-729, 2011.
• Fernando Albericio and Ramon Subirós-Funosas. (1-Cyano-2-ethoxy-2-oxoethylidenamino-oxy)dimethylaminomorpholino-carbenium hexafluorophosphate. In e-EROS Encyclopedia of Reagents for Organic Synthesis. (D. Crich, P.L. Fuchs, A.B. Charette, T. Rovis, eds.), John Wiley & Sons Ltd, Chichester, U.K., http://onlinelibrary.wiley.com/book/10.1002/047084289X (2011).
• Fernando Albericio and Ramon Subirós-Funosas. Ethyl 2-cyano-2-(hydroxyimino)acetate. In e-EROS Encyclopedia of Reagents for Organic Synthesis. (D. Crich, P.L. Fuchs, A.B. Charette, T. Rovis, eds.), John Wiley & Sons Ltd, Chichester, U.K., http://onlinelibrary.wiley.com/book/10.1002/047084289X (2011).
• Miriam Góngora-Benítez, Alessandra Basso, Thomas Bruckdorfer, Judit Tulla-Puche, Fernando Albericio. A Green Strategy for the Synthesis of Cysteine-Containing Peptides. In Proceedings of the 22nd American Peptide Symposium, Michal Lebl (ed.) American Peptide Society, pp. 14-15, 2011.
• Lidia Nieto-Rodriguez, Magda Carceller, Ramon Subirós-Funosas, Gerardo A. Acosta, Marta Paradís Bas, Ayman El-Faham, Fernando Albericio. Practical Tips on the Use of Oxyma: An Exhaustive Stability Assay. In Proceedings of the 22nd American Peptide Symposium, Michal Lebl (ed.) American Peptide Society, pp. 16-17, 2011.
• Ramon Subirós-Funosas, Ayman El-Faham, Fernando Albericio. Novel Applications of Oxyma: Minimization of Base-Driven Side Reactions. In Proceedings of the 22nd American Peptide Symposium, Michal Lebl (ed.) American Peptide Society, pp. 18-19, 2011.
• Nancy B. Iannucci, Silvia A. Camperi, María V. Miranda, Fernando Albericio, Osvaldo Cascone. Immobilized Peptide as Affinity Chromatography Ligand for Soybean Peroxidase Purification. In Proceedings of the 22nd American Peptide Symposium, Michal Lebl (ed.) American Peptide Society, pp. 98-99, 2011.
• Fanny Guzmán, Felipe León, Sergio Marshall, Claudia Ojeda, Fernando Albericio, Patricio Carvajal-Rondanelli. Comparative Study on the Antimicrobial Effect of Small Cationic Homopeptides. In Proceedings of the 22nd American Peptide Symposium, Michal Lebl (ed.) American Peptide Society, pp. 210-211, 2011.
• Nancy B. Iannucci, Axel Hollmann, María R. Diaz, Osvaldo Cascone, Fernando Albericio, Aníbal E. Disalvo. Peptide-Membrane Interaction Analysis of an Improved Antimicrobial Peptide Derived from the 107-115 hLz Fragment. In Proceedings of the 22nd American Peptide Symposium, Michal Lebl (ed.) American Peptide Society, pp. 294-295, 2011.
• Fernando Albericio, Ayman El-Faham, Myriam Gongora-Benitez, Ramon Subirós-Funosas, Judit Tulla-Puch. Solid-Phase Peptide Synthesis: State of the Art. In Proceedings of the 22nd American Peptide Symposium, Michal Lebl (ed.) American Peptide Society, pp. 406-407, 2011.
• Nancy B. Iannucci, Rodrigo González, Osvaldo Cascone, Fernando Albericio. Novel strategy for designing antimicrobial peptides: an answer to the development of drug resistance. In Science Against Microbial Pathogens: Communicating Current Research and Technological Advances. Microbiology Book Series, 3. Vol. 2. (A. Mendez-Vilas, ed). Formatex Research Center, Badajoz (Spain), 961-967, 2011.
• Silvia Cavalli, Hana Robson Marsden, Fernando Albericio, Alexander Kros. Peptide Self-Assembly. In Supramolecular Chemistry: From Molecules to Nanomaterials (Jonathan W. Steed and Philip A., eds) John Wiley & Sons, Ltd., Chichester (UK)., 5, 2293-2310 (2012).
• Pau Ruiz-Sanchis, Svetlana A. Savina, Gerardo A. Acosta, Fernando Albericio, and Mercedes Álvarez. Orthogonal Protecting Groups in the Synthesis of Tryptophanyl-Hexahydropyrroloindoles. EurJOC, 67-73 (2012).
• Luísa Custódio, Tiago Justo, Laura Silvestre, Ana Barradas, Catarina Vizetto Duarte, Hugo Pereira, Luísa Barreira, Amélia Pilar Rauter, Fernando Alberício, João Varela.Microalgae of different phyla display antioxidant, metal chelating and acetylcholinesterase inhibitory activities. Food Chem., 131, 134-140 (2012).
• Hammed H.A.M Hassan, Amel F. El-Husseiny, Abeer G. Abo-Elfady, Ayman El-Faham, Fernando Albericio. Synthesis and Thermal Properties of Novel Polyamides Containing α-Amino Acid Moieties: Structure-Property Relationship. J. Macrom. Sci., Part A: Pure & Applied Chem. 49, 45-54 (2012).
• Eleonora Marcucci,Judit Tulla-Puche, and Fernando Albericio. Solid-Phase Synthesis of N-Me IB-01212, a Multiple N-Me Cyclic Peptide. Org. Lett., 14, 612-615 (2012).
• Hiroshi Hinou, Kei Hyugaji, Fayna Garcia-Martin, Shin-Ichiro Nishimura, Fernando Albericio. H-Bonding Promotion of Peptide Solubility and Cyclization by Fluorinated Alcohols: Synthesis of Cyclic Peptide Skeleton of Antifreeze Glycopeptide, RSC, Advances, 2, 2729-2731 (2012).
• Sherine N. Khattab, Ramon Subirós-Funosas, Ayman El-Faham Fernando Albericio. Cyanoacetamide-based oxime carbonates: an efficient, simple alternative for the introduction of Fmoc with minimal dipeptide formation. Tetrahedron, 68, 3056-3062 (2012).
• Yordanka Masforrol, Jeovanis Gil, Luis Javier González, Yasset Pérez-Riverol, Jorge Fernández-de-Cossío, Aniel Sánchez, Lázaro Betancourt, Hilda Elisa Garay, Ania Cabrales, Fernando Albericio, Honqiang Yang, Roman Zubarev, Vladimir Besada, and Osvaldo Reyes. Introducing an Asp-Pro linker in the synthesis of random one-bead-one-compound hexapeptide libraries compatible with ESI-MS analysis.ACS Comb. Sci.14, 145-149 (2012).
• Miriam Góngora-Benítez, Michèle Cristau, Matthieu Giraud, Judit Tulla-Puche, Fernando Albericio. Intramolecular Click Chemistry-Based Handle for Solid-Phase Synthesis. Chem. Comm., 48, 2313-2315 (2012).
• Simón Guerrero, Raúl Herrance,Santiago Rojas, Juan F. Mena, Juan Domingo Gispert, Gerardo A. Acosta, Fernando Albericio, Marcelo J Kogan. Synthesis and In Vivo Evaluation of the Biodistribution of a 18F Labelled Conjugate Gold-Nanoparticle-Peptide with Potential Biomedical Application. Bioconjugate. Chem. 23, 399-408 (2012).
• Ramon Subirós-Funosas, Ayman El-Faham, and Fernando Albericio. Use of Oxyma as pH modulator agent to be used in the prevention of base-driven side reactions and its effect on 2-chlorotrityl chloride resin. Biopolymers (Pept. Sci), 98, 89-97 (2012).
• Anna Lagunas, Jordi Comelles, Elena Martínez, Elisabet Prats-Alfonso, Gerardo A. Acosta, Fernando Albericio, and Josep Samitier. Cell adhesion and focal contact formation on smooth RGD molecular gradients: study of non-linear concentration dependence effects. Nanomedicine: Nanotechnology, Biology, Medicine, 8, 432-439 (2012).|
• Cristina Rosés, Daniel Carbajo, Glòria Sanclimens, Josep Farrera-Sinfreu, Adriana Blancafort, Glòria Oliveras, Anna Díaz-Cirac, Eduard Bardají, Teresa Puig, Marta Planas, Lidia Feliu, Fernando Albericio and Miriam Royo.Cell-penetrating γ-Peptide/Antimicrobial Undecapeptide Conjugates with Anticancer Activity. Tetrahedron, 68, 4406-4412 (2012).
• Yahya El-Sayed Jad, Sherine N. Khattab, Ayman El-Faham, Fernando Albericio. Oxyme Based Carbonates as Useful Reagents for both N-Protection and Peptide Coupling. Molecules 17, 14361-14376 (2012).
• Elisabet Prats-Alfonso, Xavi Sisquella, Nadia Zine, Gemma Gabriel, Antón Guimerà, Javier del Campo, Rosa Villa, Adam Eisenberg, Milan Mrksich, Abdelhamid Errachid, Jordi Aguiló,and Fernando Albericio. Early Cancer Prognostic by Direct Detection of p53-Antibodies on Gold Surfaces by Impedance Measurements. Small, 8, 2106-2115 (2012).
• Luis J. Cruz,Paul J. Tacken, Felix Rueda, Joan Carles Domingo, Fernando Albericio, Carl G. Figdor. Targeting nanoparticles to dendritic cells for immunotherapy. Meth. Enzym., 509, 143-163 (2012).
• Luisa Custodio, Catarina Ferreira, Hugo Pereira, Laura Silvestre, Catarina Vizetto-Duarte, Luísa Barreira, Amélia Pilar Rauter, Fernando Albericio, João Varela. The marine halophytes Carpobrotusedulis L. and Arthrocnemum macrostachyum L. are potential sources of nutritionally important PUFAs and metabolites with antioxidant, metal chelating and anticholinesterase inhibitory activities. BOTMAR, 55, 281-288 (2012).
• Rebecca van der Westen, Leticia Hosta-Rigau, Duncan S. Sutherland, Kenneth Goldie, Fernando Albericio, Almar Postma, Brigitte Städler. Myoblast Cell Interaction with Polydopamine Coated Liposomes. Biointerphases,7(1-4), 8 (2012).
• Sergio Abad, Pau Nolis, Juan D. Gispert, Jan Spengler, Fernando Albericio, Santiago Rojas, José R. Herance. Rapid and high-yielding cysteine labelling of peptides with N-succinimidyl 4-[18F]fluorobenzoate. Chem. Comm. 48, 6118-6120 (2012).
• Miriam Góngora-Benítez, Lorena Mendive-Tapia, Iván Ramos-Tomillero, Arjen C. Breman, Judit Tulla-Puche, Fernando Albericio. Acid-Labile Cys-Protecting Groups for Fmoc/tBu Strategy: Filling the Gap. Org. Lett., 14, 5472-5475 (2012).
• Tobias M. Postma, Matthieu Giraud, Fernando Albericio. Trimethoxyphenylthio as a Highly Labile Replacement for tert-butylthio Cysteine Protection in Fmoc Solid Phase Synthesis. Org. Lett., 14, 5468-5471 (2012).
• Sherine N. Khattab, Ramon Subirós-Funosas, Ayman El-Faham Fernando Albericio.Screening of N-Hydroxy-2-Oxoacetimido Cyanide Derivatives as Substitutes for N-Hydroxysuccinimide. ChemistryOpen. 1, 147-152 (2012).
• Gemma Vilar, Judit Tulla-Puche, Fernando Albericio. Polymers and Drug Delivery Systems. Curr. Drug Deliv., 9, 367-394 (2012).
• Hortensia Rodríguez, Margarita Suárez, Fernando Albericio. Thiadiazines, N,Nheterocycles of biologicalrelevance. Molecules 17, 7612-7628 (2012)
• Fernando Albericio, Hendrik G. Kruger. Therapeutic Peptides. Future Med. Chem., 4, 1527-1531 (2012).
• Hortensia Rodríguez, Julieta Coro, Margarita Suárez, Roberto Martínez-Álvarez, Nazario Martín, Fernando Albericio. Liquid phase organic synthesis of 3,5-disubstituted 1,3,5-thiadiazinane-2-thione derivatives on polyethylene glycol (PEG) support. ARKIVOC, (viii) 326-328 (2012).
• S.L. Da Silva, C.A. Dias-Junior, P.A. Baldasso, D.C.S. Damico, B.M.A. Carvalhoa, A.G. Taranto, G.A. Costa, E. Oliveira, F. Albericio, A.M. Soares, S. Marangonic, R.R. Resende. Vascular effects and electrolyte homeostasis of the natriuretic peptide isolated from Crotalus oreganus abyssus (North American Grand Canyon rattlesnake) venom. Peptides, 36, 206-212 (2012).
• Luis J. Cruz,Felix Rueda, Paul Tacken, Fernando Albericio,Ruurd Torensma,Carl G. Figdor.Enhancing immunogenicity and cross-reactivity of HIV-1 antigens by in vivo targeting to dendritic cells. Nanomedicine, 7, 1591-1610(2012).
• Leticia Hosta-Rigau, Bettina E.B. Jensen, Kit S. Fjeldsø, Almar Postma, Guoxin Li, Kenneth N. Goldie, Fernando Albericio, Alexander N. Zelikin,Brigitte Städler. Surface-Adhered Composite Poly(Vinyl Alcohol) Physical Hydrogels: Polymersome-Aided Delivery of Therapeutic Peptides. Adv. Health. Mat., 1, 791-795 (2012).
• Miriam Góngora-Benítez, Alessandra Basso, Thomas Bruckdorfer,Miriam Royo, Judit Tulla-Puche and Fernando Albericio. Eco-friendly combination of the immobilised-PGA enzyme and the Phacm protecting group for the synthesis of cysteine-containing peptides. Chem. Eur J., 18, 16166-16176 (2012).
• Silvia Cavalli, Daniel Carbajo, Milena Acosta, Silvia Lope-Piedrafita, Ana Paula Candiota, Carles Arús, Miriam Royo, Fernando Albericio. Efficient gamma-Amino-proline-derived Cell Penetrating Peptide-superparamagnetic Iron Oxide Nanoparticle Conjugates via Aniline-Catalyzed Oxime Chemistry as Bimodal Imaging Nanoagents. ChemComm., 48,5322-5324 (2012).
• Antonio Zorzano, David Sebastián, Jana Sánchez-Wandelmer, Laia Miret, Fernando Albericio. Gene promoters and transcription control regions as therapeutic targets. In Therapeutic targets: modulation, inhibition, and activation (L.M. Botana, M.I. Loza, eds.), John Wiley & Sons, Inc., Hoboken, NJ, USA. pp. 327-350 (2012).
• Judit Tulla-Puche, Rita S. Majerle, Fernando Albericio, George Barany. Resin-to-Resin Transfer Reaction (RRTR) via Sonogashira Coupling. In Solid Phase Organic Syntheses Volume 2: Solid-phase Palladium Chemistry (Peter J. H. Scott ed.), John Wiley and Sons, Hoboken NJ, pp. 59-66, 2012.
• Peter Fransen, Daniel Pulido, Ryan Seelbach, Alvaro Mata, David Eglin, Miriam Royo, Fernando Albericio. Biofunctionalization of biopolymers with peptide conjugated dendrons. In Proceedings of the 32nd European Peptide Symposium (G. Kokotos, V. Constantinou-Kokotou, J. Matsoukas, ed.), European Peptide Society, Athenes (Greece), 2012, pp. 136-137
• Jan Spengler, Anna-Iris Fernandez-Llamazares, Fernando Albericio. Use of internal references for the quantitative HPLC-UV analysis of solid-phase reactions. In Proceedings of the 32nd European Peptide Symposium (G. Kokotos, V. Constantinou-Kokotou, J. Matsoukas, ed.), European Peptide Society, Athenes (Greece), 2012, pp. 646-647.
• Nancy B. Iannucci, Rodrigo Gonzalez, Fanny Guzman, Osvaldo Cascone, Fernando Albericio. Enhanced anti-staphylococcal activity of an analog derived from the 107-115 humanlysozyme fragment. In Proceedings of the 32nd European Peptide Symposium (G. Kokotos, V. Constantinou-Kokotou, J. Matsoukas, ed.), European Peptide Society, Athenes (Greece), 2012, pp. 158-159.
• Tobias M. Postma, Matthieu Giraud, Fernando Albericio.Alkoxyphenylthio: Novel reducing agent labile cysteine protecting groups. In Proceedings of the 32nd European Peptide Symposium (G. Kokotos, V. Constantinou-Kokotou, J. Matsoukas, ed.), European Peptide Society, Athenes (Greece), 2012, pp. 408-409.
• Maria Pastrian, Fanny Guzman, Giselle Ripoll, Juan Garona, Marina Pifano, Osvaldo Cascone, Graciella Ciccia, Fernando Albericio, Daniel Gomez, Daniel Alonso, Nancy Iannucci. Improved antiproliferative activity of desmopressin analogs assessed by Ala-scanning. In Proceedings of the 32nd European Peptide Symposium (G. Kokotos, V. Constantinou-Kokotou, J. Matsoukas, ed.), European Peptide Society, Athenes (Greece), 2012, pp. 452-453.
• Rubi Z. Vazquez, Judit Tulla-Puche, Fernando Albericio. Novel non-covalent staple peptides. In Proceedings of the 32nd European Peptide Symposium (G. Kokotos, V. Constantinou-Kokotou, J. Matsoukas, ed.), European Peptide Society, Athenes (Greece), 2012, pp. 460-461.
• Vida Castro, Hortensia Rodriguez, Fernando Albericio. Resin via click chemistry to apply in SPPS. In Proceedings of the 32nd European Peptide Symposium (G. Kokotos, V. Constantinou-Kokotou, J. Matsoukas, ed.), European Peptide Society, Athenes (Greece), 2012, pp. 602-603.
• Anna-Iris Fernandez-Llamazares, Jan Spengler, Fernando Albericio. N-Oligoethyleneglycol cyclic peptides. In Proceedings of the 32nd European Peptide Symposium (G. Kokotos, V. Constantinou-Kokotou, J. Matsoukas, ed.), European Peptide Society, Athenes (Greece), 2012, pp. 612-613.
• Ramon Subirós-Funosas, Ayman El-Faham, and Fernando Albericio (Checked by Asher Lower and Margaret Faul). Low-epimerization Peptide Bond Formation with OxymaPure: Preparation of Z-L-Phg-Val-OMe. Org. Synth., 90, 306-315 (2013).
• Luisa Custodio, Joao Patarra, Fernando Albericio, Nuno Rosa Neng, Jose M. Florencio Nogueira, Anabela Romano. Extracts from Quercus sp. acorns exhibit in vitro neuroprotective features through inhibition of cholinesterase and protection of the human dopaminergic cell line SH-SY5Y from hydrogen peroxide-induced cytotoxicity. Ind. Crops Prod. 45, 114-120 (2013).
• Vida Castro, Hortendia Rodriguez, Fernando Albericio. Wang Linker Free of Side Reactions. Org. Lett., 15, 246-249 (2013).
• Tobias M. Postma,Fernando Albericio.N-Chlorosuccinimide, an efficient reagent for on-resin disulfide formation in solid-phase peptide synthesis. Org. Lett., 15, 616-619 (2013).
• Elisabet Prats-Alfonso, Sabine Oberhansl, Anna Lagunas, Elena Martínez,Josep Samitier, Fernando Albericio. Effective and Versatile Strategy for the Total Solid-Phase Synthesis of Alkanethiols for Biological Applications. EurJOC, pp. 1233-1239 (2013).
• Miriam Góngora-Benítez, Judit Tulla-Puche, Fernando Albericio ConstellaTM(EU)–LinzessTM(US): the last milestone in the long journey of the peptide Linaclotide and its implications for the future of peptide drugs. Future Med. Chem., 5, 291-300 (2013).
• Ramon Subirós Funosas, Sherine N. Khattab, Lidia Nieto-Rodriguez, Ayman El-Faham, Fernando Albericio. Advances in acylation methodologies enabled by Oxyma-based reagents. Aldrichima Acta, 46 (1), 21-40 (2013).
• Miriam Góngora-Benítez,Judit Tulla-Puche,Fernando Albericio. Handles for Fmoc solid-phase synthesis of protected peptides. ACS Comb. Sci.,15, 217-228 (2013).
• Jan Spengler, Anna-Iris Fernandez-Llamazares, Fernando Albericio. Use of an Internal Reference for the Quantitative HPLC-UV Analysis of Solid-Phase Reactions. ACS, Comb. Sci., 15, 229-234 (2013).
• Carolina Adura, Simon Guerrero, Edison Salas, Luis Medel, Ana Riveros, Juan Mena, Jordi Arbiol, Fernando Albericio, Ernest Giralt, Marcelo J. Kogan. Stable conjugates of peptides with gold nanorods for biomedical applications with reduced effects on cell viability. ACS App. Mat. Interfaces, 5, 4076-4085 (2013).
• Judit Tulla-Puche, Miriam Góngora-Benítez, Núria Bayó-Puxan, Andrés Francesch, Carmen Cuevas, and Fernando Albericio. Enzyme-Labile Protecting Groups add a New Orthogonal Level to the Synthesis of Complex Peptides: Solid-Phase Synthesis of Thiocoraline. Angew. Chemie., 52, 5726-5730 (2013); with section cover.
• Iván Ramos-Tomillero, Lorena Mendive-Tapia, Miriam Góngora-Benítez, Ernesto Nicolas, Judit Tulla-Puche, Fernando Albericio.Understanding acid lability on Cysteine protecting groups. Molecules 18, 5155-5162 (2013).
• Jan Spengler, Fernando Albericio. Asymmetric Synthesis of α-Unsubstituted β-Hydroxy Acids. Adv. Org. Synt., 4, 3-35 (2013).
• Santiago Rojas, Paus Nolis, Juan D. Gispert, Jan Spengler, Fernando Albericio, Jose R. Herance, Sergio Abad. Efficient cysteine labelling of peptides with N-succinimidyl 4-[18F]fluorobenzenzoate: satbility study and in vivo biodistribution in rats by positron emission tomography (PET). RSC Advances, 3, 8028-8036 (2013).
• Adriana Lorente, Janire Lamariano,Fernando Albericio, Mercedes Álvarez. Tetrahydrofuran-containing Macrolides, a Fascinating Gift from the Depth Sea. Chem. Rev., 113, 4567-4610 (2013).
• Lorena Simón-Gracia, Daniel Pulido, Chantal Sevrin, Christian Grandfils, FernandoAlbericio, Miriam Royo.Biocompatible, multifunctional, and well-defined PEG-based dendritic platforms for biomedical applications. Org. Biomol. Chem., 11, 4109-4121 (2013).
• Marta Pelay-Gimeno, Judit Tulla-Puche, Fernando Albericio. “Head-to-Side Chain” Cyclodepsipeptides from Marine Origin. Mar. Drugs, 11, 1693-1717 (2013).
• Xavier Just-Baringo, Paolo Bruno, Lars K. Ottesen, Librada M. Cañedo, Fernando Albericio and Mercedes Álvarez. Total Synthesis and Stereochemical Assignment of Baringolin. Angew. Chemie., 52, 7818-7820 (2013).
• Joan Camunas-Soler, Silvia Frutos, Cristiano V Bizarro, Sara de Lorenzo, Maria Eugenia Fuentes-Perez, Roland Ramsch, Susana Vilchez, Conxita Solans, Fernando Moreno-Herrero, Fernando Albericio, Ramon Eritja, Ernest Giralt, Sukhendu B. Dev, Felix Ritort. Electrostatic Binding And Hydrophobic Collapse of Peptide-Nucleic Acid Aggregates Quantified Using Force Spectrocopy. ACSNanos,7, 5102-5113 (2013).
• Vida Castro, Juan B. Blanco-Canosa, Hortensia Rodriguez, Fernando Albericio. Imidazole-1-sulfonyl azide Based Based Diazo-Transfer Reaction for the Preparation of Azido-Solid Supports for Solid Phase Synthesis. ACS Comb. Sci., 15, 331-334 (2013).
• Anna-Iris Fernandez-Llamazares, Jesus Garcia, Vanessa Soto-Cerrato, Ricardo Perez-Tomas, Jan Spengler, Fernando Albericio. N-Triethylene glycol (N-TEG) as a surrogate for the N-methyl group. Application to Sansalvamide A peptide analogs. Chem. Commun., 49, 6430-6432 (2013).
• Luísa Custódio, Ana Luísa Escapa, João Patarra, Rosa Aligué, Fernando Albericio, Nuno Rosa Neng, José Manuel Florêncio Nogueira, Anabela Romano. Sapwood of Carob Tree (Ceratonia siliqua L.) as a Potential Source of Bioactive Compounds. Records Nat. Prod. 7, 225-229 (2013).
• Judit Tulla-Puche, Sara Auriemma, Chiara Falciani, Fernando Albericio. Orthogonal Chemistry for the Synthesis of Thiocoraline-Triostin Hybrids. Exploring their Structure-Activity Relationship. J. Med. Chem., 56, 5587-5600 (2013).
• Ramon Subiros-Funosas, Lidia Nieto-Rodriguez, Knud J. Jensen, Fernando Albericio. COMU: scope and limitations of the lastest innovation in peptide acyl transfer reagents. J. Pept. Sci., 19, 408-414 (2013).
• Sara Preciado, Lorena Mendive-Tapia, Carolina Torres-García, Rubí Zamudio-Vázquez, Vanessa Soto-Cerrato, Ricardo Perez-Tomas, Fernando Albericio, Ernesto Nicolás, Rodolfo Lavilla. Synthesis and Biological Eevaluation of a Postsynthetic Modificated Trp-Based Diketopiperazine. MedChemComm., 4, 1171-1174 (2013).
• Ingrid Cabrera, Elisa Elizondo, Olga Esteban, Jose Luis Corchero, Marta Melgarejo, Daniel Pulido, Alba Córdoba, Evelyn Moreno, Esther Vazquez, Ibane Abasolo, Simo Schwartz Jr., Antonio Villaverde, Fernando Albericio, Miriam Royo, Maria Parajo, Nora Ventosa, Jaume Veciana. Multifunctional nanovesicle-bioactive conjugates prepared by a one-step procedure using CO2-expanded solvents. NanoLett., 13, 3766-3774 (2013).
• Marta Pelay-Gimeno, Yésica García-Martín, M. Jesus Martin, Jan Spengler, J.M. Molina-Guijarro, Simon Munt, Andrés M. Francesch, Carmen Cuevas, Judit Tulla-Puche, Fernando Albericio.Total synthesis of Pipecolidepsin A, the first member of the Homophymine family. Nat. Commun., 4, 2352,(2013). DOI: 10.1038/ncomms3352
• Marta Paradís-Bas, Judit Tulla-Puche, Aikaterini A. Zompra, Fernando Albericio. RADA-16: A Tough peptide. Strategies for the synthesis and purification. EurJOC, 26, 5871-5878 (2013).
• Sara Preciado, Lorena Mendive-Tapia, Fernando Albericio, Rodolfo Lavilla. Straightforward Synthesis of C-2-Arylated Tryptophan Amino Acids and Related Compounds through Palladium Catalyzed C-H Activation. J. Org. Chem., 78, 8129-8135 (2013).
• Tobias M. Postma and Fernando Albericio. N-Chlorosuccinimide, an Efficient Peptide Disulfide Bond Forming Reagent in Aqueous Solution. RSC Advances, 3, 14277-14280 (2013).
• Silvia Vilches, Cristina Vergara, Oriol Nicolas, Gloria Sanclimens, Sandra Merino, Sonia Varon, Fernando Albericio, Miriam Royo, Jose A. del Rio, Rosalina Gavin. Neurotoxicity of prion peptides mimicking the central domain of the cellular prion protein. PLOSONE, 8, e70881 (2013).
• Ana I. Fernández-Llamazares, Jesús García, Jaume Adan, Francesc Mitjans, Jan Spengler, Fernando Albericio. The backbone N-(4-azidobutyl) linker for conjugation onto (cyclic) peptides. Org. Lett., 15, 4572-4575 (2013).
• Rajshekhar Karpoormath, Fernando Albericio, Thavendran Govender, Glenn E.M. Maguire, Hendrik G. Kruger. Synthesis and NMR elucidation of Pentacycloundecane derivedhydroxy acid peptides as potential anti-HIV-1 agents. Structural. Chem., 24, 1461-1471 (2013).
• Prabhakar Cherkupally, Gerardo A. Acosta, Lidia Nieto-Rodriguez, Jan Spengler, Hortensia Rodriguez, Sherine N. Khattab, Ayman El-Faham, Marina Shamis, Yoav Luxembourg, Rafel Prohens, Ramon Subiros-Funosas, Fernando Albericio. K-Oxyma: a strong acylation-promoting, 2-CTC resin-friendly coupling additive. EurJOC., 6372-6378 (2013).
• Xavier Just-Baringo, Fernando Albericio, Mercedes Álvarez. From 2,6-dichloronicotinic Acid to Thiopeptides’ Cores. EurJOC., 6404-6419 (2013).
• Ayman El-Faham, Zainab A.L. Marhoon, Ahmed Abdel-Megeed, Fernando Albericio. Oxyma Pure/DIC: An eficiente Reagent for the Synthesis of a Novel Series of 4-[2-(2-Acetylaminophenyl)-2-oxo-acetylamino] Benzoyl Amino Acid Ester Derivative. Molecules,18, 14747-14759 (2013).
• Silvana L. Giudicessi, Juan M. Gurevich-Messina, María C. Martínez-Ceron, Rosa Erra-Balsells, Fernando Albericio, Osvaldo Cascone, Silvia A Camperi. Friendly Strategy to Prepare Encoded One bead-One Compound Cyclic Peptide Library. ACS Comb. Sci., 15, 525-529 (2013).
• Fanny Guzmán, Sergio Marshall, Claudia Ojeda, Fernando Albericio, Patricio Carvajal-Rondanelli. Inhibitory effect of short cationic homopeptides against Gram-positive bacteria. J. Peptide Sci., 19, 792-800 (2013).
• Angela Torres,Fernando Albericio, Miriam Royo. Polyproline-OEG co-oligomeric dendrimers: A family of highly branched polyproline macromolecules. EurJoc.,8279-8287 (2013).
• Marta Pelay-Gimeno, Alessandra Meli, Judit Tulla-Puche, Fernando Albericio. Rescuing Biological Activity from Synthetic Phakellistatin 19. J. Med. Chem., 56, 9780-9788 (2013).
• João Varela, Catarina Vizetto-Duarte, Luisa Custodio, Luísa Barreira, and Fernando Albericio. Marine peptides and proteins with cytotoxic and antitumoral properties. In Marine Proteins & Peptides: Development, Biological Activities, & Industrial Perspectives (Se-Kwon Kim, ed.) Wiley-Blackwell, pp. 407-430 (2013).
• Fernando Albericio, Mercedes Alvarez, Paolo Bruno, Librada Canedo, Carmen Cuevas, Andres Francesch, Yesica Garcia-Ramos, Xavier Just, Jesus Martin, Simon Munt, Marta Pelay, Jan Spengler, Judit Tulla-Puche. State of the art in the synthesis of complex natural marine peptides. Peptide Science, Volume 50th, Japanese Peptide Society, pp. 13-16 (2013).
• Ana I. Fernández-Llamazares, Jaume Adan, Francesc Mitjans, Jan Spengler, Fernando Albericio. Tackling lipophilicity of peptide drugs: Replacement of the backbone N-methyl group of Cilengitide by N-oligoethylene glycol (N-OEG) chains. Bioconj. Chem., 25, 11-17 (2014).
• Ana I. Fernández-Llamazares, Jan Spengler and Fernando Albericio. The potential of N-Alkoxymethyl groups as potential peptide backbone protectants. Tetrahedron Lett., 55, 184-188 (2014).
• Jan Spengler, Fernando Albericio.Synthesis of all Diastereomers of 2-Amino-3-hydroxy-4,5-dimethylhexanoic acid. Eur. J. Org. Chem., 44-47 (2014).
• Ayman El-Faham, Sherine N. Khattab, Ramon Subirós-Funosas, Fernando Albericio.BOP-OXy, BOP-OBt, and BOP-OAt: Novel Organophosphinic Coupling Reagents Useful for Solution and Solid-Phase Peptide Synthesis. J. Peptide Sci., 20, 1-6 (2014).
• Nancy B. Iannucci, Lucrecia M. Curto, Fernando Albericio, Osvaldo Cascone, Jose M. Delfino. Structural glance into a novel anti-staphylococcal peptide. Biopolymers (Peptide Sci.), 102, 49-57 (2014).
• Miriam Góngora-Benítez,Judit Tulla-Puche,Fernando Albericio. Multifaceted roles of disulfide bonds. Peptides as Therapeutics. Chem. Rev., 114, 901-926 (2014).
• Rubi Zamudio-Vazquez, Fernando Albericio, Judit Tulla-Puche, Keith R. Fox. Thioster Bonds of Thiocoraline can be replaced with NME-Amide Bridges without affecting its DNA-binding properties. ACS Med. Chem. Lett., 5, 45-50 (2014).
• Xavier Just-Baringo, Fernando Albericio, Mercedes Álvarez. Thiopeptide Antibiotics: Retrospective and Redecent Advances. Marine Drugs, 12, 317-351 (2014).
• Merlyn Thandu,Valentina Rapozzi,Luigi Xodo, Fernando Albericio, Clara Comuzzi, Silvia Cavalli. “Clicking” Porphyrins to Magnetic Nanoparticles for Biomedical Applications. ChemPlusChem., 79, 90-98 (2014).
• Kayena D. Zaqueo, Anderson M. Kayano, Rodrigo Simoes-Silva, Leandro S. Moreira-Dill, Carla F.C: Fernandes, Andre L: Fuly, Vinicius G. Maltarollo, Kathia M. Honorio, Saulo Luís da Silva, Gerardo Acosta, Eliandre de Oliveira, Maria Antonia O. Caballol, Fernando Albericio, Leonardo de Azevedo Calderon, Andreimar Martins Soares, Rodrigo G. Stabeli. Isolation and biochemical characterization of a new thrombin-like serine protease from Bothrops pirajai snake venom. BioMed Res., dx.doi.org/10.1155/2014/595186; 595186/1-595186/14 (2014).
• Andres Parra, Samuel Martin-Fonseca, Francisco Rivas, Fernando J. Reyes-Zurita, Marta Medina-O’Donnell,Antonio Martinez, Andres Garcia-Granados, Jose A. Lupiañez, Fernando Albericio. Semi-synthesis of acylated triterpenes from olive-oil industry wastesfor the development of anticancer and anti-HIV agents.. Eur. J. Med. Chem., 74, 278-301 (2014)
• Walesa Martins, Paulo A. Baldasso, Kathia M. Honório, Vinicus G. Maltarollo, Rosyiara I.M.A. Ribeiro, Bruna M.A. Carvalho, Leonardo A. Calderon, Rodrigo G. Stabeli, M. Antonia O. Caballol, Gerardo Acosta, Eliandre de Oliveira, Andreimar M. Soares, Sergio Marangoni, Fernando Albericio, Saulo L. Da Silva. A novel phospholipase A2 (D49) from the venom of the Crotalus oreganus abyssus (North American Grand Canyon Rattlesnake). BioMed Res. dx.doi.org/10.1155/2014/654170; 654170/1-654170/1 (2014).
• Daniel Pulido, Fernando Albericio, Miriam Royo. Controlling multivalency and multimodality: Up to pentamodal dendritic platforms based on diethylenetriaminepentaacetic acid (DTPA) cores. Org. Lett., 16, 1318-1321 (2014).
• Tobias M. Postma,Fernando Albericio. Cysteine Pseudoprolines for Thiol Protection and Peptide Macrocyclization Enhancement in Fmoc-Based Solid-Phase Peptide Synthesis. Cysteine. Org. Lett., 16, 1772-1775 (2014).
• Tobias M. Postma, Fernando Albericio. Immobilized N-Chlorosuccinimide as a Friendly Peptide Disulfide Forming Reagent. ACS Comb. Sci., 16, 43-52 (2014).
• Javier Sánchez-Nieves, Peter Fransen, Daniel Pulido, Raquel Lorente, M. Ángeles Muñoz-Fernández, Fernando Albericio, Miriam Royo, Rafael Gómez, F. Javier de la Mata. Amphiphilic Cationic Carbosilane-PEG Dendrimers: Synthesis and Applications in Gene Therapy. Eur. J. Med. Chem., 76, 43-52 (2014).
• Saulo L. Da Silva, Edward G. Rowan, Fernando Albericio, Rodrigo G. Stábeli, Leonardo A. Calderon, Andreimar M. Soares. Animal Toxins and Their Advantages in Biotechnology and Pharmacology. BioMed Res., dx.doi.org/10.1155/2014/951561; 951561 (2014).
• Cesar Guimaraes, Silvia Andrião-Escarsoc, Bruna Mara Aparecida De Carvalho, Daniela Marchi-Salvador, Norivaldo Santos-Filho, Carlos Fernandes, M. R M Fontes, J. R. Giglio, Benedito Barraviera, Carla Fernandes, Leonardo de Azevedo Calderon, Rodrigo Guerino Stabeli, Fernando Albericio, Saulo Luís da Silva. Alkylation of histidine residues of Bothrops jararacussu venom proteins and isolated phospholipases A2: A biotechnological tool to improve the production of antibodies. BioMed Res., dx.doi.org/10.1155/2014/981923; 981923 (2014).
• Peter Fransen, Daniel Pulido, Chantal Sevrin, Christian Granfils, Miriam Royo, Fernando Albericio. High control, fast growth OEG-based dendron synthesis via a sequential two-stepprocess of copper-free diazo transfer and click chemistry. Macromol., 47, 2585-2591 (2014).
• Alvaro Siano, Paula I. Gatti, Eliandre de Oliveira, Fernando Albericio, Arturo C. Simonetta, Rafael Lajmanovich, Georgina G. Tonarelli. Antimicrobial peptides from skin secretions of Hypsiboas pulchellus. J. Nat. Prod., 77, 831-841 (2014).
• Luis J. Cruz, Felix Rueda, Lorena Simón, Begoña Cordobilla, Fernando Albericio, Joan Carles Domingo. Liposomes containing NY-ESO-1/tetanus toxoid and adjuvant peptides targeted to human DCs via Fc receptor strongly enhance immunological response in cancer vaccines. Nanomedicine, 9, 435-449 (2014);10.2217/NNM.13.66.
• María B. Pastrian, Fanny Guzmán, Giselle V. Ripoll, Juan Garona, Marina Pifano, Osvaldo Cascone, Graciela N. Ciccia, Fernando Albericio,Daniel E. Gómez, Daniel F. Alonso, Nancy B. Iannucci. Structure-activity relationship of 1-desamino-8-D-arginine vasopressin as an antiproliferative agent on human V2 receptor-expressing cancer cells, Mol. Medicine Rep., 10.3892/mmr.2014.21409, 2568-72 (2014).
• M. Godoy-Gallardo, Carles Mas-Moruno, M.C. Fernández-Calderón, C. Pérez, Josep M. Manero, Fernando Albericio, Francisco J Gil, D. Rodríguez.Covalent Immobilization of hLf1-11 Peptide onto Titanium Surface Reduces Bacterial Adhesion and Biofilm Formation. Acta Biomateria,http://dx.doi.org/10.1016/j.actbio.2014.03.026, 10, 3522-3534 (2014).
• Xavier Just-Baringo, Paolo Bruno, Cristina Pitart, Jordi Vilà, Fernando Albericio, Mercedes Álvarez. Dissecting the Structure of Thiopeptides: Assessment of Thiazoline and Tail Moieties of Baringolin and Antibacterial Activity Optimization. J. Med. Chem., 57, 4185-4195 (2014).
• Majid D. Farahani, Bahareh Honarparvar, Fernando Albericio, Glenn E. M. Maguire,Thavendran Govender,Per I. Arvidsson Hendrik G. Kruger. Proline N-oxides: Modulators of the 3D Conformation of Linear Peptides through “NO-turns. Org. Biomol. Chem. 12, 4479-4490 (2014).
• María Jesús Martín, Raquel Rodríguez-Acebes, Yésica García-Ramos,Valentín Martínez, Carmen Murcia, Isabel Digón, Isabel Marco, Rogelio Fernández, Fernando Reyes, Andrés M. Francesch, Simon Munt, Marta Pelay-Gimeno, Judit Tulla-Puche, Fernando Albericio, and Carmen Cuevas. Stellatolides, a new cyclodepsipeptide family, from the sponge Ecionemia acervus. Isolation, Solid-phase Total Synthesis and Full Structural Assignment of Stellatolide A. J. Am. Chem. Soc., 136, 6754-6762 (2014).
• Prabhakar Cherkupally, Gerardo A. Acosta,Suhas Ramesh,Beatriz G. De la Torre, Thavendran Govender,Hendrik G. Kruger,and Fernando Albericio. Solid-Phase Peptide Synthesis (SPPS), C-Terminal vs. Side-chain Anchoring: a Reality or a Myth. Amino Acids, doi: 10.1007/s00726-014-1746-7; 46, 1827-1838 (2014).
• Tobias M. Postma, Fernando Albericio. Novel Disulfide Formation Strategies in Peptide Synthesis. EurJoc., 3519-3530 (2014), with cover.
• Alberto Ruiz, Margarita Suárez, Nazario Martin, Fernando Albericio, and Hortensia Rodriguez. Morphological characterization of fullerene-androsterone conjugates. Beilstein, Nanotech., 5, 374-379 (2014).
• Xavier Just-Baringo, Fernando Albericio, Mercedes Álvarez. Chiral Thiazoline and Thiazole Building Blocks for the Synthesis of Peptide-Derived Natural Products. Curr. Topics Med. Chem. 14, 1244-1256 (2014).
• Xavier Just-Baringo, Fernando Albericio, Mercedes Alvarez. Thiopeptide Engineering: A Multidisciplinary Effort Towards Future Drugs. Angew. Chemie, 53, 6602-6616 (2014).
• Suhas Ramesh, Prabhakar Cherkupally, Beatriz G. de la Torre, Thavendran Govender, Hendrik G. Kruger, Fernando Albericio. Microreactors for peptide synthesis: looking through the eyes of twenty first century !!!Amino acids, DOI 10.1007/s00726-014-1776-1, 46, 2091-2104. (2014).
• Paola Agrigento, Fernando Albericio, Sylvie Chamoin, Isabelle Dacquignies, Halil Koc, Martin Eberle. Facile and Mild Ligation of Linear and Cyclic Peptide Thioesters. Org. Lett., 16, 3922-3925 (2014).
• Carles Mas-Moruno, R. Fraioli, Fernando Albericio, Josep M. Manero, and Francisco J. Gil. Novel peptide-based platform for the dual presentation of biologically active peptide motifs on biomaterials. ACS Appl Mater Interfaces, 6, 6525-6536 (2014).
• Luísa Custódio, Fernando Soares, Hugo Pereira, Luísa Barreira, Catarina Vizetto Duarte, Maria João Rodrigues, Amélia Pilar Rauter, Fernando Albericio, João Varela. Fatty acid composition and biological activities of Isochrysis galbana T-ISO, Tetraselmis sp. and Scenedesmus sp.: possible application in the pharmaceutical and functional food industries. J. App. Phycology, 26, 151-161 (2014).
• Andres Parra, Samuel Martin-Fonseca, Francisco Rivas, Fernando J. Reyes-Zurita, Marta Medina-O'Donnell, Eva E. Rufino-Palomares, Antonio Martinez, Andres Garcia-Granados, Jose A. Lupianez, Fernando Albericio. Solid-Phase Library Synthesis of Bi-Functional Derivatives of Oleanolic and Maslinic Acids and Their Cytotoxicity on Three Cancer Cell Lines. ACS Comb. Sci., dx.doi.org/10.1021/co500051z; 16, 428-447 (2014).
• Stella Peña, Catherine Fagundez, Andrea Medeiros, Marcelo Comini, Laura Scarone, Diver Sellanes, Eduardo Manta, Judit Tulla-Puche, Fernando Albericio, Lindsay Stewart, Vanessa Yardley, Gloria Serra. Combined Solid Phase and Solution Synthesis of Cyclohexapeptides as promising antimalarial and anti-trypanosomal agents. Med. Chem. Comm., DOI: 10.1039/C4MD00135D, 5, 1309-1316 (2014).
• Javier Ruiz-Rodríguez, Miriam Miguel, Sara Preciado, Gerardo Acosta,Jaume Adan, Axel Bidon-Chanal, F. Javier Luque, Francesc Mitjans, Rodolfo Lavilla, Fernando Albericio. Polythiazole Linkers as Functional Rigid Connectors: a New RGD Cyclopeptide with Enhanced Integrin Selectivity. Chem. Sci., DOI: 10.1039/C4SC00572D5, 3929–3935(2014).
• Ryan J. Seelbach, Peter Fransen, Fernando Albericio, Marianna Peroglio, Mauro Alini, Daniel Pulido, Miriam Royo, Patricia Lopez-Chicon, Carlos Semino, Fabian Duttenhoefer, Sebastian Sauerbier, Philipp Niemeyer, Thomas Freiman, Alvaro Mata, and David Eglin. Multivalent dendrimers presenting spatially controlled clusters of binding epitopes in thermoresponsive hyaluronan hydrogels. Acta Biomat., DOI: 10.1016/j.actbio.2014.06.028;10, 4340-4350. (2014).
• Marta Paradis-Bas,Maria Albert-Soriano, Judit Tulla-Puche, Fernando Albericio. Lineal vs Branched poly-Lysine/Arginine as Polarity Enhancer Tags. Org. Biom. Chem., DOI:10.1039/C4OB01354A, 12, 7194-7196 (2014).
• Alba Pérez-Perarnau, Sara Preciado, Claudia Mariela Palmeri, Cristina Moncunill-Massaguer, Daniel Iglesias-Serret, Diana M. González-Gironès, Miriam Miguel, Satoki Karasawa, Satoshi Sakamoto, Ana M. Cosialls, Camila Rubio-Patiño, José Saura-Esteller, Rosario Ramón, Laia Caja, Isabel Fabregat, Gabriel Pons, Hiroshi Handa, Fernando Albericio, Rodolfo Lavilla, Joan Gil. A trifluorinated thiazoline scaffold leading to proapoptotic agents targeting prohibitins. Angew. Chemie., DOI: 10.1002/anie.201405758; 53, 10150-10154 (2014).
• Marta Paradis-Bas, Judit Tulla-Puche, Fernando Albericio.2-Methoxy-4-methylsulfinylbenzyl, A Backbone Amide Safety Catch Protecting Group for Synthesis and Purification of Difficulty Sequence Peptides. DOI: 10.1002/chem.201403668; Chem., Eur. J. 20, 15031-15039 (2014), with cover.
• Joan Camunas-Soler, Silvia Frutos, Cristiano V. Bizarro, Sara de Lorenzo, Maria Eugenia Fuentes-Perez, Roland Ramsch, Susana Vilchez, Conxita Solans, Fernando Moreno-Herrero, Fernando Albericio, Ramón Eritja, Ernest Giralt, Sukhendu B. Dev, Felix Ritort. Electrostatic Binding and Hydrophobic Collapse ofPeptide-Nucleic Acid Aggregates Quantified UsingForce Spectroscopy. arXiv.org, e-Print Archive, Physics, 1-56, arXiv:1408.1069v1, (2014).
• Ariel R. Guerrero, Natalia Hassan, Carlos A. Escobar, Fernando Albericio, Marcelo J. Kogan, Eyleen Araya.Gold nanoparticles for photothermally controlled drug release. doi:10.2217/nnm.14.126; Nanomedicine9, 2023-2039 (2014).
• Yahya E. Jad,Sherine N. Khattab, Beatriz G. de la Torre,Thavendran Govender,Hendrik G. Kruger,Ayman El-Faham, Fernando Albericio. Oxyma-B, an Excellent Racemization Suppressor. Org. Biomol. Chem., 12, 8379-8385 (2014).
• Adriana Lorente,Fernando Albericio, Mercedes Álvarez. Selective formation of a Z-trisubstituted double bond using a 1-(tert-butyl)-tetrazolyl sulfone. J. Org. Chem., 79, 10648-10654 (2014).
• Prabhakar Cherkupally, Suhas Ramesh, Beatriz G. de la Torre, Thavendran Govender, Hendrik G. Kruger,Fernando Albericio.Immobilized Coupling Reagents: Synthesis of Amides/Peptides. DOI:10.1021/co500126y; ACS, Comb. Sci.,16, 579-601 (2014).
• Yahya E. Jad,Sherine N. Khattab, Beatriz G. de la Torre,Thavendran Govender,Hendrik G. Kruger,Ayman El-Faham, Fernando Albericio. TOMBU and COMBU as a novel uronium-type peptide coupling reagents derived from Oxyma-B. doi:10.3390/molecules191118953. Molecules,18953-18965 (2014).
• Carolina Torres-Garcia, Daniel Pulido, Fernando Albericio, Miriam Royo, Ernesto Nicolas. Triazene as a powerful tool for solid-phase derivatization ofphenylalanine containing peptides: Zygosporamide analogues as aproof of concept. J. Org. Chem., 79, 11409-11415 (2014).
• Sabine Oberhans, Albert G. Castano, Anna Lagunas, Elisabet Prats-Alfonso, Michael Hirtz, Fernando Albericio, Harald Fuchs, Josep Samitier, Elena Martinez. Mesopattern of immobilized bone morphogenetic protein-2 created by Microcontact Printing and Dip-pen Nanolithography influence C2C12 cell fate. RSC, Advances, DOI: 10.1039/C4RA10311D; 4, 56809-56815 (2014).
• Adriana Lorente, Kamil Makowski, Fernando Albericio, Mercedes Álvarez. Bioactive Marine Polyketides as Potential and Promising Drugs. Ann. Mar. Biol. Res., 1,1003 (2014).
• Sachin A. Pawar,Amit M. Jabgunde, Glenn E. M. Maguire, Dilip D. Dhavale,Thavendran Govender,Hendrik G. Kruger,Fernando Albericio. Conformational Comparison of Cyclic α3β Tetra- vsα4β Pentapeptides. South African J Chem.,67, 80-84 (2014).
• Silvia A. Camperi, Maria C. Martínez-Ceron, Silvana L. Giudicessi, Maria M. Marani, Fernando Albericio, O. Cascone. Peptide affinity chromatography based on combinatorial strategies for protein purification. In Protein Downstream Processing, Methods in Molecular Biology, Humana Press-Springer, 1129, 277-302 (2014).
• Sherine N Khattab, Ayman El-Faham, Ramon Subiros-Funosas, Fernando Albericio.Organophosphinic coupling reagents in peptide synthesis. Proceedings of the Annual International Conference on Chemistry, Chemical Engineering and Chemical Process, 2, 6-10 (2014).
• Ayman El-Faham, Zainab Al Marhoon,Ahmed Abdel-Megeed, Sherine Khattab, Adnan Bekhit, Fernando Albericio. α-Ketoamino acid ester derivatives as promising MAO inhibitors. Bioorg. Med. Chem. Lett., 25, 70-74 (2015).
• Janire Lamariano-Merketegi, Adriana Lorente,Alejandro Gil, Fernando Albericio, Mercedes Álvarez. Addition of vinylmetalic reagents to chiral 2-formyltetrahydofuran. EurJOC., pp. 235-241 (2015).
• Adriana Lorente, Alejandro Gil, Rogelio Fernandez, Carmen Cuevas, Fernando Albericio, Mercedes Alvarez. Phormidolides B and C, cytotoxic agents from the sea. Enantioselective synthesis of the macrocyclic core. Chem., Eur. J. 21, 150-156 (2015), with cover.
• Juan M. Gurevich-Messina, Silvana L. Giudicessi, María C. Martínez-Ceron, Gerardo Acosta, Rosa Erra-Balsells, Osvaldo Cascone, Fernando Albericio, Silvia A. Camperi. A Simple Protocol for Combinatorial Cyclic Depsipeptide Libraries Sequencing by Matrix Assisted Laser Desorption/Ionisation Mass Spectrometry. J. Pept. Sci., 21, 40-45 (2015).
• Yahya E. Jad, Gerardo A. Acosta, Sherine N. Khattab, Beatriz G. de la Torre,Thavendran Govender,Hendrik G. Kruger,Ayman El-Faham, and Fernando Albericio. Peptide Synthesis Beyond DMF: THF and ACN as Excellent and Greener Alternatives. Org. Biomol. Chem., 13, 2393-2398 (2015).
• Jyotibon Dutta, Suhas Ramesh, Siduduzo M. Radebe, Anou M. Somboro, Beatriz G. de la Torre, Hendrik G. Kruger, Sabiha Y. Essack, Fernando Albericio, Thavendran Govender. Optimized microwave assisted synthesis of LL37, a cathelicidin human antimicrobial peptide. Int. J. Peptide Res. Therap. 21, 13-20 (2015).
• Suhas Ramesh,Prabhakar Cherkupally, Thavendran Govender, Hendrik G. Kruger, Fernando Albericio, Beatriz G. de la Torre. 6-(Bromomaleimido)hexanoic Acid as a Connector for the Construction of a Multiple Branched Peptide Platform. Org. Lett., 17, 464-467 (2015).
• Marta Paradis-Bas, Judit Tulla-Puche, Fernando Albericio. Semipermanent C‑Terminal Carboxylic Acid Protecting Group:Application to Solubilizing Peptides and Fragment Condensation. Org. Lett., 17, 294-297 (2015).
• Luísa Custódio, João Patarra; Fernando Alberício; Nuno R Neng; José Manuel Florêncio Nogueira; Anabela Romano. Phenolic composition, antioxidant potential and in vitro inhibitory activity of leaves and acorns of Quercus suber on key enzymes relevant for hyperglycemia and Alzheimer disease. Ind. Crops Prod. 64, 45-51 (2015).
• Cristina de la Torre, Isolda Casanova, Gerardo Acosta, Carmen Coll, María José Moreno, Fernando Albericio, Elena Aznar, Ramón Mangues, Miriam Royo, Félix Sancenón, Ramón Martínez-Máñez. Gated Mesoporous Silica Nanoparticles Using a Double-Role Circular Peptide for the Controlled and Target-Preferential Release of Doxorubicin in CXCR4-Expresing Lymphoma Cells. Adv. Funct. Mat. 25, 687-695 (2015).
• Delia Hernandez, Giovana C. Granados, Esmeralda Sánchez, Fernando Albericio, Mercedes Álvarez. Palladium-cataluzed coupling reactions for the preparation of concatenated azoles. ARKIVOC, pp. 34-43 (2015).
• Joan Camunas-Soler, Maria Manosas, Silvia Frutos, Judit Tulla-Puche, Fernando Albericio, Felix Ritort. Single-Molecule Kinetics and Footprinting of DNA bis-intercalation: the Paradigmatic Case of Thiocoraline. Nucleic Acid Res., 43, 2767-2769 (2015).
• Susana P. Egusquiaguirre, Cristina Manguán-García, Laura Pintado-Berninches, Laura Iarriccio, Daniel Carbajo, Fernando Albericio, Miriam Royo, José Luís Pedraz, Rosa M. Hernández, Rosario Perona, Manuela Igartua. Development of surface modified biodegradable polymeric nanoparticles to deliver GSE24.2 peptide to cells: A promising approach for the treatment of defective telomerase disorders. Eur. J. Pharmac. Biopharmac., 91, 91-102 (2015).
• Carlos Heras, Iván Ramos-Tomillero,Marc Caballero, Marta Paradís-Bas, Ernesto Nicolás,Fernando Albericio, Ibério de P. R. Moreira, Josep Maria Bofill. On the mechanism of phenolic formylation mediated by TiCl4 complexes: Existence of biradical intermediates induced by valence tautomerimsm. Eur. JOC., pp. 2111-2118 (2015).
• Iván Ramos-Tomillero, Marta Paradís-Bas, Ibério de Pinho Ribeiro Moreira, Josep María Bofill, Ernesto Nicolás, Fernando Albericio. Formylation of electron-rich aromatic rings with dichloromethyl methyl ether and TiCl4. Molecules, 20, 5409-5422 (2015).
• Iván Ramos-Tomillero, Hortensia Rodríguez, Fernando Albericio. Tetrahydropyranyl (Thp), a non-aromatic acid-labile Cys protecting group for Fmoc peptide chemistry. Org. Lett., 17, 1680-1683 (2015).
• Prabhakar Cherkupally, Suhas Ramesh, Thavendran Govender,Hendrik G. Kruger,Beatriz G. de la Torre, andFernando Albericio An Efficient Solid-Phase Strategy for Total Synthesis of Naturally Occurring Amphiphilic Marine Siderophores: Amphibactin-T and Moanachelin ala-B. Org. Biomol. Chem., 13, 4760-4768 (2015).
• Anabel Molero, Marc Vendrell, Jordi Bonaventura, Julian Zachmann, Laura Lopez, Leonardo Pardo, Carme Lluis, Antoni Cortes, Fernando Albericio, Vicent Casado, Miriam Royo. A solid-phase combinatorial approach for indoloquinolizidinepeptides with high affinity at D1 and D2 dopamine receptors. Eur. J. Med. Chem., 97, 173-180 (2015).
• Yahya E. Jad, Sherine N. Khattab, Beatriz G. de la Torre, Thavendran Govender, Hendrik G. Kruger, Ayman El-Faham, Fernando Albericio. EDC.HCl and Potassium Salts of Oxyma and Oxyma-B as Superior Coupling Cocktail for Peptide Synthesis. EurJOC, 3116-3120 (2015).
• Lorena Mendive-Tapia,Sara Preciado, Jesús García, Rosario Ramón, Fernando Albericio, Rodolfo Lavilla. Two-electron Connection between Tryptophan and Phenylalanine/Tyrosine Residues: Linked, Constrained and Stapled Peptides through C-H Activation Processes.Nat. Comm., 6:8160 (2015) | DOI: 10.1038/ncomms8160.
• Claudio Zapata-Urzúa, Magdalena Pérez-Ortiz, Gerardo A. Acosta, Joan Mendoza, Lluis Yedra,Sonia Estradé, Alejandro Alvarez-Lueje, Luis Núñez-Vergara, Fernando Albericio, Rodolfo Lavilla, Marcelo J. Kogan. Hantzsch Dihydropyridines: Privileged Structures for the Formation of well-defined Gold Nanostars.J. Colloid Interf. Sci, 453, 260-269 (2015).
• Juan B. Blanco-Canosa, Brunello Nardone, Fernando Albericio, Philip E. Dawson. Chemical protein synthesis using a secondgeneration N-acylurea linker for the preparation of peptide-thioester precursors. J. Am. Chem. Soc., 137, 7197-7209 (2015).
• Markus Muttenthaler, Fernando Albericio, Philip E. Dawson. Methods, setup and safe handling for anhydrous hydrogen fluoride cleavage in Boc solid-phase peptide synthesis. Nature Protocols, 10, 1067-1083 (2015).
• Ryan J. Seelbach, Peter Fransen, Daniel Pulido, Matteo D'Este, Fabian Duttenhoefer, Sebastian Sauerbier, Thomas M. Freiman, Philipp Niemeyer, Fernando Albericio, Mauro Alini, Miriam Royo, Alvaro Mata, David Eglin. Macromol. Biosci. 15, 1035-1044 (2015).
• Catarina Vizetto-Duarte, Hugo Pereira, Carolina Bruno de Sousa, Pilar Amelia Rauter, Fernando Albericio, Luísa Custódio, Luísa Barreira, João Varela. Fatty acid profile of different species of algae of the Cystoseira genus: a nutraceutical perspective. Nat. Prod. Res., 29, 1264-1270 (2015).
• Rubi Zamudio-Vazquez, Saska Ivanova, Miguel Moreno,Maria Isabel Hernandez-Alvarez, Ernest Giralt, Axel Bidon-Chanal, Antonio Zorzano, Fernando Albericio, Judit Tulla-Puche. A New Quinoxaline-Containing Peptide Induces Apoptosis in Cancer Cells Through Autophagy Modulation. Chem. Sci., 6, 4537-4549 (2015).
• Sherine N. Khattab, Hosam H. Khalil, Adnan A. Bekhit, Mohamed Mokbel Abd El-Rahman, Ayman El-Faham, Fernando Albericio Synthesis and prelimnary biological evaluation of 1,3,5-triazine amino acid derivatives to study their MAO inhibitors.Molecules, 20, 15976-15988 (2015).
• Carme Pastells, Gerardo Acosta, Nuria Pascual, Fernando Albericio, Miriam Royo, M. Pilar Marco.An immunochemical strategy based on peptidoglycan synthetic peptide epitopes to diagnose Staphylococcus aureus infections. Anal. Chim. Acta, 889, 203-211 (2015)
• Ana I. Fernández-Llamazares, Jan Spengler, Fernando Albericio.Backbone N-modified peptides: how to meet the challenge of secondary amine acylation. Biopolymers (Pept. Sci), 104, 435-452 (2015).
• Pau Rocas, Yolanda Fernández, Simó Schwartz Jr, Ibane Abasolo, Josep Rocas, Fernando Albericio. Multifunctionalized polyurethane–polyurea nanoparticles: hydrophobically driven self-stratification at the o/w interface modulates encapsulation stability. J. Mat., Chem. B., 3, 7604-7613 (2015).
• Pau Rocas, Mireia Hoyos-Nogués, Josep Rocas, José M. Manero, Javier Gil, Fernando Albericio, Carlos Mas-Moruno. Installing Multifunctionality on Titanium with RGD-decorated Polyurethane-Polyurea Roxithromycin Loaded Nanocapsules: Towards New Osteointegrative Therapies. Adv. Health Mat., 4, 1956-1960 (2015).
• Shah Md. Abdur Rauf, Per I. Arvidsson,Fernando Albericio, Thavendran Govender, Glenn E. M. Maguire, Hendrik G. Kruger,Bahareh Honarparvar. The effect of N-methylation of amino acids (Ac-X-OMe) on solubility and conformation: A DFT study. Org. Biomol. Chem., 13, 9993-10006 (2015).
• Roxana González-Stegmaier, Fanny Guzmán, Fernando Albericio, Franz Villarroel-Espíndola, Alex Romero, Victoriano Mulero, Luis Mercado. A synthetic peptide derived from the D1 domain of flagellin induced the expression of proinflammatory cytokines in fish macrophages. Fish & Sellfish Immunol., 47, 239-244 (2015).
• Luísa Custódio, João Patarra; Fernando Alberício; Nuno R Neng; José Manuel Florêncio Nogueira; Anabela Romano. In vitro antioxidant and inhibitory activity of water decoctions of carob tree (Ceratonia siliqua L.) on cholinesterase, α-amylase and α-glucosidase. Nat. Prod. Res., 29, 2155-2159 (2015).
• Anderson M. Kayano, Rodrigo Simões-Silva, Patricia S.M. Medeiros, Vinícius G. Maltarollo, Kathia M. Honorio, Eliandre Oliveira, Fernando Albericio, Saulo L. da Silva, Anna Caroline C. Aguiar, Antonia U. Krettli, Carla F.C. Fernandes, Juliana P. Zuliani, Leonardo A. Calderon, Rodrigo G. Stábeli, Andreimar M. Soares. BbMP-1, a new metalloproteinase isolated from Bothrops brazili snake venom within vitro antiplasmodial properties. Toxicon, 106, 30-41 (2015).
• Yahya E. Jad, Gerardo A. Acosta, Tricia Naicker, Melissa Ramtahal, Ayman El-Faham, Thavendran Govender, Hendrik G. Kruger, Beatriz G. de la Torre, Fernando Albericio. Synthesis and Biological Evaluation of a Teixobactin Analogue. Org. Lett., 17, 6182-6185 (2015).
• Alejandro Gil, Adriana Lorente, Fernando Albericio, and Mercedes Álvarez. Stereoselective allylstannane addition for a convergent synthesis of a complex molecule. Org. Lett., 17,6246-6249(2015).
• Cristina Moncunill-Massaguer, José Saura-Esteller, Alba Pérez-Perarnau, Claudia Mariela Palmeri, Sonia Núñez-Vázquez, Ana M. Cosialls, Diana M. González-Gironès, Helena Pomares, Anne Korwitz, Sara Preciado, Fernando Albericio, Rodolfo Lavilla, Gabriel Pons, Thomas Langer, Daniel Iglesias-Serret, Joan Gil. A Novel prohibitin-biding compound induces the mitochondrial apoptotic pathway through NOXA and BIM upregulation. Oncotargets.,6, 41750-41765(2015), DOI: 10.18632/oncotarget.6154.
• Luísa Custódio, Fernando Soares, Hugo Pereira, Maria João Rodrigues, Luísa Barreira, Amélia Pilar Rauter, Fernando Alberício, João Varela. Botryococcus braunii and Nannochloropsis oculata extracts inhibitcholinesterases and protect human dopaminergic SH-SY5Y cellsfrom H2O2-induced cytotoxicity. J Appl Phycol27, 839–848 (2015).
• N. Sherine Khattab, Ayman El-Faham, Fernando Albericio Peptide Coupling Reactions. J. Mol. Pharm. Org. Process Res.,3, e119. doi: 10.4172/2329-9053.1000e119(2015).
• Peter Fransen, Daniel Pulido, Lorena Simón-Gracia Ana Paula Candiota, Carles Arús, Fernando Albericio, Miriam Royo.r1 and r2 relaxivities of dendrons based on a OEG-DTPA architecture: effect of Gd3+ placement and dendron functionalization. J. Nanotech., http://dx.doi.org/10.1155/2015/848020 (2015)
• Suhas Ramesh, Prabhakar Cherkupally, Thavendran Govender, Hendrik G. Kruger, Fernando Albericio,Beatriz G. de la Torre. Platforms for Peptide Vaccine Constructs.Peptide and Protein Vaccines "Advances in Protein Chemistry and Structural Biology", Elsevier, pp. 99-130 (2015), with book cover.
• Judit Tulla-Puche, Ayman El-Faham, Athanassios S. Galanis, Eliandre de Oliveira, Aikaterini A. Zompra, and Fernando Albericio. Methods for the synthesis and analysis of Peptides. In Peptide Drugs: Peptide Chemistry and Drug Design (B.M. Dunn, ed.) Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim (Germany), 2015, pp. 11-74.
• Jesus Herraiz-Cobo, Fernando Albericio, Mercedes Álvarez. The Larock Reaction. in the Synthesis of Heterocyclic Compounds, In Advances in Heterocyclic Chemistry, Vol. 116 (E.F.V. Scriven, and C.A. Ramsden, ed.), Academic Press-Elsevier, 2015, pp 1–35.
• Iván Ramos-Tomillero, Hortensia Rodríguez, Fernando Albericio.Trends to Acid-Labile Cys Protecting Groups: Thp as an Efficient and Non-Aromatic Cys Protecting Group for Fmoc Chemistry. In Proceedings of the 24th American Peptide Symposium (V. Srivastava, A. Yudin, M. Lebl ed), American Peptide Society, 2015, pp. 278-279.
• María C. Martínez-Ceron, Soledad L. Saavedra, Lucía Ávila, Silvana L. Giudicessi, Fernando Albericio, Silvia A. Camperi, and Osvaldo Cascone. One-Bead-One-Peptide Library to Purify Crotalus durissus terrificus Phosholipase A2 InProceedings of the 24th American Peptide Symposium (V. Srivastava, A. Yudin, M. Lebl ed), American Peptide Society, 2015, pp 137-138.
• Hendrik G. Kruger, Fernando Albericio. Advances in the Discovery and Development of Peptide Therapeutics. In Advances in the Discovery and Development of Peptide Therapeutics (H G. Kruger, F. Albericio, eds.). Future Medicine & Future Science, London (UK), 2015, pp 2-6.
• Anaïs F. M. Noisier, Fernando Albericio.Advance in ligation techniques for peptide and protein synthesis. In Amino Acids, Peptides, and Proteins Vol. 39 (Specialist Periodical Reports), M. Ryadnov, E. Farkas, Eds., Royal Society of Chemistry (London, UK), 2015; 1-20.
• Catarina Vizetto-Duarte, Luísa Custódio, Luísa Barreira, Manuela Moreira da Silva, Amelia P. Rauter, Fernando Albericio, João Varela. Proximate biochemical composition and mineral content of edible species from the Cystoseira genus. Botanica Marina., 59, 251-257 (2016).
• Vida Castro, Hortendia Rodriguez, Fernando Albericio. CuAAC: an Efficient Click Chemistry on Solid Phase. ACS, Comb Sci., 18, 1-14 (2016).
• Suhas Ramesh, Prabhakar Cherkupally, Thavendran Govender,Hendrik G. Kruger,Fernando Albericio, Beatriz G. de la Torre.Highly Chemoselective Ligation of Thiol- and Amino-Peptides on a Bromomaleimide Core. Chem. Commun., 52, 2334-2337 (2016).
• Luísa Custódio, Simona Laukaityte, Aschwin H. Engelen, Maria João Rodrigues, Hugo Pereira, Vizetto-Duarte, Luísa Barreira, Fernando Albericio, João Varela. A comparative evaluation of biological activities and bioactive compounds of the seagrasses Zostera marina and Z. noltei from Southern Portugal. Nat. Prod. Reports, 30, 724-728 (2016).Rodrigo González, Lorena Mendive-Tapia, María B. Pastrian, Fernando Albericio, Rodolfo Lavilla, Osvaldo Cascone, Nancy B. Iannucci. Enhanced Antimicrobial Activity of a Peptide Derived from Human Lysozyme by Tryptophan Residue Arylation. J. Peptide Sci., 22, 123-128 (2016).Yahya E. Jad, Gerardo A. Acosta, Sherine N. Khattab, Beatriz G. de la Torre, Thavendran Govender, Hendrik G. Kruger, Ayman El-Faham, Fernando Albericio. 2-MeTHF and CPME for Green Solid-Phase Peptide Synthesis. Amino Acids, 48, 419-426 (2016).
• María Camila Martínez-Ceron, Silvana Laura Giudicessi, Soledad Lorena Saavedra, Juan Manuel Gurevich-Messina, Rosa Erra-Balsells, Fernando Albericio, Osvaldo Cascone, Silvia Andrea Camperi. Latest advances in OBOC peptide libraries. Improvements in screening strategies and enlarging the family from linear to cyclic libraries. Curr. Pharmac. Biotech., 17, 449-457 (2016).
• Marta Paradis-Bas, Judit Tulla-Puche, Fernando Albericio. Making Easy the Synthesis of "Difficult Peptides": Solubilizing Strategies. Chem. Soc. Rev., 45, 631-654 (2016).
• Lorena Mendive-Tapia, Can Zhao, Ahsan R. Akram, Sara Preciado, Fernando Albericio, Martin Lee, Alan Serrels, Nicola Kielland, Nick D. Read, Kevin Dhaliwal, Rodolfo Lavilla,Marc Vendrell. Spacer-free BODIPY fluorogens for antimicrobial peptides: direct imaging of fungal infection in human pulmonary tissue.Nat. Commun., 7, 10940, doi:10.1038/ncomms10940 (2016).
• Ayman El-Faham, Saied Soliman, Sameh M. Osman, Hazem A. Ghabbour, Mohammed R. Siddiqui, Hoong-Kun Fun, Fernando Albericio. Synthesis, molecular structure and spectroscopic studies (X-ray, IR, NMR, UV-Vis) of novel 2-(4,6-dimethoxy-1,3,5-triazin-2-yl) amino acid ester derivatives. Spectrochim. Acta, Part A: Molec. Biomolec.,159, 184-198 (2016).
• Kayena D. Zaqueo, Anderson M. Kayano, Thaisa F. S. Domingos, Laura A. Moura, André L. Fuly, Saulo L. da Silva, Gerardo Acosta, Eliandre Oliveira, Fernando Albericio, Fernando B. Zanchi, Juliana P. Zuliani, Leonardo A. Calderon, Rodrigo G. Stábeli, Andreimar M. Soares. BbrzSP-32 thrombolytic enzyme, the first serine protease isolated from Bothrops brazili venom: Purification and characterization. Comparative Biochem. & Physiol. Part A,,195, 15-25 (2016).
• Catarina Vizetto-Duarte, Luísa Custódio, Gerardo Acosta, João Henrique G. Lago, Thiago R. Morais, Carolina Bruno de Sousa, Katkam N. Gangadhar, Maria João Rodrigues, Hugo Pereira, Raquel T. Lima, M. Helena Vasconcelos, Luísa Barreira, Amélia P. Rauter, Fernando Albericio, João Varela. Can macroalgae provide bioactive compounds with pharmaceutical potential? A closer look at Cystoseira tamariscifolia as a source for antioxidant and anti-hepatocarcinoma compounds. Peer J., 4, e1704 (2016).
• Patricio Carvajal-Rondanelli, Mónica Aróstica, Sergio Marshall, Fernando Albericio, Claudio Andrés Alvarez, Claudia Ojeda, Luis Felipe Aguilar, Fanny Guzmán. Inhibitory effect of short cationic homopeptides against Gram-negative bacteria. Amino Acids, 48, 1445-1456 (2016).
• Ingrid Cabrera, Ibane Abasolo, Jose Luis Corchero, Elisa Elizondo, Pilar Rivera, Evelyn Moreno, Jordi Faraudo, Santi Sala, Dolores Bueno, Elisabet Gonzalez-Mira, Merche Rivas, Marta Melgarejo, Daniel Pulido, Fernando Albericio Miriam Royo, Antonio Villaverde, Maria F. García-Parajo, Simó Schwartz Jr., Nora Ventosa, Jaume Veciana. α-Galactosidase A Loaded Nanoliposomes with Enhanced Enzymatic Activity and Intracellular Penetration. Adv. Healthcare Mat., 5, 829-840 (2016).
• Helena Pomares Claudia M Palmeri, Daniel Iglesias-Serret, Cristina Moncunill-Massaguer, José Saura-Esteller, Sonia Núñez-Vázquez, Enric Gamundi, Montserrat Arnan, Sara Preciado, Fernando Albericio, Rodolfo Lavilla, Gabriel Pons, Eva M González-Barca, Ana M Cosialls, Joan Gil. Targeting prohibitins induces apoptosis in acute myeloidleukemia cells. Oncotargets, 7, 64987-65000 (2016).
• Silvia A. Camperi, Silvana L. Giudicessi, María C. Martínez-Ceron, Juan M. Gurevich-Messina, Soledad L. Saavedra, Gerardo Acosta, Osvaldo Cascone, Rosa Erra-Balsells, Fernando Albericio. Combinatorial library screening coupled to mass spectrometry to identify valuable cyclic peptides. Current Protocols, 8, 109-130 (2016).
• Catarina Vizetto-Duarte,Luísa Custódio,Katkam N. Gangadhar,João Henrique G. Lago, Catarina Dias, Ana Marta Matos,Nuno Neng, José Manuel Florêncio Nogueira, Luísa Barreira, Fernando Albericio, Amelia P. Rauter, Joao Varela. Isololiolide, a carotenoid metabolite isolated from the brown alga Cystoseiratamariscifolia, is cytotoxic and able to induce apoptosis in hepatocarcinoma cells through caspase-3 activation, decreased Bcl-2 levels, increased p53 expression and PARP cleavage. Phytomedicine, 23, 550-557 (2016).
• Jyotibon Dutta, Praveen K. Chinthakindi, Per I. Arvidsson, Beatriz G. de la Torre, Hendrik G. Kruger, Thavendran Govender, Tricia Naicker, Fernando Albericio. A facile synthesis of NODASA-Functionalized Peptide. SynLett., 27, 1685-1688 (2016).
• Suhas Ramesh, Thavendran Govender,Hendrik G. Kruger,Fernando Albericio,Beatriz G. de la Torre. An improved and efficient strategy for the total synthesis of a colistin-like peptide. Tetrahedron Lett., 57, 1885-1888(2016).
• Alejandro Gil, Janire Lamariano-Merketeguia, Adriana Lorente, Fernando Albericio, Mercedes Álvarez. Synthesis of (E)-4-Bromo-3-methoxybut-3-en-2-one, the Key Fragment in the Polyhydroxylated Chain Common to Oscillariolide and Phormidolides A-C. Chem., Eur. J., 22, 7033-7035 (2016), with cover.
• Suhas Ramesh, Thavendran Govender,Hendrik G. Kruger,Beatriz G. de la Torre, Fernando Albericio. Short Antimicrobial Peptides (SAMPs) as a Class of Extraordinary Promise Therapeutic Agents. J. Peptide Sci., 22, 438-451 (2016).
• Ayman El-Faham,Saied M. Soliman, Hazem A. Ghabbour, Yasser A. Elnakady, Talal A. Mohaya, Mohammed R. H. Siddiqui, Fernando Albericio. Ultrasonic Promoted Synthesis of Novel 4,6-Disubstituted-s-Triazine- Schiff-Base Derivatives; Molecular Structure, Spectroscopic Studies and Their Preliminary Anti-proliferative Activities. J. Mol. Struc. 1125, 121-135 (2016).
• Georgina Flórez-Grau, Pau Rocas, Raquel Cabezón, Carolina España, Julian Panes, Josep Rocas, Fernando Albericio, Daniel Benítez-Ribas. Nanoencapsulated Budesonide in Self-Stratified Polyurethane-Polyurea Nanoparticles is Highly Effective in Inducing Human Tolerogenic Dendritic Cells. Int. J. Pharm., 511, 785-793 (2016).
• Yahya E. Jad, Beatriz G. de la Torre, Thavendran Govender, Hendrik G. Kruger, Ayman El-Faham, Fernando Albericio. Oxyma-T, a new member of the arsenal of coupling reagents. DOI: 10.1016/j.tetlet.2016.06.109. Tetrahedron Lett., 57, 3523-3525 (2016).
• Shimaa A. H. Abdel Monaim,Yahya E. Jad, Gerardo A. Acosta,Tricia Naicker,Estelle J. Ramchuran,Ayman El-Faham, Thavendran Govender, Hendrik G. Kruger, Beatriz G. de la Torre, Fernando Albericio. Re-Evaluation of the N-Terminal Substitution and the D-Residues of Teixobactin. RSC, Advances, 6, 73827-73829 (2016). Selected for the RSC Advances 10th Anniversary collection focusing on Drug design and discovery, 2021.
• Alejandro Gil, Janire Lamariano-Merketegi, Adriana Lorente, Fernando Albericio, Mercedes Álvarez. Enantioselective Synthesis of the Polyhydroxylated Chain of Oscillariolide and Phormidolides A-C. Org. Lett., 18, 4485-4487 (2016).
• Lorena Mendive-Tapia, Alexandra Bertran, Jesús García,Gerardo Acosta, Fernando Albericio, Rodolfo Lavilla. Constrained Cyclopeptides: Biaryl Formation throughPd-catalyzed C-H Activation in Peptides. Structural Control ofthe Cyclization vs Cyclodimerization Outcome. Chem. Eur. J., 22, 13114-13119 (2016).
• Marta Pelay-Gimeno, Fernando Albericio, Judit Tulla-Puche. Synthesis of Complex Head-to-Side-Chain Cyclodepsipeptides. Nature Protocols, 11, 1924-1947 (2016).
• Patricia Niño, Marta Caba,Nuria Aguilar, Emma Terricabras,Fernando Albericio, Joan-Carles Fernàndez. Efficient Three-Component Synthesis of Diversely Substituted Tetrahydro-1H-Cyclopenta[c]Quinolines. Ind. J. Chem.(Section B, Org. Chem.), 55, 854-881 (2016).
• Patricia Niño, Marta Caba,Nuria Aguilar, Emma Terricabras,Fernando Albericio, Joan-Carles Fernàndez. Povarov Reaction, Scope and Limitations: Preparation of Diversely Heterocyclic-tetrahydro-1H-Cyclopenta[c]Quinolines. Ind. J. Chem. (Section B, Org. Chem.), 55, 1117-1130 (2016).
• Patricia Niño, Marta Caba,Nuria Aguilar, Emma Terricabras,Fernando Albericio, Joan-Carles Fernàndez. Feasibility and Diastereoselectivity of Acid-mediated three-component aza-Diels–Alder reactions. Preparation of Diversely Substituted Hexahydro-2H-Pyrano[3,2-c]Quinolines. Ind. J. Chem.,55, 1384-1399 (2016).
• Suhas Ramesh, Marcelo Grijalva, Alexis Debut, Beatriz G. de la Torre, Fernando Albericio, Luis H. Cumbal. Peptides Conjugated to Silver Nanoparticles in Biomedicine – A “Value-added” Phenomenon. Biomat. Sci. 4, 1713-1725 (2016).
• Yahya E. Jad, Gerardo A. Acosta, Thavendran Govender, Hendrik G. Kruger, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio.Green Solid-Phase Peptide Synthesis-2. 2-Methytetrahydrofuran and ethyl acetate for solid-phase peptide synthesis under green condition. ACS Sust. Chem. Eng., 4, 6809-6814 (2016).
• Omar Luna, Johana Gomez, Constanza Cardenas, Fernando Albericio, Sergio H. Marshall, Fanny Guzman. Deprotection reagents in Fmoc solid phase peptide synthesis: Moving away from piperidine? Molecules, 21, 1542; doi:10.3390/molecules21111542 (2016).
• Shimaa A. H. Abdel Monaim, Yahya E. Jad,Estelle J. Ramchuran, Ayman El-Faham, Thavendran Govender,Hendrik G. Kruger, Beatriz G. de la Torre, Fernando Albericio. Lysine Scanning of Arg10-Teixobactin. Deciphering the Role of Hydrophobic and Hydrophilic Residues. ACS Omega, 1, 1262-1265(2016).
• Ximena Carolina-Pulido, Miriam Royo, Fernando Albericio, Hortensia Rodríguez. Péptidos que atraviesan la membrana celular como potenciales transportadores de fármacos (Cell Penetrating Peptides as potential drug carriers).Bionatura, 1, 208-216 (2016).http://dx.doi.org/10.21931/RB/2016.01.04.9.
• Alejandro Gil, Fernando Albericio, Mercedes Alvarez. Improvements towards the synthesis of phormidolides B and C (Avenços cap a la síntesi de les formidolides B i C).Revista Soc. Cat. Quim. 15, 42-48 (DOI: 10.2436/20.2003.01.73) 2016.
• Prabhakar Cherkupally, Suhas Ramesh, Yahya E. Jad,Thavendran Govender, Hendrik G. Kruger, Beatriz G. de la Torre, Fernando Albericio. Cyclic Peptides as Privileged Structures. In Privileged Scaffolds in Medicinal Chemistry: Design, Synthesis, Evaluation. RSC Drug Discovery Series No. 50. S. Brasse, Ed. Royal Society of Chemistry (London, UK), 2016, pp. 398-438.
• Yahya E. Jad, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Solid-Phase Peptide Synthesis, the State of the Art. Challenges and Opportunities. In Peptide-Based Drug Discovery: Challenges and Opportunities. Discovery Series No. 59. V. Srivastava, Ed. Royal Society of Chemistry (London, UK), 2017, pp. 518 – 550.http://dx.doi.org/10.1039/9781788011532
• Maria Isabel Castellanos, Carlos Mas-Moruno, Anna Grau, Xavier Serra-Picamal, Xavier Trepat, Fernando Albericio, Michael Joner, Francisco Javier Gil, Maria Pau Ginebra, Jose María Manero, Marta Pegueroles. Functionalization of CoCr surfaces with cell adhesive peptides to promote HUVECs adhesion and proliferation. App. Surf. Sci. 393, 82–92 (2017).
• Albert Canals,Raquel Arribas-Bosacoma, Fernando Albericio, Mercedes Álvarez,Joan Aymamí, Miquel Coll. Intercalative DNA binding of the marine anticancer drug Variolin B. Sci. Reports, 7, 39680 | DOI: 10.1038/srep39680 (2017).
• Anaïs F. M. Noisier, Jesús García, Ioana A. Ionut, Fernando Albericio. New hydrocarbon peptide “staple” via late-stage C(sp3)-H activation. Angew. Chem., 56, 314-318 (2017).
• Ifzan Arshad, Javeria Yameen, Aamer Saeed, Jonathan. M White,Fernando Albericio. Synthesis, Crystal Structure, DFT study of m-Methoxy-N'-(3-Methoxybenzoyl)-N-Phenylbenzohydrazide. Crystals, 7, 19; doi:10.3390/cryst7010019 (2017).
• Anamika Sharma, Ivan Ramos-Tomillero, Ayman El-Faham, Ernesto Nicolas, Hortensia Rodriguez, Beatriz G. de la Torre, Fermando Albericio. Understanding 'Thp' as protecting group in peptide chemistry. ChemOpen., 6, 168-177 (2017).
• Anamika Sharma, Ivan Ramos-Tomillero, Ayman El-Faham, Hortensia Rodriguez, Beatriz G. de la Torre., Fernando Albericio. Tetrahydropyranyl: A non aromatic, mild acid labile protecting group for hydroxyl protection in Solid Phase Peptide Synthesis. ChemOpen, 6, 206-210 (2017).
• Anamika Sharma, Yahya E. Jad, Mohammed R. H. Siddiqui, Beatriz G. de la Torre, Fernando Albericio, Ayman El-Faham.Synthesis, Characterization, and Tautomerism of 4,6-Dimethyl- Pyrimidine-2,4,6-Trione Hydrazine Derivatives. J. Chem.,2017, Article ID 5702962 https://doi.org/10.1155/2017/5702962 (2017).
• Ramon Subiros-Funosas, Lorena Mendive-Tapia, Jesus Sot, John D. Pound, Nicole Barth, Yaiza Varela, Felix M. Goñi, Margaret Paterson, Christopher D. Gregory, Fernando Albericio, Ian Dransfield, Rodolfo Lavilla, Marc Vendrell. A Trp-BODIPY cyclic peptide for fluorescence labelling of apoptotic bodies. Chem. Commun., 53, 945-948 (2017).
• Kamil Makowski, Luisa Vigevani, Fernando Albericio, Juan Valcárcel, Mercedes Alvarez. Sudemycin K: a synthetic antitumor splicing inhibitor variant with improved activity and versatile chemistry. ACS Chem. Biol., 12, 163-173 (2017).
• Anamika Sharma,Yahya E. Jad,Hazem A. Ghabbour, Beatriz G. de la Torre, Hendrik G. Kruger, Fernando Albericio,Ayman El-Faham. Synthesis, Crystal Structure and DFT Studies of 1,3-dimethyl-5-propionylpyrimidine-2,4,6(1H,3H,5H)-trione. Crystals, 7, 31; doi:10.3390/cryst7010031 (2017).
• Vida Castro, Christian Noti, Wenqian Chen, Michele Cristau, fAle, Hortensia Rodríguez, Fernando Albericio. Novel Globular Polymeric Supports for Membrane-Enhanced Peptide Synthesis. Macromolecules, 50, 1626-1634 (2017).
• Jan Spengler, Michael Barker, Constanze Schelhorn, Jesus Garcia, Maria J. Macias, Fernando Albericio. Synthesis of a Chelating Peptidomimetic Building Block. Chem. Commun., 53, 2634-2636 (2017).
• Yahya E. Jad, Thavendran Govender, Hendrik G. Kruger, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Green Solid-Phase Peptide Synthesis-3. Green solvents for Fmoc removal in peptide chemistry. Org. Process Res. Dev., 21, 365-369 (2017).
• Lorena Mendive-Tapia, Arantxa Albornoz Grados, Alexandra Bertran,Fernando Albericio, Rodolfo Lavilla. Cross-dehydrogenative couplings on tryptophan-based diketopiperazines: access to new scaffolds. Chem. Commun., 53, 2740-2743 (2017).
• Alessandra Meli, Consiglia Tedesco, Giorgio Della Sala, Rosaria Schettini, Fernando Albericio, Francesco De Riccardis, Irene Izzo. Phakillestatins: an underwater unsolved puzzle. Marine Drugs, 15, 78; doi:10.3390/md15030078 (2017).
• Beatriz G. de la Torre, Fernando Albericio. The Pharmaceutical Industry in 2016. An Analysis of FDA Drug Approvals from a Perspective of the Molecules. Molecules, 22, 368; doi:10.3390/molecules22030368 (2017).
• Lorena Mendive-Tapia,Ramon Subiros-Funosas, Can Zhao, Fernando Albericio, Nick D. Read, Rodolfo Lavilla, Marc Vendrell. Preparation of a Trp-BODIPY fluorogenic amino acid to label peptides for enhanced live-cell fluorescence imaging. Nature Protocols., 12, 1588-1619(2017). doi:10.1038/nprot.2017.048
• Alejandro Gil, Fernando Albericio, Mercedes Álvarez. Role of the Nozaki-Hiyama-Takai-Kishi reaction in the synthesis of natural products.Chem. Rev. 117, 8420-8446 (2017). doi:10.1021/acs.chemrev.7b00144
• Anamika Sharma, Hazem Ghabbour, Shams Tabrez Khan, Beatriz G. de la Torre, Fernando Albericio,Ayman El-Faham.Novel Pyrazolyl-s-Triazine Derivatives, Molecular Structure and Antimicrobial Activity. J. Molecular Struct., 1145, 244-253 (2017). https://doi-org/10.1016/j.molstruc.2017.05.040
• Magdalena Pérez-Ortiz, Claudio Zapata-Urzúa, Gerardo A. Acosta, Alejandro Álvarez-Lueje, Fernando Albericio, Marcelo J. Kogan. Gold Nanoparticles as Efficient Drug Delivery System for GLP-1 Peptides. Colloids Surfaces B, 158, 25-32 (2017). http://dx.doi.org/10.1016/j.colsurfb.2017.06.015
• Gerardo A. Acosta, Miriam Royo, Beatriz G. de la Torre, Fernando Albericio. Facile Solid-Phase Synthesis of Head-Side Chain Cyclothiodepsipetides through a Cyclative Cleavage from MeDbz-resin. Tetrahedron Lett., 58, 2788-2791 (2017). http://dx.doi.org/10.1016/j.tetlet.2017.06.008
• Ashish Kumar, Yahya E. Jad, Ayman El-Faham,Beatriz G. de la Torre, Fernando Albericio. Green Solid-Phase Peptide Synthesis 4. γ-Valerolactone and N-Formylmorpholine as Green Solvents for Solid Phase Peptide Synthesis. Tetrahedron Lett., 58, 2986–2988 (2017).https://doi.org/10.1016/j.tetlet.2017.06.058
• Haroon Mehfooz, Aamer Saeed, Fayaz Larik, Anamika Sharma, Fernando Albericio, Farukh Jabeen, Pervaiz Channar, Ulrich Flörke. Dual inhibition of AChE and BChE with C-5 substituted derivative of Meldrum’s acid; Synthesis, DFT calculations, and Molecular docking studies. Crystals, 7, 211; doi:10.3390/cryst7070211 (2017).
• Ana M Cosialls, Helena Pomares, Daniel Iglesias-Serret, José Saura-Esteller, Sonia Núñez-Vázquez, Diana M. González-Gironès, Esmeralda de la Banda, Sara Preciado, Fernando Albericio, Rodolfo Lavilla, Gabriel Pons, Eva M González-Barca, Joan Gil. The prohibitin-binding compound fluorizoline induces apoptosis in chronic lymphocytic leukemia cells through the upregulation of NOXA and synergizes with ibrutinib, 5-aminoimidazole-4-carboxamideor venetoclax. Haematologica, 102, 1587-1593 (2017). doi:10.3324/haematol.2016.162958
• Jyotibon Dutta, Sooraj Baijnath, Anou Somboro, Savania Nagiah, Fernando Albericio, Beatriz G. de la Torre, Bilijan Marjanovic-painter, Janrijn Zeevaart, Mike Sathekge, Hendrik G. Kruger, Anil Chuturgoon, Tricia Naicker, Thomas Ebenhan, Thavendran Govender. Synthesis, in vitro evaluation and 68Ga-radiolabeling of CDP1 towards PET/CT imaging of bacterial infection. Chem. Biol. Drug Design, 90, 572-579 (2017). DOI: 10.1111/cbdd.12980
• Ashish Kumar, Yahya E. Jad, Beatriz G. de la Torre, Ayman El-Faham,Fernando Albericio. Re-evaluating the stability of COMU in different solvents. J. Pept. Sci.,23, 763-768 (2017). DOI 10.1002/psc.3024
• Fernando Albericio, Gerardo A. Acosta, Ayman El-Faham, Yahya E. Jad, Ashish Kumar, Beatriz G. de la Torre. Green Solid-Phase Peptide Synthesis (GSPPS). Chimia, 71, 523 (2017). DOI: https://doi.org/10.2533/chimia.2017.511
• Shimaa A. H. Abdel Monaim, Estelle J. Ramchuran, Ayman El-Faham,Fernando Albericio, and Beatriz G. de la Torre. Converting Teixobactin into a Cationic AMP. J. Med. Chem., 60, 7476-7482 (2017).DOI: 10.1021/acs.jmedchem.7b00834
• Pervaiz Ali Channar, Aamer Saeed, Fernando Albericio, Fayaz Ali Larik, Qamar Abbas, Mubashir Hassan, Hussain Raza, Sung-Yum Seo. Sulfonamide linked ciprofloxacin derivatives as a novel class of inhibitors of jack bean urease. Synthesis of Kinetic mechanism and Bioinformatics. Molecules 22, 1352; doi:10.3390/molecules22081352 (2017).
• Felix Rueda,Christina Eich, Begoña Cordobilla, Pere Domingo, Gerardo Acosta, Fernando Albericio, Luis J. Cruz, Joan C. Domingo. Effect of TLR ligands co-encapsulated with multiepitopic antigen in nanoliposomes targeted to human Dcs via Fc receptor for cancer vaccines. Immunobiology, 222, 989-997 (2017). http.dx.doi.org/10.1016/j.imbio.2017.06.002
• Shimaa A. H. Abdel Monaim, Sikabwe Noki, Estelle J. Ramchuran, Ayman El-Faham,Fernando Albericio, and Beatriz G. de la Torre. Investigating of the N-terminus amino functional of Arg10-Teixobactin. Molecules, 22, 1632; doi:10.3390/molecules22101632 (2017).
• Carolina Velasco-Aguirre, Francisco Morales-Zavala, Edison Salas, Eduardo Gallardo-Toledo, Oscar Andonie, Luis Muñoz, Ximena Rojas, Eyleen Araya, Gerardo Acosta, Macarena Sanchez-Navarro, Ernest Giralt, Fernando Albericio, Marcelo J. Kogan. Improvement of gold nanorods delivery to the central nervous system by conjugation with the shuttle Angiopep-2. Nanomedicine, 12, 2503-2527 (2017).10.2217/nnm-20170181
• Ashish Kumar,Anamika Sharma,Elvira Haimov, Ayman El-Faham,Beatriz G. de la Torre,Fernando Albericio. Fmoc-Amox, a Suitable Reagent for the Introduction of Fmoc group. Org. Process Res. Dev., 21, 1533-1541(2017).DOI:10.1021/acs.oprd.7b00199
• Suhas Ramesh, Prabhu Cherkupally, Thavender Govender, Henrick G. Kruger, Beatriz G. de la Torre, Fernando Albericio. 21.17 Synthesis of Amides (Including Peptides) in Continuous-Flow Reactors. Science of Synthesis Knowledge Updates 1, 357-379 (2017). DOI 10.1055/sos-SD-121-00033
• Suhas Ramesh, Beatriz G. de la Torre, Fernando Albericio, Hendrik G. Kruger, Thavendran Govender.Microwave-Assisted Synthesis of Antimicrobial Peptides. In Antimicrobial Peptides. Methods in Molecular Biology, Vol. 1548(P.R. Hansen, ed), Springer (New York, USA), 2017, pp. 51-59; DOI: 10.1007/978-1-4939-6737-7_4, 2017.
• Laia Miret-Casals, David Sebastián, José Brea, Eva M. Rico-Leo, Manuel Palacín, Pedro M. Fernández-Salguero, M. Isabel Loza, Fernando Albericio, Antonio Zorzano. Identification of new activators of mitochondrial fusion reveals a link between mitochondrial morphology and pyrimidine metabolism. Cell Chem. Biol., 25, 268-278 (2018). doi.org/10.1016/j.chembiol.2017.12.001.
• Pau Rocas, Yolanda Fernández, Natalia García-Aranda, Laia Foradada, Pilar Calvo, Pablo Avilés, María José Guillén, Simó Schwartz Jr., Josep Rocas, Fernando Albericio, Ibane Abasolo. Improved Pharmacokinetic Profile of Lipophilic Anti-Cancer Drugs Using ανβ3-targeted Polyurethane-Polyurea Nanoparticles.Nanomedicine: Nanotechnology, Biology, and Medicine, 14, 257-267 (2018). doi.org/10.1016/j.nano.2017.10.009.
• Saba Alapour, Beatriz G. de la Torre, Deresh Ramjugernath, Neil A. Koorbanally, Fernando Albericio. Application of Decafluorobiphenyl (DFBP) Moiety as a linker in Bioconjugation. Bioconjugate Chem., 29, 225-233 (2018).10.1021/acs.bioconjchem.7b00800
• Alejandro Gil, Michela Giarrusso, Janire Lamariano, Adriana Lorente-Creville, Fernando Albericio, Mercedes Alvarez. Towards the Synthesis of Phormidolides. ACS Omega, 3, 2351−2362 (2018). 10.1021/acsomega.8b00125.
• Beatriz G. de la Torre, Fernando Albericio. The Pharmaceutical Industry in 2017. An Analysis of FDA Drug Approvals from the Perspective of Molecules.Molecules, 23, 533, (2018).10.3390/molecules23030533
• Pau Rocas, Cristina Cusco, Josep Rocas, Fernando Albericio. On the Importance of Polyurethane and Polyurea Nanomedicines for Future Drug Delivery. Curr. Drug Delivery, 15, 37-43 (2018).
• Iván Ramos-Tomillero, Gema Perez-Chacon,Beatriz Somovilla-Crespo, Francisco Sanchez-Madrid, Juan Manuel Domínguez, Carmen Cuevas, Juan Manuel Zapata, Hortensia Rodríguez, Fernando Albericio. Mesitylene Thiol Alkylation Approach for Antibody Conjugation. Bioconj. Chem., 29, 1199-1208 (2018). 10.1021/acs.bioconjchem.7b00828 (2018).
• Yahya E. Jad,Santosh K. Gudimella, Thavendran Govender,Beatriz G. de la Torre, Fernando Albericio. Solid-Phase Synthesis of Pyrrole Derivatives through a Multi-component Reaction Involving Lys Containing Peptides. ACS Comb. Sci., 20, 187-191 (2018). 10.1021/acscombsci.8b00006
• Claudia Vetterlein, Rodrigo Vasquez, Karen Bolaños, Gerardo Acosta, Fanny Guzman, Fernando Albericio, Freddy Celis, Marcelo Campos, Marcelo J Kogan, Eyleen Araya. Exploring the influence of Diels–Alder linker length on photothermalmolecule release from gold nanorods. Colloids Surf B. Biointerfaces Interf. Sci., 166, 323–329 (2018).doi.org/10.1016/j.colsurfb.2018.03.021
• Shimaa A. H. Abdel Monaim, Gerardo A. Acosta, Miriam Royo, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Solid-phase Synthesis of Homodetic Cyclic Peptides from Fmoc-MeDbz-resin. Tetrahedron Lett., 59, 1779–1782 (2018). doi.org/10.1016/j.tetlet.2018.03.084
• Hosam H. Khalil, Sherine N. Khattab, Adnan A. Bekhit, Mohamed Mokbel Abd El-Rahman, Beatriz G. de la Torre, Ayman El-Faham,Fernando Albericio. 1,3,5-Triazino-Peptide Derivatives: Synthesis, Characterization and their Preliminary Antileishmanial Activities. ChemMedChem, 13, 725-735 (2018).10.1002/cmdc.201700770
• Claudio A. Álvarez, Paula A. Santana, Omar Luna, Constanza Cárdenas, Fernando Albericio, María Soledad Romero, Fanny Guzmán. Chemical Synthesis and Functional Analysis of VarvA Cyclotide. Molecules, 23, 952, (2018).10.3390/molecules23040952
• Claudio A. Álvarez, Andrés Barriga, Fernando Albericio, María SoledadRomero, Fanny Guzmán.Identification of Antimicrobial Peptides in FlowersofSambucus Nigra. Molecules, 23, 1033(2018).doi:10.3390/molecules23051033
• Fanny Guzmán, Monica Aróstica, Claudio A. Álvarez, Claudio Ojeda, Fernando Albericio, Luis F. Aguilar, Sergio H. Marshall, Patricio Carvajal-Rondanelli. Understanding the Antimicrobial Properties/Activity of an 11-residue Lys Homopeptide by Alanine and Proline Scan Amino Acids, Amino Acids, 50, 557-568 (2018).doi.org/10.1007/s00726-018-2542-6
• Juan P. Aguilar, Michal Lipka, Gastón A. Primo, Edxon E. Licon-Bernal, Juan M. Fernández-Pradas, Andriy Yaroshchuk, Fernando Albericio, Alvaro Mata. 3D Electrophoresis-Assisted Lithography (3DEAL): 3D Molecular Printing to Create Functional Patterns and Anisotropic Hydrogels. Adv. Funct. Mat., 28, 1703014 (2018). 10.1002/adfm.201703014
• Othman AlMusaimi,Danah Alshaer,Beatriz G. de la Torre,Fernando Albericio. 2017 FDA Peptide Harvest. Pharmaceuticals, 11, 42 (2018), 10.3390/ph11020042
• Shimaa A. H. Abdel Monaim,Yahya E. Jad, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Teixobactin as a scaffold for unlimited new antimicrobial peptides: SAR study. Bioorg. Med. Chem., 26, 2788-2796 (2018), doi.org/10.1016/j.bmc.2017.09.040
• Ashish Kumar, Yahya Jad, Jonathan M. Collins, Fernando Albericio, Beatriz G. de la Torre. Microwave Assisted Green Solid-Phase Peptide Synthesis using -Valerolactone (GVL) as a Solvent. ACS Sust. Chem. Eng., 6, 8034−8039 (2018), 10.1021/acssuschemeng.8b01531
• Soledad L. Saavedra, Lucía Ávila,Silvana L. Giudicessi, Fernando Albericio, Silvia A. Camperi, Osvaldo Cascone, María Camila Martínez Ceron. Natural snake venom inhibitors and their pharmaceutical uses: possibilities and challenges. Curr. Pharmaceuticals Design, 24, 1737-1747 (2018).
• Estelle J. Ramchuran, Anou M. Somboro, Shimaa A. H. Abdel Monaim, R. Daniel G. Amoako, Raveen Parboosing, Hezekiel M. Kumalo, Nikhil Agrawal, Fernando Albericio, Beatriz G. de la Torre,Linda A. Bester. In vitro evaluation of Teixobactin derivatives against clinically relevant bacterial isolates. Frontiers Microbiol., 9, 1535 (2018), doi: 10.3389/fmicb.2018.01535.
• Risa Takayama, Shun Hayakawa, Hiroshi Hinou, Fernando Albericio, Fayna Garcia-Martin. Further applications of the classical amide coupling reagents: microwave assisted esterification on solid-phase. J. Peptide Sci. e3111(2018). https://doi.org/10.1002/psc.3111.
• Fernando Albericio, Ayman El-Faham. Choosing the Right Peptide Coupling Reagent for Each Reaction A Twenty Five Years Journey. Org Process Res. Dev., 22, 760-772 (2018).
• Othman AlMusaimi, Yahya E. Jad, Ashish Kumar, Jonathan M. Collins, Alessandra Basso, Beatriz G. de la Torre, Fernando Albericio. Investigating Green ethers for the precipitation of peptides after global deprotection in solid-phase peptide synthesis. Curr. Opinion Green Sust. Chem., 11, 99-103 (2018).
• Olivier Ndogo Eteme, Yves Oscar Nganso Ditchou, Ernestine Zondegoumba, Beatriz G. de la Torre, Fernando Albericio, Celine Nkenfou Nguefeu, David Setchaba Kanye, Barthelemy Nyasse. New Derivative of Lophirone A from the Roots of Allexis Batangae (Violaceae) and Evaluation of Antibacterial, Antioxidant and Antiplasmodial Activities. Int. J. Recent Sci. Res.,9, 6(E), 27541-27544 (2018).DOI:http://dx.doi.org/10.24327/ijrsr.2018.0906.2281
• Tanzeela Abdul Fattah, Aamer Saeed, Fernando Albericio. Recent Advances towards Sulfur (VI) Fluoride Exchange (SuFEx) Click Chemistry. J. Fluorine Chem., 213, 87-112 (2018).
• Jan Spengler, Juan Bautista Blanco Canosa, Luciano Forni, Fernando Albericio. One-Pot Peptide Ligation−Oxidative Cyclization Protocol for the Preparation of Short-/Medium-Size Disulfide Cyclopeptides. Org. Lett., 20, 4306−4309 (2018). DOI: 10.1021/acs.orglett.8b01741.
• Shimaa A. H. Abdel Monaim, Jessica T. Mhlongo, Ashish Kumar, Ayman El-Faham, Fernando Albericio, Beatriz G. de la Torre. Formation of Nα-Terminal 2-Dialkyl Amino Oxazoles from Guanidinated Derivatives under Mild Conditions. Org. Biomol. Chem., 16, 5661–5666 (2018).
• Salvatore Bongarzone,Marta Nadal,Zuzanna Kaczmarska, Cristina Machón, Mercedes Álvarez, Fernando Albericio, Miquel Coll. Structure-driven discovery of α,γ-diketoacid inhibitors against UL89 herpesvirus terminase. ACS Omega., 3, 8497-8505 (2018).
• Helena Martin-Gomez, Uwe Linne, Fernando Albericio, Judit Tulla-Puche, Julian D. Hegemann. Investigation of the Biosynthesis of the Lasso Peptide Chaxapeptin Using an E. coli-based Production System. J. Nat. Prod., 81, 2050-2056 (2018).
• Anamika Sharma, Sikabwe Noki,Sizwe J. Zamisa, Heba A. Hazzah, Zainab M. Almarhoon, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Exploiting Thiobarbituric Acid Scaffold for Antibacterial Activity. ChemMedChem., 13, 1923-1930(2018). DOI: 10.1002/cmdc.201800414
• Soledad L. Saavedra, María C. Martínez Ceron, Silvana L. Giudicessi, Guillermina Forno, M. Belen Bosco, Mariela M. Marani, Rosa Erra-Balsells, Fernando Albericio, Osvaldo Cascone, Silvia A. Camperi. Single Step Recombinant Human Growth Hormone (rhGH) Purification from Milk by Peptide Affinity Chromatography. Biotechnol. Progress, 34, 999-1005 (2018). DOI 10.1002/btpr.2645
• Anamika Sharma,Ayman El-Faham,Beatriz G. de la Torre, Fernando AlbericioExploring the OrthogonalChemoselectivity of 2,4,6-Trichloro-1,3,5-triazine (TCT) as a Trifunctional Linker with Different Nucleophiles: Rules of the Game. Frontiers Chem., 6, 516 (2018). doi: 10.3389/fchem.2018.00516
• Anamika Sharma,Ashish Kumar, Shimaa A. H. Abdel Monaim,Yahya E. Jad, Ayman El-Faham,Beatriz G. de la Torre, Fernando Albericio. N-Methylation in amino acids and peptides: Scope and limitations. Biopolymers, 109:e23110 (2018) doi.org/10.1002/bip.23110.
• Rabia Qamar, Aamer Saeed, Maria Saeed, Zaman Ashraf, Qamar Abbas, Mubashir Hassan, Fernando Albericio. Synthesis, carbonic anhydrase inhibitory activity and antioxidant activity of some 1,3-oxazine derivatives. Drug Develop. Res., 79, 352-361 (2018).
• Alvaro Siano, Maria Veronica Humpola, Eliandre de Oliveira, Fernando Albericio, Arturo C. Simonetta, Rafael Lajmanovich, Georgina G. Tonarelli. Leptodactylus latrans Amphibian Skin Secretions as a Novel Source for the Isolation of Antibacterial Peptides. Molecules, 23, 2943 (2018); doi:10.3390/molecules23112943 (2018).
• Saba Alapour, Anamika Sharma, Beatriz G. de la Torre, Deresh Ramjugernath, Neil A. Koorbanally, Fernando Albericio. Perfluorophenyl Derivatives as Unsymmetrical Linkers for Solid Phase Conjugation. Frontiers Chem., 6, 589(2018).doi: 10.3389/fchem.2018.00589
• Judith Palà-Pujadas, Fernando Albericio, Juan Bautista Blanco-Canosa. Peptide ligations using aryloxycarbonyl-o-methylaminoanilides: Chemical synthesis of palmitoylated-Sonic Hedgehog. Angew. Chem., 57, 16120 –16125 (2018).
• Anamika Sharma, Sizwe J. Zamisa, Sikabwe Noki, Zainab M. Almarhoon,Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Crystal structure, spectroscopic studies and theoretical studies of thiobarbituric acid derivatives: understanding the hydrogen-bonding patterns. Acta Crystall. Section C, Struct. Chem., 74, 1703-1714 (2018).
• LaiaMiret-Casals, Aida Baelo, Esther Julián, Josep Astola, Ariadna Lobo-Ruiz, Fernando Albericio, Eduard Torrents. Hydroxylamine derivatives as a new paradigm in the search of antibacterial agents. ACS Omega, 3, 17057-17069 (2018).
• Othman AlMusaimi, Yahya E. Jad, Ashish Kumar, Ayman El-Faham, Jonathan M. Collins, Alessandra Basso, Beatriz G. de la Torre,Fernando Albericio. Greening the Solid-phase Peptide Synthesis Process. 2-MeTHF for the incorporation of First Amino Acid and Precipitation of Peptides after Global Deprotection. Org Process Res. Dev., 22,1809-1816(2018). DOI: 10.1021/acs.oprd.8b00335
• Helena Martin-Gomez, Fernando Albericio, Judit Tulla-Puche. A Lasso-Inspired Bicyclic Peptide: Synthesis, Structure and Properties. Chem., Eur. J., 24, 19250-19257(2018).https://doi.org/10.1002/chem.201803899.
• Soledad L. Saavedra, Gabriela R. Barredo, María C. Martínez-Ceron, Silvana L. Giudicessi, Osvaldo Cascone, Fernando Albericio, Silvia A. Camperi. Design, synthesis and applications of short-peptide and peptidomimetic ligands for affinity chromatography. In Handbook on Protein Purification: Industry Challenges and Technological Developments, N. Labrou, EG. Chronopoulou, F. Ataya. Eds. Nova Science Publishers, Inc. (Hauppauge, NY), pp. 19-50, 2018. ISBN: 978-1-53614-365-2
• Beatriz G. de la Torre, Ashish Kumar, Yahya E. Jad, Ayman El-Faham,Jonathan M. Collins, Simona Serban, Othman Al Musaimi,Fernando Society Albericio. Solid-phase Peptide Synthesis: the Greener, the Better. In Proceedings of the 35th European Peptide Symposium. P.B. Timmons, C.M. Hewage, M. Lebl, Eds. European Peptide -Prompt Scientific Publication. pp. 99-101, 2018.
• Gabriela R. Barredo, Silvana L. Giudicessi, María C. Martínez-Ceron, Soledad L. Saavedra, Gustavo Mahler, Fernando Albericio, Osvaldo Cascone, Silvia A. Camperi. Bevacizumab purification by peptide affinity chromatography. In Proceedings of the 35th European Peptide Symposium. P.B. Timmons, C.M. Hewage, M. Lebl, Eds. European Peptide Society-Prompt Scientific Publication. pp. 130-132, 2018.
• Ashish Kumar, Yahya E. Jad, Ayman El-Faham,Beatriz G. de la Torre, Fernando Albericio. Diethylphosphoryl-OxymaB (DEPO-B) as a Solid Coupling Reagent for Amide Bond Formation. Lett. Org. Chem., 16, 30-33 (2019).10.2174/1570178615666180612074420
• Shimaa A. H. Abdel Monaim, Anou M. Somboro, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Bacteria Hunt Bacteria Through Very Intriguing Cyclic Peptides. ChemMedChem., 14, 24-51 (2019). https://doi.org/10.1002/cmdc.201800597.
• Yahya E. Jad,Ashish Kumar,Ayman El-Faham,Beatriz G. de la Torre, Fernando Albericio. Green Transformation of Solid-Phase Peptide Synthesis.ACS Sust. Chem. Eng., 74, 3671-3683 (2019). DOI: 10.1021/acssuschemeng.8b06520
• Beatriz G. de la Torre, Fernando Albericio. The Pharmaceutical Industry in 2018. An Analysis of FDA Drug Approvals from the Perspective of Molecules.Molecules, 24, 809 (2019),doi: 10.3390/molecules24040809.
• Daniel Carbajo, Peter Fransen,Ayman El-Faham, Miriam Royo,Fernando Albericio. Pseudo-Wang Handle for the Preparation of Fully Protected Peptides. Synthesis of Liraglutide by Fragment Condensation. Org. Lett., 21, 2459-2463 (2019).DOI: 10.1021/acs.orglett.9b00813
• Othman Al Musaimi,Simona Serban, Yahya E. Jad, Zhichao Ma, Ashish Kumar, Cheng Ji, Beatriz G. de la Torre,Alessandra Basso, Fernando Albericio. Jetting Manufacturing of Resins for Solid-Phase Peptide Synthesis. Chem. Today, 37 (1) (January-February), 20-23 (2019).
• Othman Al Musaimi, Simona Serban, Yahya E. Jad, Zhichao Ma, Ashish Kumar, Cheng Ji, Beatriz G. De La Torre, Nathan R. East, Alessandra Basso, Fernando Albericio. New manufacturing process to produce highly uniform resins with excellent performances in Solid Phase Peptide Synthesis. Chem. Today, 37 (2), Monographic special issue: Oligonucleotides & Peptides-February (February-March), 8-10 (2019).
• Muhammad Farooq,Anamika Sharma, Zainab M. Almarhoon, Abudalla Al-Dhfyan, Ayman El-Faham, Nael Abu Taha, Mohammad A.M Wadaan,Beatriz G. de la Torre, Fernando Albericio. Design and synthesis of mono-and di-pyrazolyl-s-triazine derivatives, their anticancer profile in human cancer cell lines, and invivo toxicity studies in zebrafish embryos. Bioorg. Chem., 87,457–464 (2019) https://doi.org/10.1016/j.bioorg.2019.03.063
• Danah Al Shaer, Othman Al Musaimi, Fernando Albericio,Beatriz G. de la Torre. 2018 FDA TIDES Harvest. Pharmaceuticals,12, 52 (2019), doi:10.3390/ph12020052.
• Ashish Kumar, Adewumi Niyi-Thompson, K. P. Nandhini, Jonathan M. Collins, Fernando Albericio,Beatriz G. de la Torre. Troubleshooting of Using GVL in Green Solid-Phase Peptide Synthesis. Org Process Res. Dev., 23, 1096-1100 (2019). https://doi.org/10.1021/acs.oprd.9b00073
• Verónica Hortigüela, Enara Larrañaga, Anna Lagunas, Gerardo A. Acosta, Fernando Albericio, Jordi Andilla, Pablo Loza-Álvarez, Elena Martínez. Large-area biomolecule nanopatterns on diblock copolymer surfaces for cell adhesion studies. Nanomaterials, 9, 579 (2019), doi:10.3390/nano9040579
• Carolina Bruno De Sousa, Marta Oliveira, Jorge Macridachis, Luís Brito, Catarina Vizetto-Duarte, Claudia Florindo, Sarah Hendrickx, Louis Maes, Thiago R. Morais, Miriam Uemi, Luís Neto, Lídia Dionísio, Sofia Cortes, Luísa Barreira, Luísa Custódio, Fernando Albericio, Lenea Campino, João Henrique G. Lago, João Varela. Report of in vitro antileishmanial properties of Iberian Macroalgae. Nat. Prod. Res., 33, 1778-1782 (2109).https://doi-org.sire.ub.edu/10.1080/14786419.2018.1434637
• Anamika Sharma,Zainab M. Almarhoon, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Efficient Route to Synthesize Enamines from Enols. Lett. Org. Chem., 16, 538-540 (2019). 10.2174/1570178616666190409145118
• Daniel Carbajo,Ayman El-Faham, Miriam Royo, Fernando Albericio. Optimized Stepwise Synthesis of the API Liraglutide using BAL-resin and pseudo-prolines. ACS Omega, 4, 8674-8680 (2109). DOI: 10.1021/acsomega.9b00974
• Jael Fernandez, Gerardo Acosta, Daniel Pulido, Marek Malý, José Luis Copa-Patiño, Juan Soliveri de Carranza, Miriam Royo, Rafael Gómez,Fernando Albericio, Paula Ortega, F. Javier de la Mata. Carbosilane Dendrons-Peptides Nanoconjugates as Antimicrobial Agents. Molec. Pharmac., 16, 2661-2674 (2019)
• Othman Al Musaimi,Ayman El-Faham, Zainab Almarhoon, Alessandra Basso, Beatriz G. de la Torre,Fernando Albericio. Bypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentylmethyl Ether (CPME): A Morphological Perspective. Polymers, 11, 874 (2019), doi:10.3390/polym11050874
• Fanny Guzmán, Genezareth Wong, Tanya Román, Constanza Cárdenas, Claudio Alvárez, Paulina Schmitt, Fernando Albericio, Verónica Rojas. Identification of Antimicrobial Peptides from the Microalgae Tetraselmis suecica (Kylin) Butcher and Bactericidal Activity Improvement. Marine Drugs, 2019, 17, 453; doi:10.3390/md17080453.
• Othman Al Musaimi,Ayman El-Faham, Alessandra Basso, Beatriz G. de la Torre,Fernando Albericio. γ-Valerolactone (GVL): An eco-friendly anchoring solvent in solid-phase peptide synthesis. Tetrahedron Lett., 60, 151058 (2019). https://doi.org/10.1016/j.tetlet.2019.151058
• Márió Gajdács, Fernando Albericio. Antibiotic Resistance: From the Bench to Patients. Antibiotics, 8, 129 (2019).doi:10.3390/antibiotics8030129
• Anamika Sharma, Rotimi Sheyi, Ashish Kumar, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Investigating the Triorthogonal Chemoselectivity. Effect of Azide Substitution on the Triazine Core. Org. Lett., 21, 7888-7892 (2019).
• Shaveer Ramkisson, Yahaya E. Jad, Anamika Sharma, Beatriz G. de la Torre, Fernando Albericio. OctaGel Resin - A New PEG-PS-based Solid Support for Solid-Phase Peptide Synthesis. Lett. Org. Chem., 12, 935-940 (2019). DOI: 10.2174/1570178616666190913153605.
• Helena Martin-Gómez, Marta Jorba, Fernando Albericio, Miguel Viñas, Judit Tulla-Puche. Chemical Modification of Microcin J25 Reveals New Insights on the Stereospecific Requirements for Antimicrobial Activity. Int. J. Molecular Sci., 20, 5152 (2019); doi:10.3390/ijms20205152
• Ashish Kumar, Anamika Sharma, Beatriz G. de la Torre, Fernando Albericio. Scope and Limitation of γ-Valerolactone (GVL) as a Green Solvent to be use with Base for the Fmoc removal in SPPS. Molecules, 24, 4004 (2019); doi:10.3390/molecules24214004
• Othman Al Musaimi, Alessandra Basso, Beatriz G. de la Torre, Fernando Albericio. Calculating Resin Functionalization in Solid-Phase Peptide Synthesis Using a Standardized Method based on Fmoc Determination. ACS, Comb. Sci., 21, 717-721 (2019). doi: 10.1021/acscombsci.9b00154
• Sinenhlanhla N. Mthembu, Anamika Sharma, Fernando Albericio, Beatriz G. de la Torre. 2-(Dibenzylamino)butane-1,4-dithiol (DABDT), a Friendly Disulfide Reducing Reagent Compatible with a Broad Range of Solvents. Org. Lett., 21, 10111-10114 (2019). https://doi.org/10.1021/acs.orglett.9b04106
• Gabriela R. Barredo, Silvana L. Giudicessi, María C. Martínez Cerona, Soledad L. Saavedra, Santiago Rodriguez, Lucas Filgueira Risso, Rosa Erra-Balsells, Gustavo Mahler, Fernando Albericio, Osvaldo Casconea, Silvia A. Camperi. A short peptide fragment of the vascular endothelial growth factor as a novel ligand for bevacizumab purification. Protein Expression & Purification, 165, 105500 (2020). https://doi.org/10.1016/j.pep.2019.105500
• Rakia Abd Alhameed, Zainab Almarhoon, Sarah I. Bukhari, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Synthesis and Antimicrobial Activity of a New Series of Thiazolidine-2, 4-diones Carboxamide and Amino acid Derivatives. Molecules, 25, 105 (2020).doi:10.3390/molecules25010105
• Ayman El-Faham, Muhammad Farooq, Zainab Almarhoon, Rakia Abd Alhameed, Mohammad A.M. Wadaan, Beatriz G. de la Torre, Fernando Albericio. Di- and tri-substituted s-triazine derivatives: Synthesis, characterization anticancer activity in human breast-cancer cell lines and developmental toxicity in zebrafish embryos. Bioorg. Chem., 94, 103397 (2020).https://doi.org/10.1016/j.bioorg.2019.103397
• Ayman El-Faham, Anamika Sharma, Muhammad Farooq, Zainab Almarhoon, Rakia Abd Alhameed, Mohammad A.M. Wadaan, Beatriz G. dela Torre, Fernando Albericio. Protocol for synthesis of Di- and tri-substituted s-triazine derivatives.MethodsX, 7, 100825 (2020). https://doi.org/10.1016/j.mex.2020.100825
• Beatriz G. de la Torre, Fernando Albericio. The Pharmaceutical Industry in 2019. An Analysis of FDA Drug Approvals from the Perspective of Molecules. Molecules, 25, 745 (2020)doi:10.3390/molecules25030745.
• Gabriela R. Barredo, Silvana L. Giudicessi, María C. Martínez Ceron, Soledad L. Saavedra, Santiago Rodriguez, Lucas Filgueira Risso, Rosa Erra-Balsells, Gustavo Mahler, Fernando Albericio, Osvaldo Cascone, Silvia A. Camperi. Protocol for bevacizumab purification using Ac-PHQGQHIGVSK-agarose. MethodsX 7,100769 (2020), doi: http://dx.doi.org/10.1016/j.pep.2019.105500
• Danah Al Shaer, Othman Al Musaimi, Fernando Albericio, Beatriz G. de la Torre. 2019 FDA TIDES (Peptides and Oligonucleotides) Harvest. Pharmaceuticals, 13, 40 (2020), doi:10.3390/ph13030040
• Iván Ramos-Tomillero, Gema Perez-Chacon, Beatriz Somovilla-Crespo, Francisco Sánchez-Madrid, Carmen Cuevas, Juan Manuel Zapata, Juan Manuel Domínguez, Hortensia Rodríguez, Fernando Albericio. From Ugi multicomponent reaction to linkers for bioconjugation. ACS Omega, 5, 7424-7431 (2020), https://doi-org.sire.ub.edu/10.1021/acsomega.0c00099
• Pablo Lara, Sujey Palma, Edison Salas, Iva Polakovicova, Simón Guerrero, Lorena Lobos, America Campos, Luis Muñoz, Carla Jorquera, Manuel Varas, Jorge Cancino, Eloisa Arias, Jaime Villegas, Luis J. Cruz, Fernando Albericio, Eyleen Araya, Alejandro Corvalan, Andrew F.G. Quest, Marcelo Kogan. Gold nanoparticle based double-labeling of melanoma extracellular vesicles to determine the specificity of uptake by cells and preferential accumulation in small metastatic lung tumors. J, Nanobiotech., 18, 20 (2020), https://doi.org/10.1186/s12951-020-0573-0 (2020).
• Edgar Cristóbal-Lecina, Daniel Pulido, Pau Martin-Malpartida, Maria Macias, Fernando Albericio, Miriam Royo. Synthesis of Stable Cholesteryl- Polyethylene Glycol-Peptide Conjugates with Non-Disperse PEG Lengths.ACS Omega, 5, 5508-5519 (2020).10.1021/acsomega.0c0013
• Othman Al Musaimi, Beatriz G. de la Torre, Fernando Albericio. Efforts Greening Fmoc/tBu Solid-Phase Peptide synthesis. Green Chem., 22, 996-1018 (2020).https://doi.org/10.1039/C9GC03982A
• M. Ali, Assem Barakat, Ayman El-Faham, Hessa H. Al-Rasheed, Kholoud Dahlous, Abdullah Mohammed Al-Majid, Anamika Sharma, Sammer Yousuf, Mehar Sanam, Zaheer Ul-Haq, M. Iqbal Choudhary, Beatriz G. de la Torre, Fernando Albericio.Synthesis and characterization of thiobarbituric acid enamine derivatives, and evaluation of their α-Glucosidase inhibitory and anti-glycation activity. J. Enzyme Inhib. Med. Chem., 35, 692-701 (2020).DOI: 10.1080/14756366.2020.1737045
• Pedro Jara-Guajardo, Pablo Cabrera, Freddy Celis, Mónica Soler, Isadora Berlanga, Nicole Parra-Munoz, Gerardo Acosta, Fernando Albericio, Fanny Guzman, Marcelo Campos, Alejandra Alvarez, Francisco Morales-Zavala, Marcelo J. Kogan. Gold nanoparticles mediate improved detection of -amyloid aggregates by fluorescence. Nanomaterials, 10, 690 (2020), doi:10.3390/nano10040690
• Othman Al Musaimi, Benjamin D. Summers, Alessandra Basso, Beatriz G. de la Torre, Fernando Albericio, Simona Serban. Efficient Peptide Manufacture as a Combination of Solid Phase Synthesis and Purification. Chem. Today, 38 (2) (March-April), 18-21 (2020).https://www.teknoscienze.com/Contents/Riviste/Sfogliatore/CO2_2020/20/
• Gerardo A. Acosta, Laura Murray, Miriam Royo, Beatriz G. de la Torre, Fernando Albericio. Solid-Phase Synthesis of Side-Chain to Tail Tyr-Cyclodepsipeptides through a Cyclative Cleavage from Fmoc-MeDbz/MeNbz resins. Frontiers Chem., 8:298 (2020); doi: 10.3389/fchem.2020.00298
• Rotimi Sheyi, Anamika Sharma, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Phenol as a Modulator in the Chemical Reactivity of TCT: Rules of the Game II. Aust. J. Chem., 73, 352–356 (2020). https://doi.org/10.1071/CH19524
• Jessica T. Mhlongo, Edikarlos Brazil, Beatriz G. de la Torre, Fernando Albericio. Naturally Occurring Oxazole-Containing Peptides. Marine Drugs, 18, 203 (2020), doi:10.3390/md18040203.
• Natalia L. Cancelarich, Natalia Wilke, Maria L. Fanani, Daniel C. Moreira, Luis O. Perez, Eder Barbosa, Alexandra Plácido, Renato Socodatto, Camila C. Portugal, João B. Relvas, Beatriz G. de la Torre, Fernando Albericio, José R. Leite, Néstor G. Basso, Mariela M. Marani. Somuncorins: A new class of bioactive peptides of the endemic endangered Patagonian frog Pleorodema somuncurense. J. Nat. Prod., 83, 972-984 (2020), ttps://doi.org/10.1021/acs.jnatprod.9b00906.
• Soledad L. Saavedra, Gerardo Acosta, Lucía Ávila, Silvana L. Giudicessi, Silvia A. Camperi, Fernando Albericio, Osvaldo Cascone, María C. Martínez Ceron. Use of a phosphopeptide as a ligand to purify phospholipase A2 from the venom of Crotalus durisuss terrificus by affinity chromatography. J. Chromat. B., 1146, 122070 (2020); https://doi.org/10.1016/j.jchromb.2020.122070
• Mahama Alhassan, Othman Al Musaimi, Jonathan M. Collins, Fernando Albericio, Beatriz G. de la Torre. Cleaving Protected Peptides from 2-ChloroTrityl Chloride Resin. Moving Away from Dichloromethane. Green Chem., 22, 2840-2845 (2020). Doi:10.1039/D0GC00834F.
• Beatriz G. de la Torre, Fernando Albericio. Peptide Therapeutics 2.0. Molecules25, 2293(2020); doi:10.3390/molecules25102293
• Silvia A. Camperi, Gerardo A. Acosta, Gabriela R. Barredo, Lucía C. Iglesias-García, Cleopatra Alves da Silva Caldeira, María C. Martínez-Ceron, Silvana L. Giudicessi, Osvaldo Cascone, Fernando Albericio. Synthetic peptides to produce antivenoms against the Cys-rich toxins of arachnids. Toxicon X , 6, 100038 (2020). https://doi.org/10.1016/j.toxcx.2020.100038
• M. Ali, Assem Barakat, Ayman El-Faham, Abdullah Mohammed Al-Majid, Sammer Yousuf, Sajda Ashraf, Zaheer Ul-Haq, M. Iqbal Choudhary, Beatriz G. de la Torre, Fernando Albericio. Enamine barbiturates and thiobarbiturates as a new class of bacterial urease inhibitors. Applied Sci., 10, 3523 (2020). doi:10.3390/app10103523
• Beatriz G. de la Torre, Ashish Kumar, Mahama Alhassan, Christoph Bucher, Fernando Albericio, John Lopez. Successful Development of a Method for the Incorporation of Fmoc-Arg(Pbf)-OH in Solid-Phase Peptide Synthesis using N Butylpyrrolidinone (NBP) as Solvent. Green Chem., 22, 3162-3169 (2020). doi: 10.1039/C9GC03784E
• Anamika Sharma, Assem Barakat, Hessa H. Al-Rasheed, Abdullah Mohammed Al-Majid, Sammer Yousuf, M. Iqbal Choudhary, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Crystal Structure and Theoretical Investigation of Thiobarbituric Acid Derivatives as Non-Linear Optical (NLO) materials. Crystals, 10, 442 (2020); doi:10.3390/cryst10060442
• Hesaa Al Rasheed, Kholood Dahlous, Anamika Sharma, Essam N. Sholkamy, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Barbiturate and Thiobarbiturate-based s-Triazine hydrazine Derivatives with Promising Anti-proliferative Activity. ACS Omega, 5, 15805-15811 (2020). doi: 10.1021/acsomega.0c00468|
• Mahama Alhassan, Ashish Kumar, John Lopez, Fernando Albericio, Beatriz G. de la Torre. Revising the NO2 as a protecting group of Arginine Side-Chain in Solid-Phase Peptide Synthesis. Int. J. Molecular Sci., 21, 4464 (2020), doi:10.3390/ijms21124464
• Sinenhlanhla N. Mthembu, Anamika Sharma, Fernando Albericio, Beatriz G. de la Torre. Breaking a Couple: Disulfide Reducing Agents. ChemBioChem., 21, 1947-1954 (2020).https://doi.org/10.1002/cbic.202000092
• Lila M. Gierasch, Fernando Albericio, Claudio Toniolo. Dedicated to a peptide chemist of few words and immense impact: Louis A. Carpino. Biopolymers (Peptide Sci.), 112¸ e24185 (2020); doi: 10.1002/pep2.24185
• Ayman El-Faham, Fernando Albericio. Carpino's Protecting Groups, beyond the Boc and the Fmoc. Biopolymers (Peptide Sci.), 112¸ e24164 (2020); doi: 10.1002/pep2.24164
• Songbai Zhang, Vega Lloveras, Daniel Pulido, Flonja Liko, Luiz F. Pinto, Fernando Albericio, Miriam Royo, José Vidal-Gancedo. Radical dendrimers based on biocompatible oligoethylene glycol dendrimers as contrast agents for MRI. Pharmaceutics, 12, 772 (2020); doi:10.3390/pharmaceutics12080772
• Hortensia Rodriguez, Fernando Albericio, Nelson Santiago. Iberoamerican network for the development of therapeutic peptides REDIPEPT (Red Iberoamericana para el desarrollo de péptidos terapéuticos, REDIPEPT). Bionatura, 5, 1177-1180(2020); doi: 10.21931/RB/2020.05.03.1
• Danah Al Shaer, Fernando Albericio, Beatriz G. de la Torre. Solid-Phase Synthesis of Peptides Containing 1-Hydroxypyridine-2-one (1,2-HOPO). Tetrahedron Lett., 61, 152299 (2020), doi: 10.1016/j.tetlet.2020.152299
• Rotimi Sheyi, Anamika Sharma, Ashish Kumar, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio.1,3,5-Triazine as Core for the Preparation of Dendrons. Arkivoc, iii, 64-73 (2020); DOI: 10.24820/ark.5550190.p011.245
• Fanny Guzmán, Adriana Gauna, Omar Luna, Tanya Román, Claudio Álvarez, Fernando Albericio, Constanza Cárdenas. The Tea-Bag Protocol for Comparison of Fmoc Removal Reagents in Solid-Phase Peptide Synthesis. Amino Acids, 52, 1201-1205 (2020); doi: 10.1007/s00726-020-02883-8
• Danah Al Shaer, Othman Al Musaimi, Beatriz G. de la Torre, Fernando Albericio. Hydroxamate Siderophores: natural occurrence, chemical synthesis, iron binding affinity and use as trojan horses against pathogens. Eur. J. Med. Chem., 208, 112791 (2020); doi: 10.1016/j.ejmech.2020.112791
• Othman Al Musaimi, Benjamin D. Summers, Mahama Alhassan, Beatriz G. De La Torre, Fernando Albericio, Simona Serban, Alessandra Basso. Analytical methodologies to assure successful peptide synthesis when utilizing polystyrene/DVB resins. Chem. Today, 38 (5) (September-October), 48-51 (2020). https://www.teknoscienze.com/Contents/Riviste/Sfogliatore/CO5_2020/50/
• Danah Al Shaer, Beatriz G. de la Torre, Fernando Albericio. Protocol for Efficient Solid-Phase Synthesis of Peptides Containing 1-Hydroxypyridine-2-one (1,2-HOPO). MethodsX, 7, 101082 (2020). doi: 10.1016/j.mex.2020.101082
• Ashish Kumar, Mahama Alhassan, John Lopez, Fernando Albericio, Beatriz G. de la Torre. N‐Butylpyrrolidinone for Solid‐Phase Peptide Synthesis is Environmentally Friendlier and Synthetically Better than DMF. ChemSusChem, 13, 5288–5294 (2020); https://doi.org/10.1002/cssc.202001647
• Gloria Colom, J. Pablo Salvador, Gerardo Acosta, Fernando Albericio, Miriam Royo, Pilar Marco. Competitive ELISA for N-terminal pro-brain natriuretic peptide (NT-proBNP) determination in human plasma. Analyst, 145, 6719–6727 (2020).https://doi.org/10.1039/d0an00650e
• Anamika Sharma, Ashish Kumar, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Exploiting azido-dichloro-triazine as a linker for regioselective incorporation of peptides through their N, O, S functional groups. Bioorg. Chem., 104, 104334 (2020). doi: 10.1016/j.bioorg.2020.104334
• Rakia Abd Alhameed, Zainab Almarhoon, Anamika Sharma, Essam N. Sholkamy, Beatriz G. de la Torre, Fernando Albericio, Ayman El-Faham. Novel 4,6-disubstituted s-Triazin-2-yl Amino Acid Derivatives as Promising Antifungal Agents. J. Fungi, 6, 237 (2020), https://doi.org/10.3390/jof6040237
• Diana Imhof, Durba Roy, Fernando Albericio.Editorial: Chemical Design and Biomedical Applications of Disulfide-rich Peptides: Challenges and Opportunities. Frontiers Chem., 8, 586377 (2020), doi: 10.3389/fchem.2020.586377.
• Srinivasa R. Manne, Beatriz G. de la Torre,Ayman El-Faham,Fernando Albericio.OxymaPure Coupling Reagents: Beyond Solid Phase Peptide Synthesis. Synthesis, 52, 3189-3210 (2020), doi: 10.1055/s-0040-1706296
• Mariela Marani, Silvana Aguilar, Ana P. Cuzziol Boccioni, Natalia L. Cancelarich, Néstor G. Basso, Fernando Albericio. Identification of New Ocellatin Antimicrobial Peptides by cDNA Precursors Cloning in the Frame of this Family of Intriguing Peptides. Antibiotics, 9, 751 (2020); doi:10.3390/antibiotics9110751
• Mbuso Faya, Heba A. Hazzah, Calvin A. Omolo, Nikhi Agrawal,Ruma Maji, Pavan Walwaker, Chunderika Mocktar, Bongani Nkambule, Sanjeev Rambharose, Fernando Albericio, Beatriz G. de la Torre, Thirumala Govender. Novel Formulation of Antimicrobial Peptides Enhances Antimicrobial Activity Against Methicillin-resistant Staphylococcus aureus (MRSA). Amino Acids,52, 1439–1457(2020); doi: 10.1007/s00726-020-02903-7
• Amit Chakraborty, Anamika Sharma, Fernando Albericio, Beatriz G. de la Torre. Disulfide Based Protecting Groups for Cysteine Side Chain.Org. Lett., 22, 9644-9647(2020).https://dx.doi.org/10.1021/acs.orglett.0c03705
• Vidya Kaipanchery, Anamika Sharma, Fernando Albericio, Beatriz G. de la Torre. Insights into chemistry of amphibactin-metal interaction (M3+) and its role in antibiotic resistance. Sci. Reports, 10, 21049 (2020). https://doi.org/10.1038/s41598-020-77807-3
• Mona Abdelmoneem, Mahmoud Abd Elwakil, Sherine Khattab, Maged Helmy, Adnan Bekhit, Mohammad Abdulkader, Amira Zaky, Mohamed Teleba, Kadria Elkhodairy, Fernando Albericio, Ahmed Elzoghby. Lactoferrin-Dual Drug Nanoconjugate: Synergistic Anti-Tumor Efficacy of Docetaxel and the NF-κB inhibitor Celastrol. Mat. Sci. Engin. C, 118, 111422 (2021). doi: 10.1016/j.msec.2020.111422
• Iván Ramos-Tomillero, Marisa K. Sánchez, Hortensia Rodríguez, Fernando Albericio. Relation Structure Acid Lability Relationship of N-alkylated-α,α-dialkylglycine obtained via a Ugi Multicomponent Reaction. Molecules, 26, 197 (2021), https://doi.org/10.3390/molecules26010197
• Silvana L. Giudicessi, Soledad L. Saavedra, Alejandra B. Cardillo, Silvia A. Camperi, Osvaldo Cascone, Fernando Albericio, María C. Martínez Ceron. Green solvents in the biotechnology-based pharmaceutical industry. In Green Sustainable Process for Chemical and Environmental Engineering and Science, Inamuddin, R. Boddula, M.I. Ahamed, A.M. Asiri, Eds. Elsevier, USA, 87-104 (2021). https://doi.org/10.1016/B978-0-12-821885-3.00012-8
• Gabriela R. Barredo, Soledad L. Saavedra, Maria C. Martinez-Ceron, Silvana L. Giudicessi, Mariela M. Marani, Fernando Albericio, Osvaldo Cascone, and Silvia A. Camperi. Design of Affinity Chromatography Peptide Ligands Through Combinatorial Peptide Library Screening. In Protein Downstream Processing: Design, Development, and Application of High and Low-Resolution, N. Labrou, Ed., Springer-Nature, Methods, Methods in Molecular Biology, 2178, 217-243 (2021), https://doi.org/10.1007/978-1-0716-0775-6_16.
• Beatriz G. de la Torre, Fernando Albericio. The Pharmaceutical Industry in 2020. An Analysis of FDA Drug Approvals from the Perspective of Molecules. Molecules, 26, 627 (2021). https://doi.org/10.3390/molecules26030627
• Narva Deshwar Kushwaha, Sizwe J. Zamisa, Babita Kushwaha, Anamika Sharma, Francis Kayambaa, Srinivas Reddy Merugu, Ab Majeed Ganai, Vincent A. Obakachi, Fernando Albericio, Rajshekhar Karpoormath. Synthesis, Crystal structure, Spectroscopic and Photophysical studies of novel FluorinatedQuinazoline derivatives. J. Molec. Struc., 1231, 129951 (2021); https://doi.org/10.1016/j.molstruc.2021.129951
• Anamika Sharma, Rotimi Sheyi, Beatriz G. de la Torre, Ayman Al-Faham, Fernando Albericio. s-Triazine: A privileged structure for drug discovery and bioconjugation. Molecules, 26, 864 (2021). https://doi.org/10.3390/molecules26040864
• Othman Al Musaimi, Danah Al Shaer, Fernando Albericio, Beatriz G. de la Torre. 2020 FDA TIDES (Peptides and Oligonucleotides) Harvest. Pharmaceuticals, 14, 145 (2021).https://doi.org/10.3390/ph14020145
• Sonia Núñez-Vázquez, Ismael Sánchez-Vera, José Saura-Esteller, Ana M Cosiall, Anaïs FM Noisier, Fernando Albericio, Rodolfo Lavilla, Gabriel Pons, Daniel Iglesias-Serret, Joan Gil1. NOXA upregulation by the prohibitin-binding compound fluorizoline is transcriptionally regulated by integrated stress response-induced ATF3 and ATF4. FEBS J., 288, 1271-1285 (2021). doi:10.1111/febs.15480
• Azizah M. Malebari, Rakia Abd Alhameed, Zainab Almarhoon, Muhammad Farooq, Mohammad A.M. Wadaan, Anamika Sharma, Beatriz G. de la Torre, Ayman El-Faham, Fernando Albericio. The anti-proliferative and apoptotic effect of novel synthesized s-triazine dipeptide series, and developmental toxicity screening in zebrafish embryos. Molecules, 26, 1170 (2021), https://doi.org/10.3390/molecules26041170
• Osama R. M. Metawea, Mona A. Abdelmoneem, Nesreen Saied Haiba, Hosam H. Khalil, Mohamed Teleb, Ahmed O. Elzoghby, Asmaa F. Khafaga, Ahmed E. Noreldin, Fernando Albericio, Sherine N. Khattab. A novel ‘smart’ PNIPAM-based copolymer for breast cancer targeted therapy; synthesis, and characterization of dual pH/temperature-responsive lactoferrin-targeted PNIPAM-co-AA. Colloids Surfaces B:Biointerfaces., 202, 111694 (2021). https://doi.org/10.1016/j.colsurfb.2021.111694
• Othman Al Musaimi, Richard Wisdom, Peter Talbiersky, Beatriz G. de La Torre, Fernando Albericio. Propylphosphonic anhydride (T3P) as Coupling Reagent for Solid-Phase Peptide Synthesis. ChemistrySelect, 6, 2649-2657 (2021), whith cover. doi.org/10.1002/slct.202100123
• Jet Yeo, Ludmila Peeva, Seoyeon Chung, Piers Gaffney, Daeok Kim, Carla Luciani, Sergey Tsukanov, Kevin Seibert, Michael Kopach, Fernando Albericio, Andrew Livingston. Liquid phase peptide synthesis via one-pot nanostar sieving (PEPSTAR). Angew. Chem., 60, 7786 – 7795 (2021). doi.org/10.1002/anie.202014445
• Zoltan Dekan, Thomas Kremsmayr, Peter Keov, Mathilde Godin, Ngari Teakle, Leopold Dürrauer, Huang Xiang, Dalia Gharib, Christian Bergmayr, Roland Hellinger, Marina Gay, Marta Vilaseca, Dennis Kurzbach, Fernando Albericio, Paul F. Alewood, Christian W. Gruber, Markus Muttenthaler. Nature-inspired dimerization as a strategy to modulate neuropeptide pharmacology exemplified with vasopressin and oxytocin. Chem. Sciences, 12, 4057–4062 (2021). DOI: 10.1039/d0sc05501h
• Othman Al Musaimi, Danah Al Shaer, Beatriz G. de la Torre, Fernando Albericio. Green Circular Economy Applied to Peptide Synthesis. Chem. Today, 39 (2) (March-April) 18-21 (2021). https://www.teknoscienze.com/Contents/Riviste/Sfogliatore/CO2_2021/20/
• Beatriz G. de la Torre, Shaveer Ramkissom, Fernando Albericio, John Lopez. Refractive Index: The Ultimate Tool for Real-Time Monitoring of Solid-Phase Peptide Synthesis. Greening the Process. Org. Proc. Res. Develop., 25, 1047-1053 (2021),with cover https://doi.org/10.1021/acs.oprd.1c00051
• Carlos M. Jiménez-Munoz, Marta López, Fernando Albericio, Kamil Makowski. Targeting energy expenditure. Drugs for obesity treatment. Pharmaceuticals, 14, 435 (2021). https://doi.org/10.3390/ph14050435
• Paula Andrea Santana, Carlos Jara-Gutiérrez, Marco Mellado, Juan Carlos Forero, Andrés Barriga, Fanny Guzmán, Fernando Albericio, Claudio Andrés Álvarez. Dual redox properties of Elderflowers Polyphenol-Enriched Extract in Salmonid Leukocytes. Elect. J. Biotech., 52, 13–20 (2021). https://doi.org/10.1016/j.ejbt.2021.04.004
• Vincent Martin, Sandip Jadhav, Peter H. G. Egelund, Raphael Liffert, Henrik Johansson Castro, Tobias Krüger, Kim F. Haselmann, Sebastian Thordal Le Quement, Fernando Albericio, Frank Dettner, Carolin Lechner, Ralph Schönleber, Daniel Sejer Pedersen. Harnessing polarity and viscosity to identify green binary solvent mixtures as viable alternatives to DMF in solid-phase peptide synthesis. Green Chem., 23, 3295-3311 (2021), with cover DOI: 10.1039/d1gc00603g
• Sandip Jadhav, Vincent Martin, Peter H. G. Egelund, Henrik Johansson Castro, Tobias Krüger, Franziska Richner, Sebastian Thordal Le Quement, Fernando Albericio, Frank Dettner, Carolin Lechner, Ralph Schönleber, Daniel Sejer Pedersen. Replacing DMF in solid-phase peptide synthesis: Varying the composition of green binary solvent mixtures as a tool to mitigate common side-reactions. Green Chem., 23, 3312-3321(2021). DOI: 10.1039/d1gc00604e.
• Estelle J. Ramchuran, Isabel Pérez-Guillén, Linda A. Bester, Rene Khan, Fernando Albericio, Miguel Viñas, Beatriz G. de La Torre. Super-Cationic Peptide Dendrimers. Synthesis and Evaluation as Antimicrobial Agents. Antibiotics,10, 695 (2021). https://doi.org/10.3390/antibiotics10060695.
• Francisco Morales-Zavala, Pedro Jara-Guajardo, David Chamorro, Ana L. Riveros,America Chandia-Cristi, Nicole Salgado, Paola Pismante, Ernest Giralt, Macarena Sanchez, Eyleen Araya-Fuentes, Rodrigo Vazquez, Gerardo Acosta, Fernando Albericio, Alejandra Alvarez R, Marcelo J. Kogan. In vivo micro computed tomography detection and decrease in amyloid load by using multifunctionalized gold nanorods: a neurotheranostic platform for Alzheimer’s disease. Biomater. Sci., 9, 4178–4190 (2021); DOI: 10.1039/d0bm01825b.
• Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Late Advances on Synthesis, Purification, and Characterization of Peptides and their Applications. Appl. Sci. 11, 5593 (2021); https://doi.org/10.3390/app11125593
• Nayara Braga Emidio, Hue N. T. Tran, Asa Andersson, Philip E Dawson, Fernando Albericio, Irina Vetter, Markus Muttenthaler. Improving the gastrointestinal stability of linaclotide. J. Med. Chem., 64, 8384-8390 (2021); https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c00380, with cover.
• Shaveer Ramkisson, Hessa H. Al-Rasheed, Kholood A. Dahlous, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Scope and Limitations of Barbituric and Thiobarbituric Amino Acid Derivatives as Protecting Groups for Solid Phase Peptide Synthesis. Towards to a Green Protecting Group. ChemistrySelect6, 6626-6630 (2021), https://doi.org/10.1002/slct.202101539.
• Margarita Suárez, Kamil Makowski, Reinier Lemos, Luis Almagro, Hortensia Rodríguez, María Ángeles Herranz, Dolores Molero, Orlando Ortiz, Enrique Maroto, Fernando Albericio, Yasujiro Murata, Nazario Martín. An Androsterone-H2@C60 hybrid: Synthesis, Properties and Molecular Docking Simulations with SARS-Cov-2. ChemPlusChem,86, 972–981 (2021); doi.org/10.1002/cplu.202000770; with cover.
• María C. Martínez Ceron, Lucía Ávila, Silvana L. Giudicessi, Juan M. Minoia, Matías Fingermann, Silvia A. Camperi, Fernando Albericio, Osvaldo Cascone. Fully Automated Screening of a Combinatorial Library to Avoid False Positives: Application to Tetanus Toxoid Ligand Identification. ACS Omega, 6, 18756−18762 (2021); https://doi.org/10.1021/acsomega.1c01814
• Nikita Devnarain, Ayman Y. Waddad, Beatriz G. de la Torre, Fernando Albericio, Thirumala Govender. Novel biomimetic human TLR2-derived peptides for potential targeting of lipoteichoic acid: An in-silico assessment. Biomedicines, 9, 1063 (2021). https://doi.org/10.3390/biomedicines9081063.
• Danah Al Shaer, Fernando Albericio, Beatriz G. de la Torre. Synthesis of new peptide-based Ligands with 1,2-HOPO pendant chelators. The thermodynamic evaluation of their iron (III) complexes. ChemistrySelect, 6, 7674-7681 (2021); doi.org/10.1002/slct.202102105
• Fanny Guzmán, Adriana Gauna, Tanya Román, Omar Luna, Claudio Álvarez, Claudia Pareja-Barrueto, Luis Mercado, Fernando Albericio, Constanza Cárdenas. Tea-Bags for Fmoc Solid-Phase Peptide Synthesis, an Example of Circular Economy. Molecules, 26, 5035 (2021); https://doi.org/10.3390/molecules26165035.
• Ashish Kumar, Anamika Sharma, Beatriz G. de la Torre, Fernando Albericio. Rhodiasolv PolarClean – A Greener Alternate in Solid-Phase Peptide Synthesis. Green Chem. Lett. Rev., 14, 544-549 (2021). https://doi.org/10.1080/17518253.2021.1965663
• Rashmi Voleti, Sofia Bali, Jaime Guerrero, Jared Smothers, Charis Springhower, Gerardo A. Acosta, Kyle Brewer, Fernando Albericio, Josep Rizo. Evaluation of the tert-butyl group as a probe for NMR studies of macromolecular complexes. J. Biomol. NMR, 75, 347–363 (2021); https://doi.org/10.1007/s10858-021-00380-y
• Srinivasa R. Manne, Omar Luna, Gerardo A. Acosta, Miriam Royo, Ayman El-Faham, Gyorgy Orosz, Beatriz G. de la Torre, Fernando Albericio. Amide Formation: Choosing the Safer Carbodiimide in Combination with OxymaPure to avoid HCN Release. Org. Lett., 23, 6900−6904(2021); https://doi.org/10.1021/acs.orglett.1c02466
• Clinton G. L. Veale, Maria Mateos-Jimenez, Michaelone C. Vaaltyn, Ronel Muller, Matodzi P. Makhubu, Mahama Alhassan, Beatriz de la Torre, Fernando Albericio, C. Logan MacKay, Adrienne L. Edkinsc, David J. Clarke. A New Native Mass Spectrometry Platform Identifies Inhibitors of the HSP90 – HOP Protein-Protein Interaction. Chem. Commun., 57, 10919–10922 (2021); DOI: 10.1039/d1cc04257b
• Karen Bolaños, Macarena Sánchez-Navarro, Ernest Giralt, Gerardo Acosta, Fernando Albericio, Marcelo J. Kogan, Eyleen Araya. NIR and glutathione trigger the surface release of methotrexate linked by Diels-Alder adducts to anisotropic gold nanoparticles. Mat. Sci. Eng. C, 131, 112512 (2021); https://doi.org/10.1016/j.msec.2021.112512
• R. Manne, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Minimizing Side-Reactions During Srinivasa Amide Formation using DIC and OxymaPure in Solid-Phase Peptide Synthesis. Tetrahedron Lett., 85, 153462 (2021); https://doi.org/10.1016/j.tetlet.2021.153462
• Amit Chakraborty, Fernando Albericio, Beatriz G. de la Torre. Chemoselective Disulfide Formation by Thiol-Disulfide Interchange in SIT-Protected Cysteinyl Peptides. J. Org. Chem., 87, 708-712 (2022).https://doi.org/10.1021/acs.joc.1c02705
• Beatriz G. de la Torre, Fernando Albericio. The Pharmaceutical Industry in 2021. An Analysis of FDA Drug Approvals from the Perspective of Molecules. Molecules, 27, 1075 (2022); https://doi.org/10.3390/molecules27031075
• Srinivasa Rao Manne, Anamika Sharma, Andrius Sazonovas, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. Understanding OxymaPure as Peptide Coupling Additive. A Guide to the New Oxyma Derivatives. ACSOmega, 7, 6007−6023 (2022); https://doi.org/10.1021/acsomega.1c06342
• Rotimi Sheyi, Beatriz G. de la Torre, Fernando Albericio. Linkers: An Assurance for Controlled Delivery of Antibody Drug Conjugates. Pharmaceutics, 14, 396 (2022). https://doi.org/10.3390/pharmaceutics14020396
• Danah Al Shaer, Othman Al Musaimi, Fernando Albericio, Beatriz G. de la Torre. 2021 FDA TIDES (Peptides and Oligonucleotides) Harvest. Pharmaceuticals, 15, 222 (2022). https://doi.org/10.3390/ph15020222
• Enrique-J. Montagut, Gerardo Acosta, Fernando Albericio, Miriam Royo, Gerard Godoy-Tena, Alicia Lacoma, Cristina Prat, J.-Pablo Salvador, M.-Pilar Marco. Direct Quantitative Immunochemical Analysis of the Autoinducer Peptide IV (AIP-IV) for Diagnosing and Stratifying Staphylococcus aureus infections. ACS Infect. Dises., 8, 645−656 (2022). https://doi.org/10.1021/acsinfecdis.1c00670
• Damilola C. Akintayo, Beatriz G. de la Torre, Yongfu Li, Fernando Albericio. Li-Resin – A Fiber Polyacrylamide Resin for Solid-Phase Peptide Synthesis. Polymers, 14, 928 (2022); https://doi.org/10.3390/polym14050928
• Fernando Albericio. Consolidation of Peptides and Oligonucleotides (TIDES) in the Pharmaceutical Arena. Chem. Today, 40 (2), 26-27 (2022).
• Alexis Eras, Danna Castillo, Margarita Suarez, Nelson Santiago Vispo, Fernando Albericio, Hortensia Rodriguez. Chemical Conjugation in Drug Delivery Systems. Frontiers Chem., 10, 889083 (2022); doi: 10.3389/fchem.2022.889083
• Sinenhlanhla N. Mthembu, Amit Chakraborty, Ralph Schönleber, Fernando Albericio, Beatriz G. de la Torre. Solid-Phase Synthesis of C-Terminal Cysteine Peptide Acids. Org. Proc. Res. Develop., 26, 3323−3335 (2022).
• Ashish Kumar, Anamika Sharma, Beatriz G. de la Torre, Fernando Albericio. In-situ Fmoc Removal – A Suistainable Solid-Phase Peptide Synthesis Approach.Green Chem., 24, 4887–4896 (2022); DOI
• Nomfundo Ncobeni, Hendrik G Kruger, Fernando Albericio, Beatriz G. de la Torre, Raveen Parboosing. Active targeting of CD4+ T lymphocytes by PEI-capped, peptide-functionalized gold nanoparticles. Nanotechnology, 33, 405101 (2022).
• Ihab Shawish, Assem Barakat Ali Dalbahi, Aziza M. Malebari, Mohamed S. Nafie, Adnan A. Bekhit, Amgad Albohy, Alamgir Khan, Zaheer Ul-Haq, Matti Haukka, Beatriz G. de la Torre, Fernando Albericio, Ayman . Synthesis and antiproliferative activity of a new series of mono- and bis-(dimethylpyrazolyl)-s-triazine derivatives targeting EGFR/PI3K/AKT/mTOR signaling cascades. ACS Omega, 28, 24858–24870 (2022).
• Juan P. Saucedo, Fernando Gushque, Nelson Santiago Vispo, Jenny Rodriguez, Marco Esteban Gu-diño Gomezjurado, Fernando Albericio, Markus P. Telkamp, Frank Alexis. Marine Arthropods as Source of Antimicrobial Peptides. Marine Drugs, 20, 501 (2022); 10.3390/md20080501.
• Ihab Shawish, Assem Barakat, Ali Dalbahi, Walhan Alshaer, Fadwa Daoud, Dana A. Alqudah, Mazhar Al Zoubi, Ma’mon M. Hatmal, Mohamed S. Nafie, Matti Haukka, Anamika Sharma, Beatriz G. de la Torre, Fernando Albericio, Ayman El-Faham. Acetic acid mediated for one-pot synthesis of novel pyrazolyl s-triazine derivatives for the targeted therapy of triple-negative breast (MDA-MB-231) cancer cells via EGFR/PI3K/AKT/mTOR signaling cascades. Pharmaceutics, 14, 1558 (2022).10.3390/pharmaceutics14081558
• Sisa Chalán-Gualán, Vida Castro, Ruth Oropeza, Margarita Suárez, Fernando Albericio, Hortensia Rodríguez. 3,4-Dihydro-2(1H)-pyridones as building blocks of synthetic relevance. Molecules, 27, 5070 (2022), 10.3390/molecules27165070.
• Anamika Sharma, Ashish Kumar, Beatriz G. de la Torre, Fernando Albericio. Liquid Phase Peptide Synthesis (LPPS), a Third Wave for the Preparation of Peptides. Chem. Rev.,122, 13516−13546 (2022); https://doi.org/10.1021/acs.chemrev.2c00132
• Srinivasa Rao Manne, Amit Chakrovarthy, Karin Rustler, Thomas Bruckdorfer, Beatriz G. de la Torre, Fernando Albericio. Solid-Phase Synthesis of an “Inaccessible” hGH-Derived Peptide Using a Pseudoproline Monomer and SIT-Protection for Cysteine. ACS Omega, 7, 28487−28492 (2022); https://doi.org/10.1021/acsomega.2c03261
• Talia Chetty, Jessica T. Mlongo, Ayman Y. Waddad, Fernando Albericio, Beatriz G. de la Torre. Novel CA(1-7)M(2-9) analogues: Synthesis, characterization and antibacterial evaluation. ACS Med. Chem. Lett., 13, 1370−1377 (2022). https://doi.org/10.1021/acsmedchemlett.2c00270
• K. P. Nandhini, Fernando Albericio, Beatriz G. de la Torre. 2-Methoxy-4-methylsulfinylbenzyl alcohol as a Safety-Catch Linker for the Fmoc/tBu Solid-Phase Peptide Synthesis Strategy. J. Org. Chem., 87, 9433-9442 (2022); https://doi.org/10.1021/acs.joc.2c01057
• Sikabwe Noki, Edikarlos Brazil, Haixiang Zhang, Thomas Bruckdorfer, Beatriz G. de la Torre, Fernando Albericio. Solid-Phase Peptide Synthesis Using a Four-Dimensional (Safety-Catch) Protecting Group Scheme. J. Org. Chem., 87, 9443−9453 (2022); doi.org/10.1021/acs.joc.2c01056
• Da’san M. M. Jaradat, Othman Al Musaimi, Fernando Albericio. Advances in Solid-Phase Peptide Synthesis in Aqueous Media. Green Chem., 24, 6360-6372 (2022); DOI: 10.1039/d2gc02319a.
• Mònica Bravo, Elena Calama, Vicente García-González, Teresa Domènech, Mònica Córdoba, Inés Roger, Julio Cortijo, Miriam Góngora-Benítez, Marta Paradís-Bas, Barry Collins, Andy Davis, Fernando Albericio, Carlos Puig, Mònica Aparici. Pharmacological characterization of novel peptide inhibitor of the Keap1-Nrf2 protein-protein interaction. Biochem. Pharma, Biochemical Pharmacology 204, 115226 (2022); https://doi.org/10.1016/j.bcp.2022.115226.
• Roberto Rojas, Mónica Aróstica, Patricio Carvajal-Rondanelli, Fernando Albericio, Fanny Guzmán, Constanza Cárdenas. Relationship between type II polyproline helix secondary structure and thermal hysteresis activity of short homopeptides. Elect. J. Biotech., 59, 62-73 (2022); https://doi.org/10.1016/j.ejbt.2022.08.003
• Reinier Lemos, Fiorella Ortiz, Luis Almagro, Kamil Makowski, Nazario Martin, Fernando Albericio, Margarita Suárez, Hortensia Rodríguez. Morphological behavior of fullerene-steroid hybrids derivatives. Surf Interface Anal., 54, 1041–1051 (2022). doi/10.1002/sia.7129
• Alexander C. Martins, Mariana Y. Oshiro, Fernando Albericio, Beatriz G. de la Torre, Gustavo José V. Pereira, Rodrigo V. Gonzaga. Trends and Perspectives of Biological Drug Approvals by the FDA: a Review from 2015 to 2021. Biomedicines, 10, 2325 (2022); https://doi.org/10.3390/biomedicines10092325
• Srinivasa Rao Manne, Damilola C. Akintayo, Omar Luna, Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio. tert-Butylethylcarbodiimide as an Efficient Substitute for Diisopropylcarbodiimidein Solid-Phase Peptide Synthesis. Understanding the Side-Reaction of Carbodiimides with OxymaPure. Org. Proc. Res. Develop., 26, 2894–2899 (2022); https://doi.org/10.1021/acs.oprd.2c00220
• Damilola C. Akintayo, Srinivasa Rao Manne, Beatriz G. de la Torre, Yongfu Li, Fernando Albericio. A practical peptide synthetic workflow using Amino-Li-Resin. Methods Protoc., 5, 72 (2022); https://doi.org/10.3390/mps5050072
• Isabel Pérez-Guillén, Òscar Domènech, Adrià Botet-Carreras, Alexandra Merlos, Josep M. Sierra, Fernando Albericio, Beatriz G. de la Torre, M. Teresa Montero, Miguel Viñas, Jordi H. Borrell. Studying Lipid Membrane Interactions of a Super-Cationic Peptide in Model Membranes and Living Bacteria. Pharmaceutics, 14, 2191 (2022). https://doi.org/10.3390/pharmaceutics14102191
• Othman Al Musaimi, Lucia Lombardi, Daryl R. Williams, Fernando Albericio. Strategies for Improving Peptide Stability and Delivery.Pharmaceuticals, 15, 1283 (2022); https://doi.org/10.3390/ph15101283
• 1054.Beatriz G. de la Torre, Fernando Albericio. Practical Protocols for Solid-Phase Peptide Synthesis 4.0. Methods Protoc., 5, 85 (2022); https://doi.org/10.3390/mps5060085
• Ihab Shawish, Mohamed S. Nafie, Assem Barakat, Ali Dalbahi, Hessa H. Al-Rasheed, M. Ali, Walhan Alshaer, Mazhar Al Zoubi, Samha Al Ayoubi, Beatriz G. de la Torre, Fernando Albericio, Ayman El-Faham. Pyrazolo-s-Triazine with Indole Motif as a Novel of Epidermal Growth Factor Receptor/ Cyclin-Dependent Kinase 2 Dual Inhibitors. Frontiers Chem., 10, 1078163. doi: 10.3389/fchem.2022.1078163 (2022).
• Mónica Aróstica, Roberto Rojas, Luis Felipe Aguilar,Patricio Carvajal-Rondanelli, Fernando Albericio, Fanny Guzmán, Constanza Cárdenas. Arginine homopeptide of 11 residues as a model of cell penetrating peptide in the interaction with bacterial membranes. Membranes, 12, 1180 (2022); https://doi.org/10.3390/membranes12121180
• JesicaA. Rodríguez, Gabriela R. Barredo-Vacchelli, Lucia C. Iglesias-García, Gerardo Acosta, Fernando Albericio, Silvia Camperi. Identification and Synthesis of Immunogenic Peptides to Produce Tityus Antivenom. In Proceedings of the 36th European Peptide Symposium, Michal Lebl, Editor, European Peptide Society, pp. 43-44, 2022; https://doi.org/10.17952/36EPS.2022.043
• Lucía C. Iglesias-García, Jésica A. Rodríguez, Gabriela R. Barredo- Vacchelli, Juan M. Minoia, Gerardo Acosta, Fernando Albericio, Silvia A. Camperi. Identification and Synthesis of Epitopes from a Phoneutria Nigriventer Toxin to Produce Immunogens. In Proceedings of the 36th European Peptide Symposium, Michal Lebl, Editor, European Peptide Society, pp. 45-46, 2022;https://doi.org/10.17952/36EPS.2022.045
• Gabriela R. Barredo-Vacchelli, Silvana L. Giudicessi, Fernando Albericio, Osvaldo Cascone, Silvia A. Camperi. Magnetic Affinity Nanoparticles for Bevacizumab Adsorption. In Proceedings of the 36th European Peptide Symposium, Michal Lebl, Editor, European Peptide Society, pp. 127-129, 2022; https://doi.org/10.17952/36EPS.2022.127
• Fernando Albericio. Drug Discovery: a Multifactorial Ecosystem. Explor Drug Sci., 1, 1-5 (2023). https://doi.org/10.37349/eds.2022.00001
• Srinivasa Rao Manne, Karin Rustler, Thomas Bruckdorfer, Beatriz G. de la Torre, Fernando Albericio. Incorporation of Pseudoproline Monomer (Fmoc-Thr[ψMe,Mepro]-OH) Facilitates Efficient Solid Phase Synthesis of Difficult Peptides. Tetrahedron Lett.,115, 154301(2023); https://doi.org/10.1016/j.tetlet.2022.154301
• Beatriz G. de la Torre, Fernando Albericio. The Pharmaceutical Industry in 2022. An Analysis of FDA Drug Approvals from the Perspective of Molecules. Molecules, 28, 1038. (2023); https://doi.org/10.3390/molecules28031038.
• Jésica Ayelén Rodríguez, Gabriela Romina Barredo-Vacchelli, Lucía Candela Iglesias-García, Ariadna María Birocco, Agustín Blachman, Graciela Cristina Calabrese, Gerardo Acosta, Fernando Albericio, Silvia Andrea Camperi. Design and synthesis of peptides from Phoneutria nigriventer δ-ctenitoxin-Pn2a for antivenom production. Inter. J. Peptide Prot. Res. Therap., 29, 25 (2023); https://doi.org/10.1007/s10989-023-10491-9.
• Othman Al Musaimi, Danah Al Shaer, Fernando Albericio, Beatriz G. de la Torre. 2022 FDA TIDES (Peptides and Oligonucleotides) Harvest. Pharmaceuticals,16, 336 (2023); https://doi.org/10.3390/ph16030336
• M. Veronica Humpola, Roque Spinelli, Melina Erben, Virginia Perdomo, Georgina G. Tonarelli, Fernando Albericio, Alvaro S. Siano. D and N-Methyl Amino Acids for Modulating the Therapeutic Properties of Antimicrobial Peptides and Lipopeptides. Antibiotics 12,821 (2023).https://doi.org/10.3390/antibiotics12050821
• K. P. Nandhini, Danah Al Shaer, Fernando Albericio, Beatriz G. de la Torre. Chemical Synthesis of Peptide Nucleic Acids (PNAs). Chem. Soc. Rev., 52, 2764-2789 (2023); DOI: 10.1039/d2cs00049k
• Sisa Chalán-Gualán, Iván Ramos-Tomillero, Thibault Terencio, Lola De Lima, Daniela G. Navas-León, Margarita Suarez, Nelson Santiago Vispo, Fernando Albericio, Hortensia Rodríguez. Cysteine-Based Perfluorinated Derivatives: A Theoretical and Experimental Study. ChemPlusChem, 88,e202300028(2023); doi.org/10.1002/cplu.202300028.
• K. P. Nandhini, Mahama Alhassan, Clinton G. L. Veale, Fernando Albericio, Beatriz G. de la Torre. Troubleshooting Side Reactions Occurring in Methionine Containing Peptides During the Cleavage from Resin. ACS Omega, 8, 15631–15637 (2023); doi.org/10.1021/acsomega.3c01058.
• Hamid Aziz, Aamer Saeed, Jim Simpson, Fernando Albericio, Anwar Ul-Hamid, Hesham R El-Seedi, Mehwish Huma Nasir. New Polymorphs of 1-Benzylidenethiosemicarbazides: Crystal Structure, Hirshfeld Surface Analysis and DFT studies. J. Iran. Chem. Soc., 20,1831–1842 (2023); doi.org/10.1007/s13738-023-02800-2.
• Yomna M. Elmorshedy, Mohamed Teleb, Marwa A. Sallam, Kadria A. Elkhodairy, Mohammed Bahey-El-Din, Doaa A Ghareeb, Shaymaa A Abdulmalek, Shimaa A. H. Abdel Monaim, Adnan A. Bekhit, Ahmed O. Elzoghby. Fernando Albericio, Sherine N. Khattab. Engineered Microencapsulated Lactoferrin Nanoconjugates for OralTargeted Treatment of Colon Cancer. Biomacromolecules, 24,2149-2163 (2023); doi.org/10.1021/acs.biomac.3c00037.
• Alexander C. Martins, Fernando Albericio, Beatriz G. de la Torre. FDA Approvals of Biologics in 2022. Biomedicines11, 1434 (2023). https://doi.org/10.3390/biomedicines11051434
• Fatima Tuz Zahra, Aamer Saeed, Khansa Mumtaz, Fernando Albericio. Tropylium Ion, an Intriguing Moiety in Organic Chemistry. Molecules, 28, 4095 (2023); doi.org/10.3390/molecules28104095
• Fernando Albericio. Peptides and Oligonucleotides, common trends as drugs. Chem. Today, 41(3), 2-5 (2023);
• Fanny Guzmán, Mónica Aróstica, Adriana Gauna, Fernando Albericio, Constanza Cárdenas. Peptides, Solid-Phase Synthesis and Characterization: Tailor-made Methodology. Elect. J. Biotech., 64, 27–33 (2023); https://doi.org/10.1016/j.ejbt.2023.01.005
• Umair Rauf, Ghulam Shabir, Saba Bukhari, Fernando Albericio, Aamer Saeed. Contemporary Developments in Ferrocene Chemistry: Physical, Chemical, Biological and Industrial Aspects. Molecules, 28, 5765 (2023); https://doi.org/10.3390/molecules28155765
• Fatima Tuz Zahra, Aamer Saeed, Atteeque Ahmed, Hammad Ismail, Muhammad Umar Ijaz, Fernando Albericio. Synthesis of Amantadine clubbed N-Aryl amino thiazoles as potent Urease, α-Amylase &αGlucosidase inhibitors, kinetic and molecular docking studies.RSC Advances, 13, 24988–25001 (2023), DOI: 10.1039/d3ra05330j.
• Jessica T. Mlongo, Ayman Y. Waddad, Fernando Albericio, Beatriz G. de la Torre. Antimicrobial Peptide Synergies for Fighting InfectiousDiseases. Adv. Sci.10, 2300472 (2023); 10.1002/advs.202300472.
• Babita Kushwaha, Sinenhlanhla N. Mthembu, Anamika Sharma, Fernando Albericio, Beatriz G. de la Torre. Serinol-Based Versatile Disulfide-Reducing Reagent. Molecules, 28, 5489 (2023); doi.org/10.3390/molecules28145489
• Ghulam Shabir, Aamer Saeed, Wajeeha Zahid, Fatima Naseer, Zainab Riaz, Nafeesa Khalil, Muneeba, Fernando Albericio. Chemistry and Pharmacology of Fluorinated Drugs Approved by FDA (2016-2022). Pharmaceuticals,16, 1162(2023); https://doi.org/10.3390/ph16081162
• Tanya Román, Gerardo Acosta, Beatriz G. de la Torre, Constanza Cárdenas, Fanny Guzmán, Fernando Albericio. Improving 2-Chlorotrityl Chloride (2-CTC) Resin Activation. Methods Protoc., 6, 82 (2023);. https://doi.org/10.3390/mps6050082
• Tanya Román, Gerardo Acosta, Constanza Cárdenas, Beatriz G. de la Torre, Fanny Guzmán, Fernando Albericio. Synthesis of Fmoc-N-Me-AA-OH Using 2-CTC Resin as Temporary and Reusable Protecting Group. Methods Protoc., 6, 110 (2023)/ https://doi.org/ 10.3390/mps6060110.
• K. P. Nandhini, Sikabwe Noki, Edikarlos Brazil, Fernando Albericio, Beatriz G. de la Torre. A Safety-Catch Protecting Group Strategy for Synthesis of Peptide Nucleic Acids (PNA) compatible with Boc-Chemistry. Org. Biomol. Chem., 21, 8125-8135 (2023). DOI: 10.1039/d3ob01348k
• Rafel Prohens, Rafael Barbas, Gerardo Acosta, Beatriz G. de la Torre, Fernando Albericio, Antonio Frontera.An Experimental and Computational Investigation of the elusive anhydrous form of Oxyma-B. CrystEngComm., 25, 5818–5826(2023), DOI: 10.1039/d3ce00741c
• Pedro Jara-Guajardo, Francisco Morales-Zavala, Karen Bolaños, Ernest Giralt, Eyleen Araya, Gerardo Acosta, Fernando Albericio, Alejandra Alvarez, Marcelo J. Kogan. Differential detection of amyloid aggregates in old animals using gold nanorods by computerized tomography: a Pharmacokinetic and bioaccumulation study. Int. J. Nanomedicine, 18, 8169–8185 (2023); I https://doi.org/10.2147/IJN.S435472.
• Sinenhlanhla N. Mthembu, Amit Chakraborty, Ralph Schönleber, Fernando Albericio, Beatriz G. de la Torre. Morpholine, a Strong Contender for Fmoc removal in Solid-Phase Peptide Synthesis. J. Peptide Sci.,30, e3538 (2024); https://doi.org/10.1002/psc.3538
• Amanda Phungula, Ayman Waddad, Marcos Daniel Fernandez Leyes, Paolo Di Gianvincenzo, Bruno Espuche, Sergio Enrique Moya, Fernando Albericio, Beatriz Garcia de la Torre. Self-Assembly of NrTP6 Cell-Penetrating Lipo-Peptide with variable number of lipid chains: impact of phosphate ions on lipid association. J. Colloid & Interf. Sci., 654, 124-133 (2024); https://doi.org/10.1016/j.jcis.2023.09.161
• Beatriz G. de la Torre, Fernando Albericio. The Pharmaceutical Industry in 2023: An Analysis of FDA Drug Approvals from the Perspective of Molecules. Molecules, 29, 585 (2024); doi.org/10.3390/molecules29030585
• Amit Chakraborty, Sinenhlanhla N. Mthembu, Beatriz G. de la Torre, Fernando Albericio. Ready to use Cysteine Thiol Protecting Groups in SPPS, a Practical Overview. Org. Proc. Res. Develop., 28, 26-45 (2024); https://doi.org/10.1021/acs.oprd.3c00425
• Danah Al Shaer, Othman Al Musaimi, Fernando Albericio, Beatriz G. de la Torre. 2023 FDA TIDES (Peptides and Oligonucleotides) Harvest. Pharmaceuticals, 17, 243 (2024). https://doi.org/10.3390/ph17020243.
• James Sherwood, Fernando Albericio, Beatriz G. de la Torre. N,N-Dimethyl formamide (DMF) European Restriction Demands Solvent Substitution in Research and Development. ChemSusChem,17,e202301639(2024); doi.org/10.1002/cssc.202301639.
• Ndumiso Mthethwa, KP. Nandhini, Ashish Kumar, Anamika Sharma, Beatriz G de la Torre, Fernando Albericio. Towards Sustainable Solid Phase Peptide Synthesis Strategy – In situ Fmoc removal. Green Chem. Lett. Rev., 17, 2325993 (2024). DOI: 10.1080/17518253.2024.2325993.
• KP. Nandhini,Nosipho Cele, Beatriz G de la Torre, Fernando Albericio. Triethyl phosphate as a Green Solvent for Solid-Phase Peptide Synthesis (SPPS). Green Chem. Lett. Rev., 17, 2330639 (2024). DOI: 10.1080/17518253.2024.2330639.
• Sikabwe Noki, Beatriz G. de la Torre, Fernando Albericio. Safety-catch Linkers for Solid-Phase Peptide Synthesis. Molecules, 29, 1429 (2024); doi.org/10.3390/molecules29071429
• Alexander C. Martins, Beatriz G. de la Torre, Fernando Albericio. Glucagon-like peptide-1 and glucose-dependent insulinotropic polypeptide agonists for the treatment of obesity and diabetesmellitus. Explor. Drug Sci., 2, 126-143 (2024); https://doi.org/10.37349/eds.2024.00039.
• Farhanah N Sallie, Leandrie Pienaar, Andrea Lubbe, Sanelisiwe P Xhakaza, Srinivasa R Manne, Beatriz G. de la Torre, Fernando Albericio, William MU Daniels, Aletta ME Millen, Sooraj Baijnath. Neurobehavioral changes in a rodent model of ACTH-induced HPA axis dysfunction. Brain Res., 1834 148913 (2024); https://doi.org/10.1016/j.brainres.2024.148913
• Hlobisile Nzama, Srinivasa R Manne, Damilola C. Akintayo, Beatriz G. de la Torre, Fernando Albericio. Ethylthio-1H-tetrazole (ETT) as coupling additive for the solid-phasesynthesis (SPS) of hindered amino acid-containing peptides. Tetrahedron Lett., 142, 155108 (2024); https://doi.org/10.1016/j.tetlet.2024.155108
• Rotimi Sheyi,Jessica T. Mhlongo, Marta Jorba, Ester Fusté, Anamika Sharma, Miguel Viñas, Fernando Albericio, Paula Espinal, Beatriz G. de la Torre. 1,3,5-Triazine as BranchingConnector for the Construction ofNovel Antimicrobial PeptideDendrimers: Synthesis and BiologicalCharacterization. Int. J. Mol. Sci.,25, 5883(2024); https://doi.org/10.3390/ijms25115883
• Kwazi Masuku, Luis M. Menéndez-Mendez, Sikabwe Noki, Beatriz G. de la Torre, Fernando Albericio, Susana Fernández, Miguel Ferrero, Anna Aviñó, Ramon Eritja, Carme Fàbrega. The synthesis of solid supports carrying base labile linkers to generate 3’-phosphateoligonucleotides.Bioorg. Med. Chem. Lett. 109, 129819 (2024).
• Lorena N. Cancelarich, Miriam Arrulo, Sariah Trillo Gugliotti, Eder A. Barbosa, Daniel C. Moreira, Néstor G. Basso, Orlando L. Pérez, Catia Texeira, Paula Gomes, Beatriz G. de la Torre, Fernando Albericio, Peter Eaton, Jose R.A. Leite, Mariela M. Marani Mariela. First bioprospecting study of skin host-defense peptides in Odontoprhynusamericanus (Anura: Odontophrynidae). J. Nat. Prod., 87, 1714−1724 (2024); DOI: 10.1021/acs.jnatprod.4c00184
• Clinton G.L. Veale, Amit Chakraborty, Richwell Mhlanga, Fernando Albericio, Beatriz de la Torre, Adrienne L. Edkins, David J. Clarke. A Native Mass Spectroscopy Approach to Qualitatively Elucidate Interfacial Epitopes of Transient Protein-Protein Interactions. Chem. Comm., 60, 5844–5847 (2024); DOI: 10.1039/d4cc01251h
• Anamika Sharma, Ashish Kumar, Beatriz G. de la Torre, Fernando Albericio. Third Wave for Peptides Synthesis: Liquid Phase Peptide Synthesis (LPPS). In Sustainability in Tides Chemistry: Green Approaches to Oligonucleotides and Oligopeptides Synthesis, L. Ferrazzano,A. Tolomelli, W. Cabri, Eds. Royal Society of Chemistry (London, UK), 2024, pp. 85 – 108; 10.1039/9781837674541-00085; doi.org/10.1039/9781837674541-00085.
• Omar F. Luna, Yomkippur V. Perez, Daniele P. Ferrari, Sana S. Sayedipour, Miriam Royo, Gerardo A. Acosta, Luis J. Cruz, Frauke Alves, Erik Agner, Magne O. Sydnes, Fernando Albericio. Impact of N-terminal PEGylation on Synthesis and Purification of Peptide-based Cancer Epitopes for Pancreatic Ductal Adenocarcinoma (PDAC). ACS Omega., 9, 34544−34554(2024); doi/10.1021/acsomega.4c02604
• Alexander C. Martins, Mariana Y. Oshiro, Fernando Albericio, Beatriz G. de la Torre. Food and Drug Administration (FDA) Approvals of Biologics Drugs in 2023. Biomedicines,12, 1992 (2024); https://doi.org/10.3390/biomedicines12091992
• 1104.Hlobisile Nzama, Srinivas Rao Manne, Oleg Marder, Gyorgy Orosz, Beatriz G. de la Torre, Fernando Albericio..Unveiling the Quaternary Carbodiimide Symphony: Harmonizing Green Chemistry in Peptide Synthesis. Green Chem. Lett. Rev., 17, 2392826 (2024); https://doi.org/10.1080/17518253.2024.2392826
• Amit Chakraborty, Fernando Albericio, Beatriz G. de la Torre. Sec-isoamyl mercaptan (SIT), a Multi-Faceted Disulfide Based Protecting Group for Cysteine Thiol. Int. J. Pep. Res. Ther., 30, 72 (2024). https://doi.org/10.1007/s10989-024-10650-6
• Christiaan A. Gouws, Tricia Naicker, Beatriz G. de la Torre, Fernando Albericio, Janie Duvenhage, Hendrik G. Kruger, Biljana Marjanovic-Painter, Sipho Mdanda, Jan R. Zeevaart, Thomas Ebenhan, Thavendran Govender. 68Ga-Radiolabeling of Nodasa-Functionalized Phage Display-Derived Peptides For Prospective Assessment AsTuberculosis-Specific PET Radiotracers. J. Labelled Comp. Radiopharm., 67, 360-374 (2024); https://doi.org/10.1002/jlcr.4120.
• Constanza Cárdenas, Paula Santana, Claudio Álvarez, Luis Mercado, Sergio Marshall, Fernando Albericio, Fanny Guzmán. Synthetic peptides as valuable and versatile tools for research: Our 20 years journey in Chile. Explor. Drug Sci., 2, 701-718 (2024); https://doi.org/10.37349/eds.2024.00070
• Michael O. Okpara, Michaelone C. Vaaltyn, Jessica L. Watson, Mahama Alhassan, Fernando Albericio, Beatriz G. de la Torre, David J. Clarke, Clinton G. L. Veale, Adrienne L. Edkins. Modulators of the Hop-HSP90 Protein-Protein Interaction Disrupt Early-Stage of KSHV Lytic Replication. ACS Infect. Dis., 10, 3853−3867 (2024); https://doi.org/10.1021/acsinfecdis.4c00429
• Sikabwe Noki, Luana Lastella, Simona Serban, Alessandra Basso, Gyorgy Orosz, Beatriz G de la Torre, Fernando Albericio. Triethyl Phosphate (TEP)-Dimethylsulfoxide (DMSO), as Green Solvent Mixture for Solid-Phase Peptide Synthesis (SPPS), Green Chem. Lett. Rev., 18, 2438068 (2025); https://doi.org/10.1080/17518253.2024.2438068
• Cesar A. Roque-Borda, Laura Maria Duran Gleriani Primo, Kaila Petronila Medina-Alarcón, Isabella Cardeal Campos, Camila De Fátima Nascimento, Mauro M. S. Saraiva, Angelo Berchieri Junior, Ana Marisa Fusco-Almeida, Maria José Soares Mendes-Giannini, Joao Perdigao, Fernando Rogério Pavan, Fernando Albericio. AntimicrobialPeptides: A PromisingAlternativetoConventionalAntimicrobials in CombatPolymicrobialBiofilms. Adv. Sci., 12, 2410893 (2025). DOI: 10.1002/advs.202410893
• Hessa H. Al-Rasheed, Sarah A. Al-Khamis, Assem Barakat, Aliaa A. Masoud, Ahmed A. Sobhy, Doaa A. Gharee, Beatriz G. de la Torre, Fernando Albericio, Ayman El-Faham. Design and synthesis of s-triazine-Isatin hybrids with potent anticancer activity, targeting A549 lung adenocarcinoma via EGF inhibition. Tetrahedron., 171, 134424 (2025), https://doi.org/10.1016/j.tet.2024.134424
• Hessa H. Al-Rasheed, Sizwe J. Zamisa, Ihab Shawish, Assem Barakat,Ayman El-Faham, Beatriz G. de la Torre, Fernando Albericio, Anamika Sharma. Synthesis and structural characterization of s-triazine derivatives and theirphotophysical properties. ResultsChem., 13, 101966 (2025); https://doi.org/10.1016/j.rechem.2024.101966
• Amanda Phugula, Sofia Zuffi, SunisaThongsom, Paolo Di Gianvincenzo,Santiago Gimenez Reyes, Ana Beatriz Caribé dos Santos Valle, FredericoPittella, Fernando Albericio, Beatriz Garcia de la Torre, Sergio Moya. Lauryl-NrTP6 lipopeptide self-assembled nanorods for nuclear target delivery ofdoxorubicin. Nanoscale, 17, 4659-4669 (2025).
• Beatriz G. de la Torre, Fernando Albericio. The Pharmaceutical Industry in 2024: An Analysis of FDA Drug Approvals from the Perspective of Molecules. Molecules,30, 482 (2025). https://doi.org/10.3390/molecules30030482
• Beatriz G. de la Torre, Ndumiso Mthethwa, Srinivas Rao Manne, John Lopez, Fernando Albericio. Looking Inside the SPPS Reactor through a Refractometer: On-line Quantification of the Resin Loading, Org. Proc. Res. Develop., 29, 411-417 (2025), https://doi.org/10.1021/acs.oprd.4c00431.
• Othman Al Musaimi, Danah Al Shaer, Beatriz G. de la Torre, Fernando Albericio. 2024 FDA TIDES (Peptides and Oligonucleotides) Harvest. Pharmaceuticals, 18, 291 (2025)https://doi.org/10.3390/ph18030291.
• Sikabwe Noki, Hossain Saneii, Beatriz G. de la Torre, Fernando Albericio. Base labile safety catch linker. Synthesis and Applications in Solid Phase Peptides Synthesis. Int. J. Molec. Sc. 26, 2210 (2025). https://doi.org/10.3390/ijms26052210
• Amit Chakraborty, Fernando Albericio, Beatriz G. de la Torre .On-Resin Acetamidomethyl (Acm) Removal and Disulfide Formation in Cysteinyl Peptides Using N-Chlorosuccinimide (NCS) in the presence of other Cys protecting groups. Int. J. Molec. Sci., 26, 2523 (2025); https://doi.org/10.3390/ijms26062523
• Kwazi Masuku, Anamika Sharma, Sikabwe Noki, Sizwe Zamisa, Ayman El-Faham, Beatriz G de la Torre, and Fernando Albericio. Synthesis and Structural Confirmation of PyHOPO and its Applicability in Racemization Reduction in Solid-Phase Peptide Synthesis. Tetrahedron Lett., 160, 155520 (2025); https://doi.org/10.1016/j.tetlet.2025.155520
• Daniele P. Ferrari, O. Çobanoglu, Sana S. Sayedipour, Omar F. Luna, Sonia A.N.Ferkel, D. Agorku, Yomkippur Perez, Luis J. Cruz, Fernando Albericio, FrançoisTrottein, Frauke Alves, Frauke, Marietta Andrea Markus, Fernanda Ramos-Gomes. Anti-tumor efficacy of a mesothelin-based nanovaccine in a KPC orthotopic mouse model of pancreatic cancer. Vaccines, 13, 314 (2025); https://doi.org/10.3390/vaccines13030314
• Sinenhlanhla N. Mthembu, Amit Chakraborty, Ralph Schönleber, Fernando Albericio, Beatriz G. de la Torre. Minimizing S-tButylatedCys-Peptide Formation during Final Global Deprotection in Solid-Phase Peptide Synthesis.Org. Proc. Res. Develop., 29, 691-703 (2025);https://doi.org/10.1021/acs.oprd.4c00443.
• Mohadeseh Zare, Laura Colomina Alfaro, Antonella Bandiera, Esra Mutlu, David Grossin, Fernando Albericio, Sarah A. Kuehne, Zubair Ahmed, Artemis Stamboulis. Enzyme-Responsive Coatings Supporting Dual Functionality: OsteoblastPromotion and Antimicrobial Activity for Orthopaedic Implants. ACS, App. Bio. Mat., 8, 2899−2915(2025); https://doi.org/10.1021/acsabm.4c01731.
• Hlobisile Nzama, K.P Nandhini, Karin Rustler, Raimund Maier, Thomas Bruckdorfer, Beatriz G. de la Torre, Fernando Albericio. Investigating the synthesis of dodeca oligomers of Sarcosine using Fmoc-Sar-OH, Fmoc-(Sar)2-OH and Fmoc-(Sar)4-OH. Chem. Today (Chimica Oggi), 43(2), 12-16 (2025).
• Cesar Augusto Roque-Borda, Marco Roberto Chávez-Morán, Laura Maria Duran Gleriani Primo, José C. E. Márquez Montesinos, Vinicius Martinho Borges Cardoso, Mauro MS Saraiva, Caroline Maria Marcos, MarlusChorilli, Fernando Albericio, Beatriz G. de la Torre, Fernando Rogério Pavan, AndréiaBagliottiMenguin. Alginate-pectin microparticles embedding self-assembling antimicrobial peptides and resveratrol for antimicrobial and anti-inflammatory applications. Food Hydrocolloids, 167, 111454 (2025); https://doi.org/10.1016/j.foodhyd.2025.111454
• Mani Kaushal, Ashish Kumar, Hassan Gamal, Sinenhlanhla N. Mthembu, XiaoKang Kou, Beatriz G. de la Torre, Fernando Albericio. Determination of Diketopiperazine Formation during the Solid-Phase Synthesis of C-Terminal Acid Peptides. Chemistry-Methods, 5, e202500035(2025); https://doi.org/10.1002/cmtd.202500035.
• Giovanni Vivenzio, Sikabwe Noki, Amit Chakraborty, John Lopez. Beatriz G de la Torre, Fernando Albericio. Scope and Limitations of the Use of Methanesulfonic Acid (MSA) as a Green Acid for Global Deprotection in Solid-Phase Peptide Synthesis. ChemSusChem, 18, e202402752(2025); doi.org/10.1002/cssc.202402752.
• Christiaan A. Gouws, Tricia Naicker, Janie Duvenhage, Beatriz G. de la Torre, Fernando Albericio, Thavendran Govender. Gallium-68-NODASA-Functionalized D-Lysine Radiosynthesis and first-line in vitro characterization –a potential PET imaging agent for infection. J. South Afric. Chem. Soc., inpress (2025).
• Tanya Román, Paula Santana, Claudio Álvarez, Juan Pablo Cumilla, Fernando Albericio, Fanny Guzmán. In the search for caligidosis treatments: Antimicrobial peptides targeting Caligusrogercresseyi acetylcholinesterase. Pharmaceutics, submitted.
• Pablo Sebastián Espinel, Lilian Spencer, Fernando Albericio, Hortensia Rodríguez. Development and Characterization of Chitosan-Polyvinylpyrrolidone Nanoparticles for Antimicrobial Drug Delivery Applications. Pharmaceutics, submitted.
• Marwaan Rylands,Daniel A. Kusza, David J. Clarke, Beatriz G. de la Torre, Fernando Albericio, Adrienne L. Edkins, Clinton G.L. Veale. STD and WLOGSY NMR Based Fingerprinting Reveals Subtle and Biologically Relevant Differences in SLiM Binding. ChemPhysChem, submitted.
• Somayeh Rezaei, Mark Fonteyne, Luis J. Cruz, Nada Badr, AjinkaManelkar, MahinSaberi, Ronald L.P. van Vlierberghe, Alexander L. Vahrmeijer, Christina Eich, Fernando Albericio, Louise van der Weerd, Peter J.K. Kuppen. Rectal Cancer Molecular Tumor Imaging using Nanoparticles Targeted by a Novel GRPR-binding Peptide for Fluorescence Image-guided Surgery.Biomaterials, submitted.
• Cesar Augusto Roque-Borda, Laura Maria Duran Gleriani Primo, Marco Roberto Chávez Morán, Lavan Sharif, Fernando Albericio, João Perdigão, Fernando Rogério Pavan.Exploiting the Potential of Siderophore-Drug and Siderophore-Peptide Conjugates: A Novel Approach to Combat Carbapenemases-Producing Bacteria. Medicinal Res. Rev., submitted.
• Rotimi Sheyi, Paolo Di Gianvincenzo, Pummarin, Siwanut, Desire Di Silvio, Chanchai Booml, Fernando Albericio, Beatriz G. de la Torre, Sergio E. Moya. Supramolecular assemblies of cationic synthetic Lys and Leu amino acid peptides driven by amine phosphate interactions. Macromol. Chem. Phys., submitted.
• Simón Guerrero, Natalia Hassan, Eyleen Araya, Edison Salas, ItaloMoglia, Roger Prades, Solange Massa, Fernando Albericio, Meritxell Teixido, Ernest Giralt, Elaindre de Oliveira, Marcelo Kogan. Enhancing Brain Drug Delivery: Mimicking Protein Corona with Apolipoprotein E on Peptide-Modified Gold Nanoparticles, submitted.
• Lucia Lombardi, Valentina Del Genio,Fernando Albericio,Daryl R. Williams. Biomimetic Marvels in Drug Design: Unveiling the Synergy of Peptidomimetics and Proteomimetics for Pioneering Next-Generation Therapeutics. Chem. Rev., submitted.
• Cesar Augusto Roque Borda, Qi Zhang, Thi Phuong Truc Nguyen, Thi Thu Hoai Nguyen, HimadriMedhi, HeitorLeocádio de Souza Rodrigues, Christian S. Canales Carnero, Darcy Sutherland, Naiera M. Helmy Mohamed, Prasanna Babu Araveti, Beatriz G. de la Torre, Fernando Albericio, Fernando Rogério Pavan. Synergistic combinations of antimicrobial peptides and conventional antibiotics: a key strategy to extend the resistance timeline against WHO priority bacteria. Pharmacological Rev., submitted.
• Hessa H. Al-Rasheed, Sarah A. Al-Khamis, Assem Barakat, Aliaa A. Masoud, Ahmed A. Sobhy, Maha El Demellawy, Doaa A. Gharee, Anamika Sharma, Beatriz G. de la Torre, Fernando Albericio,Ayman El-Faham. s-Triazine-2-Pyridinecarboxaldehyde Hybrids: Design and Anticancer Efficacy Against A549 Lung Adenocarcinoma via EGF Inhibition. Eur. J. Med. Chem. Reports., submitted.
• Cesar Augusto Roque-Borda, Kaila Petronila Medina-Alarcón, João Paulo Soler Gonçalves Pereira, Thais Cristina dos AnjosSevilhano, Brigitte Aguilar-Morón, Fernando Díaz-Cárdenas, Lucas Silva da Cruz, Francisco Humberto Xavier-Júnior, Eduardo Festozo Vicente, Joao Perdigao, Beatriz G. de la Torre. Fernando Albericio, Fernando Rogério Pavan. RepositioningAntimicrobialPeptidesAgainst WHO-PriorityFungi
• David O. Juma, Sizwe J. Zamisa, Anamika Sharma, Unathi Bongoza, Eric M Njogu.Fernando Albericio, Bernard Omondia. Computational and structural insights into the zwitterionic and neutral forms of N-substituted hydroxyformamidines in the solid state. CrystEngComm., submitted.

• Paul Lloyd-Williams, Fernando Albericio, and Ernest Giralt. Chemical Approaches to the Synthesis of Peptides and Proteins. CRC, Boca Raton (FL, USA), 1997.

• https://orcid.org/0000-0002-8946-0462
• https://www.scopus.com/authid/detail.uri?authorId=7005138070
• https://loop.frontiersin.org/people/520559